| P to Q |
| Inhibited enzyme |
Inhibitor |
Product # |
| p21ras and other small G proteins |
(-)-Perillic acid |
P7083 |
| p38 MAP kinase inhibitor |
SKF-86002 >99 % (HPLC) |
S0193 |
| p38 MAP kinase inhibitor |
SB 239063 >98 % (HPLC) |
S0569 |
| Papain |
Antipain hydrochloride |
A6191 |
| Papain |
Cystamine dihydrochloride |
C7255 |
| Papain |
Chymostatin |
C7268 |
| Papain |
Cystatin from chicken egg white |
C8917 |
| Papain |
3,4-Dichloroisocoumarin |
D7910 |
| Papain |
E-64 |
E3132 |
| Papain |
Ebselen |
E3520 |
| Papain |
Gly-Gly-Tyr-Arg |
G5386 |
| Papain |
Leupeptin trifluoroacetate salt |
L2023 |
| Papain |
a2-Macroglobulin from human plasma |
M6159 |
| Papain |
Na-p-Tosyl-L-lysine chloromethyl ketone hydrochloride |
T7254 |
| PARP Poly(ADP-ribose) Polymerase |
3-Aminobenzamide |
A0788 |
| PARP Poly(ADP-ribose) Polymerase |
4-Amino-1,8-naphthalimide |
A0966 |
| PARP Poly(ADP-ribose) Polymerase |
5-Aminoisoquinolinone Hydrochoride |
A7479 |
| PARP Poly(ADP-ribose) Polymerase |
DPQ |
D5314 |
| PARP Poly(ADP-ribose) Polymerase |
eEB-47 |
E8405 |
| PARP Poly(ADP-ribose) Polymerase |
1,5-Isoquinolinediol |
I-138 |
| PARP Poly(ADP-ribose) Polymerase |
5-Iodo-6-amino-1,2-benzopyrone |
I2784 |
| PARP Poly(ADP-ribose) Polymerase |
PJ-34 |
P4365 |
| PARP Poly(ADP-ribose) Polymerase |
6(5H)-Phenanthridinone |
P8852 |
| PARP Poly(ADP-ribose) Polymerase |
TIQ-A >98% (HPLC) solid |
T2825 |
| Penicillinase |
3,4-Dichloroisocoumarin |
D7910 |
| Pepsin |
Pepstatin A |
P5318 |
| Pepsin |
Pepsinostreptin |
P7424 |
| Pepsin |
Phenylmethanesulfonyl fluoride |
P7626 |
| Peptidyl transferase |
Lycorine hydrochloride |
L5139 |
| Peroxidase |
Quercetin dihydrate |
Q0125 |
| Peroxidase |
Sodium azide |
S2002 |
| P-Glycoprotein |
PGP-4008 |
P6490 |
| P-Glycoprotein |
Reversin 121 |
R1276 |
| P-Glycoprotein |
Reversin 205 |
R1401 |
| Phenylalanine ammonia-lyase |
4-Hydroxybenzhydrazide |
H9882 |
| Phosphatase, Alkaline |
Diethylenetriaminepentaacetic acid |
D6518 |
| Phosphatase, Alkaline |
Ethylenediaminetetraacetic acid tripotassium salt dihydrate |
E0270 |
| Phosphatase, Alkaline |
Ethylene glycol-bis(2-aminoethylether)-N,N,N',N'-tetraacetic acid |
E4378 |
| Phosphatase, Alkaline |
(-)-Tetramisole hydrochloride |
L9756 |
| Phosphatase, Alkaline |
1,10-Phenanthroline monohydrate |
P9375 |
| Phosphatase, Alkaline |
Tetramisole hydrochloride |
T1512 |
| Phosphatidylinositol 3-kinase |
LY-294,002 hydrochloride |
L9908 |
| Phosphatidylinositol 3-kinase |
Wortmannin from Penicillium funiculosum |
W1628 |
| Phosphodiesterase (PDE III), cGMP-inhibited |
Trequinsin hydrochloride |
T2057 |
| Phosphodiesterase 3',5'-Cyclic Nucleotide |
4-(3-Butoxy-4-methoxybenzyl)imidazolidin-2-one |
B8279 |
| Phosphodiesterase 3',5'-Cyclic Nucleotide |
