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 Enzyme Inhibitor Index

Enzyme Explorer
 
   
TO FIND AN INHIBITOR TO YOUR ENZYME...

1. Search alphabetically for the enzyme to inhibit in the table below
2. You will find the classic inhibitor and its Product Number on the same line
3. Click on the Product # to access product listing and related information including:
Product Information Sheets, C of A and MSDS
 
  A to C
D to K
L to O
P to Q
R to Z
P to Q
Inhibited enzyme Inhibitor Product #
p21ras and other small G proteins (-)-Perillic acid P7083
p38 MAP kinase inhibitor SKF-86002 >99 % (HPLC) S0193
p38 MAP kinase inhibitor SB 239063 >98 % (HPLC) S0569
Papain Antipain hydrochloride A6191
Papain Cystamine dihydrochloride C7255
Papain Chymostatin C7268
Papain Cystatin from chicken egg white C8917
Papain 3,4-Dichloroisocoumarin D7910
Papain E-64 E3132
Papain Ebselen E3520
Papain Gly-Gly-Tyr-Arg G5386
Papain Leupeptin trifluoroacetate salt L2023
Papain a2-Macroglobulin from human plasma M6159
Papain Na-p-Tosyl-L-lysine chloromethyl ketone hydrochloride T7254
PARP Poly(ADP-ribose) Polymerase 3-Aminobenzamide A0788
PARP Poly(ADP-ribose) Polymerase 4-Amino-1,8-naphthalimide A0966
PARP Poly(ADP-ribose) Polymerase 5-Aminoisoquinolinone Hydrochoride A7479
PARP Poly(ADP-ribose) Polymerase DPQ D5314
PARP Poly(ADP-ribose) Polymerase eEB-47 E8405
PARP Poly(ADP-ribose) Polymerase 1,5-Isoquinolinediol I-138
PARP Poly(ADP-ribose) Polymerase 5-Iodo-6-amino-1,2-benzopyrone I2784
PARP Poly(ADP-ribose) Polymerase PJ-34 P4365
PARP Poly(ADP-ribose) Polymerase 6(5H)-Phenanthridinone P8852
PARP Poly(ADP-ribose) Polymerase TIQ-A >98% (HPLC) solid T2825
Penicillinase 3,4-Dichloroisocoumarin D7910
Pepsin Pepstatin A P5318
Pepsin Pepsinostreptin P7424
Pepsin Phenylmethanesulfonyl fluoride P7626
Peptidyl transferase Lycorine hydrochloride L5139
Peroxidase Quercetin dihydrate Q0125
Peroxidase Sodium azide S2002
P-Glycoprotein PGP-4008 P6490
P-Glycoprotein Reversin 121 R1276
P-Glycoprotein Reversin 205 R1401
Phenylalanine ammonia-lyase 4-Hydroxybenzhydrazide H9882
Phosphatase, Alkaline Diethylenetriaminepentaacetic acid D6518
Phosphatase, Alkaline Ethylenediaminetetraacetic acid tripotassium salt dihydrate E0270
Phosphatase, Alkaline Ethylene glycol-bis(2-aminoethylether)-N,N,N',N'-tetraacetic acid E4378
Phosphatase, Alkaline (-)-Tetramisole hydrochloride L9756
Phosphatase, Alkaline 1,10-Phenanthroline monohydrate P9375
Phosphatase, Alkaline Tetramisole hydrochloride T1512
Phosphatidylinositol 3-kinase LY-294,002 hydrochloride L9908
Phosphatidylinositol 3-kinase Wortmannin from Penicillium funiculosum W1628
Phosphodiesterase (PDE III), cGMP-inhibited Trequinsin hydrochloride T2057
Phosphodiesterase 3',5'-Cyclic Nucleotide 4-(3-Butoxy-4-methoxybenzyl)imidazolidin-2-one B8279
Phosphodiesterase 3',5'-Cyclic Nucleotide Calcineurin bovine brain C1907
Phosphodiesterase 3',5'-Cyclic Nucleotide Etazolate hydrochloride E1896
Phosphodiesterase 3',5'-Cyclic Nucleotide Furosemide F4381
Phosphodiesterase 3',5'-Cyclic Nucleotide 8-Methoxymethyl-3-isobutyl-1-methylxanthine M2547