Calcineurin bovine brain |
C1907 |
| Phosphodiesterase 3',5'-Cyclic Nucleotide |
Etazolate hydrochloride |
E1896 |
| Phosphodiesterase 3',5'-Cyclic Nucleotide |
Furosemide |
F4381 |
| Phosphodiesterase 3',5'-Cyclic Nucleotide |
8-Methoxymethyl-3-isobutyl-1-methylxanthine |
M2547 |
| Phosphodiesterase 3',5'-Cyclic Nucleotide |
Quercetin dihydrate |
Q0125 |
| Phosphodiesterase 3',5'-Cyclic Nucleotide |
Phosphoramidon disodium salt |
R7385 |
| Phosphodiesterase I |
Diethylenetriaminepentaacetic acid |
D6518 |
| Phosphodiesterase I |
Ethylenediaminetetraacetic acid tripotassium salt dihydrate |
E0270 |
| Phosphodiesterase I |
Ethylene glycol-bis(2-aminoethylether)-N,N,N',N'-tetraacetic acid |
E4378 |
| Phosphodiesterase I |
1,10-Phenanthroline monohydrate |
P9375 |
| Phosphodiesterase III |
Cilostamide |
C7971 |
| Phosphodiesterase III |
Quazinone |
Q3504 |
| Phosphodiesterase III and IV |
Zardaverine |
Z3003 |
| Phosphodiesterase IV |
ICI 63197 >99 % (HPLC) solid |
I8283 |
| Phosphodiesterase IV |
Rolipram |
R6520 |
| Phosphodiesterase IV |
YM 976 ³99 % (HPLC) solid |
Y4877 |
| Phosphodiesterase V |
T-1032 |
T7692 |
| Phosphodiesterase V |
T-0156 |
T8067 |
| Phosphodiesterase 7 |
BRL50481 |
B0936 |
| Phosphodiesterase V |
T-0156 |
T8067 |
| Phosphodiesterase, c-GMP specific |
1-(3-Chlorophenylamino)-4-phenylphthalazine |
C6085 |
| Phosphogluconic dehydrogenase, 6- |
Iodoacetamide |
I1149 |
| Phosphogluconic dehydrogenase, 6- |
Iodoacetamide |
I6125 |
| Phosphoinositide-3-Kinase |
PX-866 |
P4998 |
| Phospholipases |
Methyl g-linolenyl fluorophosphonate |
M2689 |
| Phospholipases |
Methyl linolenyl fluorophosphonate |
M2814 |
| Phospholipase A 2 |
Arachidonyl trifluoromethyl ketone |
A-231 |
| Phospholipase A 2 |
Aristolochic acid |
A5512 |
| Phospholipase A 2 |
Diethylenetriaminepentaacetic acid |
D6518 |
| Phospholipase A 2 |
DL-erythro-Dihydrosphingosine |
D6908 |
| Phospholipase A 2 |
7,7-Dimethyl-(5Z,8Z)-eicosadienoic acid |
D8008 |
| Phospholipase A 2 |
Flunixin meglumine salt >99 % (HPLC) solid |
F0429 |
| Phospholipase A 2 |
Methyl arachidonyl fluorophosphonate |
M2939 |
| Phospholipase A 2 |
MJ33 lithium salt |
M3315 |
| Phospholipase A 2 |
1,10-Phenanthroline monohydrate |
P9375 |
| Phospholipase A 2 |
sPLA2 inhibitor solid >99 % (HPLC) |
S3319 |
| Phospholipase A 2 |
U-73122 |
U6756 |
| Phospholipase A 2 (non-pancreatic) |
Ro 23-9358 solid >99% (HPLC) |
R0279 |
| Phospholipase A2, Calcium-dependent |
Palmityl trifluoromethyl ketone |
P8727 |
| Phospholipase A2, Secretory |
Ro 23-9358 solid >99% (HPLC) |
R0279 |
| Phospholipase C |
Compound 48/80 |
C2313 |
| Phospholipase C |
Diethylenetriaminepentaacetic acid |
D6518 |
| Phospholipase C |
Ethylenediaminetetraacetic acid tripotassium salt dihydrate |
E0270 |
| Phospholipase C |
Ethylene glycol-bis(2-aminoethylether)-N,N,N',N'-tetraacetic acid |
E4378 |
| Phospholipase C |
1,10-Phenanthroline monohydrate |
P9375 |
| Phospholipase C |
U-73122 |
U6756 |
| Phospholipase C, phosphatidylcholine-specific |
O-Tricyclo[5.2.1.02,6]dec-9-yl dithiocarbonate potassium salt |
T8543 |
| Phospholipase C, phosphatidylinositol-specific |
Sodium iodoacetate |
I2512 |
| Phospholipase C, phosphatidylinositol-specific |
Iodoacetic acid |
I4386 |
| Phospholipase C, phosphatidylinositol-specific |
Sodium iodoacetate |
I9148 |
| Phospholipase D |
Ethylenediaminetetraacetic acid tripotassium salt dihydrate |
E0270 |
| Phospholipase D |
Ethylene glycol-bis(2-aminoethylether)-N,N,N',N'-tetraacetic acid |
E4378 |
| Plasmin |
Aprotinin from bovine lung |
A1153 |
| Plasmin |
6-Aminohexanoic acid |
A2504 |
| Plasmin |
Antipain hydrochloride |
A6191 |
| Plasmin |
Antithrombin III from human plasma |
A2221 |
| Plasmin |
6-Aminohexanoic acid |
A7824 |
| Plasmin |
4-(2-Aminoethyl)benzenesulfonyl fluoride hydrochloride |
A8456 |
| Plasmin |
Antithrombin III from bovine plasma |
A9141 |
| Plasmin |
Bdellin from leeches |
B3906 |
| Plasmin |
Esterase inhibitor C-1 from human plasma |
C2412 |
| Plasmin |
Diisopropyl fluorophosphate |
D0879 |
| Plasmin |
3,4-Dichloroisocoumarin |
D7910 |
| Plasmin |
Esterase inhibitor C-1 from human plasma |
E0518 |
| Plasmin |
Elastatinal |
E0881 |
| Plasmin |
Gabexate mesylate |
G2417 |
| Plasmin |
Leupeptin trifluoroacetate salt |
L2023 |
| Plasmin |
a2-Macroglobulin from human plasma |
M6159 |
| Plasmin |
Phenylmethanesulfonyl fluoride |
P7626 |
| Plasmin |
Urinary Trypsin Inhibitor Fragment |
U4751 |
| Pro-caspase 3 |
N-Acetyl-Glu-Ser-Met-Asp-al |
A1341 |
| Pro-caspase 3 |
N-Acetyl-Ile-Glu-Thr-Asp-al |
A1216 |
| Proline dipeptidase |
Phosphonoacetic acid |
P6909 |
| Prostaglandin H synthetases 1 (COX-1) and 2 (COX-2) |
Ketorolac tris salt |
K1136 |
| Asp-specific proteases |
2-Aminobenzoyl-Ala-Phe-Ala-Phe-Asp-Val-Phe-nitro-Tyr-Asp trifluoroacetate salt |
A9971 |
| Protease (Non-selective serine and cysteine protease inhibitor) |
a-Boc-Deacetylleupeptin |
B7530 |
| Protease HIV-1ANT |
Acetyl-pepstatin |
A4815 |
| Protease of Bacteroides gingivalis |
Histatin 5 |
H6027 |
| Proteases, serine and cysteine |
Propionyl-leupeptin hemisulfate |
L3402 |
| Proteasome inhibitor |
Z-Leu-Leu-Phe-CHO |
C0358 |
| Proteasome inhibitor |
Z-Leu-Leu-Leu-B(OH)2 |
C9857 |
| Proteasome inhibitor |
Lactacystin |
L6785 |
| Proteasome inhibitor |
clasto-Lactacystin b-lactone |
L7035 |
| Protein kinase A |
6-Bnz-cAMP |
B4560 |
| Protein kinase A |
H-9 dihydrochloride |
H-123 |
| Protein kinase A |
8-Bromoadenosine-3',5'-cyclic monophosphorothioate, Rp-isomer |