Phosphodiesterase 3',5'-Cyclic Nucleotide Quercetin dihydrate Q0125
Phosphodiesterase 3',5'-Cyclic Nucleotide Phosphoramidon disodium salt R7385
Phosphodiesterase I Diethylenetriaminepentaacetic acid D6518
Phosphodiesterase I Ethylenediaminetetraacetic acid tripotassium salt dihydrate E0270
Phosphodiesterase I Ethylene glycol-bis(2-aminoethylether)-N,N,N',N'-tetraacetic acid E4378
Phosphodiesterase I 1,10-Phenanthroline monohydrate P9375
Phosphodiesterase III Cilostamide C7971
Phosphodiesterase III Quazinone Q3504
Phosphodiesterase III and IV Zardaverine Z3003
Phosphodiesterase IV ICI 63197 >99 % (HPLC) solid I8283
Phosphodiesterase IV Rolipram R6520
Phosphodiesterase IV YM 976 ³99 % (HPLC) solid Y4877
Phosphodiesterase V T-1032 T7692
Phosphodiesterase V T-0156 T8067
Phosphodiesterase 7 BRL50481 B0936
Phosphodiesterase V T-0156 T8067
Phosphodiesterase, c-GMP specific 1-(3-Chlorophenylamino)-4-phenylphthalazine C6085
Phosphogluconic dehydrogenase, 6- Iodoacetamide I1149
Phosphogluconic dehydrogenase, 6- Iodoacetamide I6125
Phosphoinositide-3-Kinase PX-866 P4998
Phospholipases Methyl g-linolenyl fluorophosphonate M2689
Phospholipases Methyl linolenyl fluorophosphonate M2814
Phospholipase A 2 Arachidonyl trifluoromethyl ketone A-231
Phospholipase A 2 Aristolochic acid A5512
Phospholipase A 2 Diethylenetriaminepentaacetic acid D6518
Phospholipase A 2 DL-erythro-Dihydrosphingosine D6908
Phospholipase A 2 7,7-Dimethyl-(5Z,8Z)-eicosadienoic acid D8008
Phospholipase A 2 Flunixin meglumine salt >99 % (HPLC) solid F0429
Phospholipase A 2 Methyl arachidonyl fluorophosphonate M2939
Phospholipase A 2 MJ33 lithium salt M3315
Phospholipase A 2 1,10-Phenanthroline monohydrate P9375
Phospholipase A 2 sPLA2 inhibitor solid >99 % (HPLC) S3319
Phospholipase A 2 U-73122 U6756
Phospholipase A 2 (non-pancreatic) Ro 23-9358 solid >99% (HPLC) R0279
Phospholipase A2, Calcium-dependent Palmityl trifluoromethyl ketone P8727
Phospholipase A2, Secretory Ro 23-9358 solid >99% (HPLC) R0279
Phospholipase C Compound 48/80 C2313
Phospholipase C Diethylenetriaminepentaacetic acid D6518
Phospholipase C Ethylenediaminetetraacetic acid tripotassium salt dihydrate E0270
Phospholipase C Ethylene glycol-bis(2-aminoethylether)-N,N,N',N'-tetraacetic acid E4378
Phospholipase C 1,10-Phenanthroline monohydrate P9375
Phospholipase C U-73122 U6756
Phospholipase C, phosphatidylcholine-specific O-Tricyclo[5.2.1.02,6]dec-9-yl dithiocarbonate potassium salt T8543
Phospholipase C, phosphatidylinositol-specific Sodium iodoacetate I2512
Phospholipase C, phosphatidylinositol-specific Iodoacetic acid I4386
Phospholipase C, phosphatidylinositol-specific Sodium iodoacetate I9148
Phospholipase D Ethylenediaminetetraacetic acid tripotassium salt dihydrate E0270
Phospholipase D Ethylene glycol-bis(2-aminoethylether)-N,N,N',N'-tetraacetic acid E4378
Plasmin Aprotinin from bovine lung A1153
Plasmin 6-Aminohexanoic acid A2504
Plasmin Antipain hydrochloride A6191
Plasmin Antithrombin III from human plasma A2221
Plasmin 6-Aminohexanoic acid A7824
Plasmin 4-(2-Aminoethyl)benzenesulfonyl fluoride hydrochloride A8456
Plasmin Antithrombin III from bovine plasma A9141
Plasmin Bdellin from leeches B3906
Plasmin Esterase inhibitor C-1 from human plasma C2412
Plasmin Diisopropyl fluorophosphate D0879
Plasmin 3,4-Dichloroisocoumarin D7910
Plasmin Esterase inhibitor C-1 from human plasma E0518
Plasmin Elastatinal E0881
Plasmin Gabexate mesylate G2417
Plasmin Leupeptin trifluoroacetate salt L2023
Plasmin a2-Macroglobulin from human plasma M6159
Plasmin Phenylmethanesulfonyl fluoride P7626
Plasmin Urinary Trypsin Inhibitor Fragment U4751
Pro-caspase 3 N-Acetyl-Glu-Ser-Met-Asp-al A1341
Pro-caspase 3 N-Acetyl-Ile-Glu-Thr-Asp-al A1216
Proline dipeptidase Phosphonoacetic acid P6909
Prostaglandin H synthetases 1 (COX-1) and 2 (COX-2) Ketorolac tris salt K1136
Asp-specific proteases 2-Aminobenzoyl-Ala-Phe-Ala-Phe-Asp-Val-Phe-nitro-Tyr-Asp trifluoroacetate salt A9971
Protease (Non-selective serine and cysteine protease inhibitor) a-Boc-Deacetylleupeptin B7530
Protease HIV-1ANT Acetyl-pepstatin A4815
Protease of Bacteroides gingivalis Histatin 5 H6027
Proteases, serine and cysteine Propionyl-leupeptin hemisulfate L3402
Proteasome inhibitor Z-Leu-Leu-Phe-CHO C0358
Proteasome inhibitor Z-Leu-Leu-Leu-B(OH)2 C9857
Proteasome inhibitor Lactacystin L6785
Proteasome inhibitor clasto-Lactacystin b-lactone L7035
Protein kinase A 6-Bnz-cAMP B4560
Protein kinase A H-9 dihydrochloride H-123
Protein kinase A 8-Bromoadenosine-3',5'-cyclic monophosphorothioate, Rp-isomer B2432
Protein kinase A H-89 B1427
Protein kinase A 8-Bromo-2'-monobutyryladenosine-3',5'-cyclic monophosphorothioate, Rp-isomer B2557
Protein kinase A 8-Chloroadenosine-3',5'-cyclic monophosphorothioate, Rp-isomer C0610
Protein kinase A 8-(4-Chlorophenylthio)adenosine-3',5'-cyclic Monophosphorothioate, RP-isomer C0735
Protein kinase A ML-9 C1172
Protein kinase A Chelerythrine chloride C2932
Protein kinase A HA-1004 hydrochloride G1274
Protein kinase A 8-Hexylaminoadenosine-3',5'-monophosphothioate, Rp-isomer H2036
Protein kinase A 8-Hydroxyadenosine-3',5'-monophosphorothioate, Rp-isomer H2161
Protein kinase A HA-100 I1392
Protein kinase A ML-7 I2764
Protein kinase A H-7 I6891
Protein kinase A H-7 dihydrochloride I7016
Protein kinase A KT 5720 K3761
Protein kinase A Myricetin M6760
Protein kinase A N-(2-[Methylamino]ethyl)-5-isoquinolinesulfonamide hydrochloride M9656
Protein kinase A 8-Bromo-b-phenyl-1,N2-ethenoguanosine 3':5'-cyclic monophosphorothioate sodium salt >99 % (HPLC) powder B6684
Protein kinase A Protein Kinase Inhibitor from rabbit P0300
Protein kinase A Protein Kinase Inhibitor porcine heart P0393
Protein kinase A Protein Kinase Inhibitor from rabbit muscle P5015
Protein kinase A Rp-8-PIP-cAMPS P5865
Protein kinase A Protein Kinase Inhibitor from bovine heart P8140
Protein kinase β II CGP53353 C7866
Protein kinase C H-9 dihydrochloride H-123
Protein kinase C GF 109203X hydrochloride B6292
Protein kinase C Bisindolylmaleimide II B3056
Protein kinase C Bisindolylmaleimide III acetate salt B3181
Protein kinase C Bisindolylmaleimide IV B3306