B2432 |
| Protein kinase A |
H-89 |
B1427 |
| Protein kinase A |
8-Bromo-2'-monobutyryladenosine-3',5'-cyclic monophosphorothioate, Rp-isomer |
B2557 |
| Protein kinase A |
8-Chloroadenosine-3',5'-cyclic monophosphorothioate, Rp-isomer |
C0610 |
| Protein kinase A |
8-(4-Chlorophenylthio)adenosine-3',5'-cyclic Monophosphorothioate, RP-isomer |
C0735 |
| Protein kinase A |
ML-9 |
C1172 |
| Protein kinase A |
Chelerythrine chloride |
C2932 |
| Protein kinase A |
HA-1004 hydrochloride |
G1274 |
| Protein kinase A |
8-Hexylaminoadenosine-3',5'-monophosphothioate, Rp-isomer |
H2036 |
| Protein kinase A |
8-Hydroxyadenosine-3',5'-monophosphorothioate, Rp-isomer |
H2161 |
| Protein kinase A |
HA-100 |
I1392 |
| Protein kinase A |
ML-7 |
I2764 |
| Protein kinase A |
H-7 |
I6891 |
| Protein kinase A |
H-7 dihydrochloride |
I7016 |
| Protein kinase A |
KT 5720 |
K3761 |
| Protein kinase A |
Myricetin |
M6760 |
| Protein kinase A |
N-(2-[Methylamino]ethyl)-5-isoquinolinesulfonamide hydrochloride |
M9656 |
| Protein kinase A |
8-Bromo-b-phenyl-1,N2-ethenoguanosine 3':5'-cyclic monophosphorothioate sodium salt >99 % (HPLC) powder |
B6684 |
| Protein kinase A |
Protein Kinase Inhibitor from rabbit |
P0300 |
| Protein kinase A |
Protein Kinase Inhibitor porcine heart |
P0393 |
| Protein kinase A |
Protein Kinase Inhibitor from rabbit muscle |
P5015 |
| Protein kinase A |
Rp-8-PIP-cAMPS |
P5865 |
| Protein kinase A |
Protein Kinase Inhibitor from bovine heart |
P8140 |
| Protein kinase β II |
CGP53353 |
C7866 |
| Protein kinase C |
H-9 dihydrochloride |
H-123 |
| Protein kinase C |
GF 109203X hydrochloride |
B6292 |
| Protein kinase C |
Bisindolylmaleimide II |
B3056 |
| Protein kinase C |
Bisindolylmaleimide III acetate salt |
B3181 |
| Protein kinase C |
Bisindolylmaleimide IV |
B3306 |
| Protein kinase C |
Bisindolylmaleimide VI |
B3556 |
| Protein kinase C |
Bisindolylmaleimide VII |
B3681 |
| Protein kinase C |
Bisindolylmaleimide VIII acetate salt |
B3806 |
| Protein kinase C |
Bisindolylmaleimide X hydrochoride |
B3931 |
| Protein kinase C |
ML-9 |
C1172 |
| Protein kinase C |
Chelerythrine chloride |
C2932 |
| Protein kinase C |
Calphostin C from Cladosporium cladosporioides |
C6303 |
| Protein kinase C |
Dequalinium analog, C-14 Linker |
D2064 |
| Protein kinase C |
D-erythro-Dihydrosphingosine |
D3314 |
| Protein kinase C |
DL-erythro-Dihydrosphingosine |
D6908 |
| Protein kinase C |
rac-2-Ethoxy-3-hexadecanamido-1-propylphosphocholine |
E3645 |
| Protein kinase C |
rac-2-Ethoxy-3-octadecanamido-1-propylphosphocholine |
E3770 |
| Protein kinase C |
Hexadecyl phosphocholine |
H6772 |
| Protein kinase C |
Hypericin |
H9252 |
| Protein kinase C |
Hypocrellin A |
H9410 |