Protein kinase C Bisindolylmaleimide VI B3556
Protein kinase C Bisindolylmaleimide VII B3681
Protein kinase C Bisindolylmaleimide VIII acetate salt B3806
Protein kinase C Bisindolylmaleimide X hydrochoride B3931
Protein kinase C ML-9 C1172
Protein kinase C Chelerythrine chloride C2932
Protein kinase C Calphostin C from Cladosporium cladosporioides C6303
Protein kinase C Dequalinium analog, C-14 Linker D2064
Protein kinase C D-erythro-Dihydrosphingosine D3314
Protein kinase C DL-erythro-Dihydrosphingosine D6908
Protein kinase C rac-2-Ethoxy-3-hexadecanamido-1-propylphosphocholine E3645
Protein kinase C rac-2-Ethoxy-3-octadecanamido-1-propylphosphocholine E3770
Protein kinase C Hexadecyl phosphocholine H6772
Protein kinase C Hypericin H9252
Protein kinase C Hypocrellin A H9410
Protein kinase C HA-100 I1392
Protein kinase C ML-7 I2764
Protein kinase C 1-(5-Isoquinolinesulfonyl)-3-methylpiperazine dihydrochloride I6391
Protein kinase C H-7 dihydrochloride I7016
Protein kinase C Hispidin H5257
Protein kinase C KT 5823 K1388
Protein kinase C Melittin from honey bee venom M2272
Protein kinase C Myricetin M6760
Protein kinase C rac-2-Methoxy-3-hexadecanamido-1-propylphosphocholine M7795
Protein kinase C rac-2-Methoxy-3-octadecanamido-1-propylphosphocholine M8045
Protein kinase C Myristoyl-Phe-Ala-Arg-Lys-Gly-Ala-Leu-Arg-Gln M8814
Protein kinase C Palmitoyl-DL-Carnitine Chloride P4509
Protein kinase C Protein Kinase C Fragment 19-31 Amide P2235
Protein kinase C Protein Kinase C Inhibitor, Myristoylated P3115
Protein kinase C Protein Kinase C Fragment 19-36 P8462
Protein kinase C Rottlerin R5648
Protein kinase C DL-Stearoylcarnitine chloride S2381
Protein kinase C Staurosporine from Streptomyces sp. S4400
Protein kinase C Staurosporine aglycone S3939
Protein kinase C D-Sphingosine S7049
Protein kinase C Na-p-Tosyl-L-lysine chloromethyl ketone hydrochloride T7254
Protein kinase C N,N,N-Trimethylsphingosine chloride T6067
Protein Kinase C beta Hispidin H5257
Protein kinase, DNA dependent 4,5-Dimethoxy-6-nitrobenzaldehyde >99% solid D9192
Protein kinase, DNA dependent 1-(2-Hydroxy-4-morpholin-4-yl-phenyl)ethanone I2159
Protein kinase, DNA dependent NU7026 solid ³99% I2159
Protein kinase, DNA dependent NU7026 solid >99% N1537
Protein kinase erbB2,2 Geldanamycin from Streptomyces hygroscopicus G3381
Protein kinase G I alpha 8-(4-Chlorophenylthio)-guanosine 3',5'-cyclic monophosphorothioate, Rp Isomer triethylammonium salt C-240
Protein kinase G Arg-Lys-Arg-Ala-Arg-Lys-Glu A8186
Protein kinase G HA-1004 hydrochloride G1274
Protein kinase G N-(2-[Methylamino]ethyl)-5-isoquinolinesulfonamide hydrochloride M9656
Protein Kinase, Calmodulin dependent Rottlerin R5648
Protein Kinase II, Calmodulin dependent Autocamtide 2-related inhibitory peptide trifluoroacetate salt A4308
Protein Kinase II, Calmodulin dependent Calmodulin Kinase II Inhibitor from rat C1360
Protein Kinase II, Calmodulin dependent KN-62 I2142
Protein Kinase II, Calmodulin dependent KN-93 K1385
Protein Kinase p38 MAPK SB-200646 hydrochloride >98 % (HPLC) S0568
Protein Kinase p38 MAPK SB 202190 >99 % (HPLC) S7067
Protein kinase v-src Geldanamycin from Streptomyces hygroscopicus G3381
Protein Kinase, cRAF1 GW5074 G6416
Protein kinase, tyrosine Amiloride hydrochloride hydrate A7410
Protein kinase, tyrosine Chelerythrine chloride C2932
Protein kinase, tyrosine Daidzein D7802
Protein kinase, tyrosine Herbimycin A from Streptomyces hygroscopicus H6649
Protein kinase, tyrosine Lavendustin A L2400
Protein kinase, tyrosine Lavendustin C L1289
Protein kinase, tyrosine Quercetin dihydrate Q0125
Protein kinase, tyrosine ST638 solid >99% S5139
Protein kinase, tyrosine ; competitive inhibitor of ATP Genistein G6649
Protein kinase, tyrosine ; competitive inhibitor of ATP Genistein G6776
Protein kinase, tyrosine blocks production of TNF-alpha Tyrphostin AG 126 T9177
Protein kinase, tyrosine blocks production of TNF-alpha Tyrphostin AG 1288 T9302
Protein kinase, tyrosine p56lck Damnacanthal D6309
Protein kinase, tyrosine Syk, p40 and p56 Piceatannol P0453
Protein kinase, tyrosine, EGF receptor Daphnetin D5564
Protein kinase, tyrosine, EGF receptor 2,5-Dihydroxycinnamic acid methyl ester D2667
Protein kinase, tyrosine, EGF receptor Geldanamycin from Streptomyces hygroscopicus G3381
Protein kinase, tyrosine, EGF receptor GW583340 dihydrochloride solid ³97% (HPLC) G3545
Protein kinase, tyrosine, EGF receptor SU 4312 >99 % (HPLC) S8567
Protein kinase, tyrosine, EGF receptor Tyrphostin 1 T7040
Protein kinase, tyrosine, EGF receptor Tyrphostin 23 T7165
Protein kinase, tyrosine, EGF receptor Tyrphostin 25 T7290
Protein kinase, tyrosine, EGF receptor Tyrphostin 46 T7415
Protein kinase, tyrosine, EGF receptor Tyrphostin 47 T7540
Protein kinase, tyrosine, EGF receptor Tyrphostin 51 T7665
Protein kinase, tyrosine, EGF receptor Tyrphostin 63 T7790
Protein kinase, tyrosine, EGF receptor Tyrphostin A9 T-182
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 1007 T5943
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 1024 T6068
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 1112 T6193
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 112 T6943
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 1478 T4182
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 34 T6318
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 494 T4318
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 527 T4443
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 528 T4568
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 537 T4693
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 555 T4818
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 556 T4943
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 658 T5068
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 698 T5193
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 825 T5443
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 835 T5568
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 974 T5818
Protein kinase, tyrosine, EGF receptor Tyrphostin AG 1433 T5317
Protein kinase, tyrosine, EGF receptor SU 5416 >98 % (HPLC)