| Protein kinase C |
HA-100 |
I1392 |
| Protein kinase C |
ML-7 |
I2764 |
| Protein kinase C |
1-(5-Isoquinolinesulfonyl)-3-methylpiperazine dihydrochloride |
I6391 |
| Protein kinase C |
H-7 dihydrochloride |
I7016 |
| Protein kinase C |
Hispidin |
H5257 |
| Protein kinase C |
KT 5823 |
K1388 |
| Protein kinase C |
Melittin from honey bee venom |
M2272 |
| Protein kinase C |
Myricetin |
M6760 |
| Protein kinase C |
rac-2-Methoxy-3-hexadecanamido-1-propylphosphocholine |
M7795 |
| Protein kinase C |
rac-2-Methoxy-3-octadecanamido-1-propylphosphocholine |
M8045 |
| Protein kinase C |
Myristoyl-Phe-Ala-Arg-Lys-Gly-Ala-Leu-Arg-Gln |
M8814 |
| Protein kinase C |
Palmitoyl-DL-Carnitine Chloride |
P4509 |
| Protein kinase C |
Protein Kinase C Fragment 19-31 Amide |
P2235 |
| Protein kinase C |
Protein Kinase C Inhibitor, Myristoylated |
P3115 |
| Protein kinase C |
Protein Kinase C Fragment 19-36 |
P8462 |
| Protein kinase C |
Rottlerin |
R5648 |
| Protein kinase C |
DL-Stearoylcarnitine chloride |
S2381 |
| Protein kinase C |
Staurosporine from Streptomyces sp. |
S4400 |
| Protein kinase C |
Staurosporine aglycone |
S3939 |
| Protein kinase C |
D-Sphingosine |
S7049 |
| Protein kinase C |
Na-p-Tosyl-L-lysine chloromethyl ketone hydrochloride |
T7254 |
| Protein kinase C |
N,N,N-Trimethylsphingosine chloride |
T6067 |
| Protein Kinase C beta |
Hispidin |
H5257 |
| Protein kinase, DNA dependent |
4,5-Dimethoxy-6-nitrobenzaldehyde >99% solid |
D9192 |
| Protein kinase, DNA dependent |
1-(2-Hydroxy-4-morpholin-4-yl-phenyl)ethanone |
I2159 |
| Protein kinase, DNA dependent |
NU7026 solid ³99% |
I2159 |
| Protein kinase, DNA dependent |
NU7026 solid >99% |
N1537 |
| Protein kinase erbB2,2 |
Geldanamycin from Streptomyces hygroscopicus |
G3381 |
| Protein kinase G I alpha |
8-(4-Chlorophenylthio)-guanosine 3',5'-cyclic monophosphorothioate, Rp Isomer triethylammonium salt |
C-240 |
| Protein kinase G |
Arg-Lys-Arg-Ala-Arg-Lys-Glu |
A8186 |
| Protein kinase G |
HA-1004 hydrochloride |
G1274 |
| Protein kinase G |
N-(2-[Methylamino]ethyl)-5-isoquinolinesulfonamide hydrochloride |
M9656 |
| Protein Kinase, Calmodulin dependent |
Rottlerin |
R5648 |
| Protein Kinase II, Calmodulin dependent |
Autocamtide 2-related inhibitory peptide trifluoroacetate salt |
A4308 |
| Protein Kinase II, Calmodulin dependent |
Calmodulin Kinase II Inhibitor from rat |
C1360 |
| Protein Kinase II, Calmodulin dependent |
KN-62 |
I2142 |
| Protein Kinase II, Calmodulin dependent |
KN-93 |
K1385 |
| Protein Kinase p38 MAPK |
SB-200646 hydrochloride >98 % (HPLC) |
S0568 |
| Protein Kinase p38 MAPK |
SB 202190 >99 % (HPLC) |
S7067 |
| Protein kinase v-src |
Geldanamycin from Streptomyces hygroscopicus |
G3381 |
| Protein Kinase, cRAF1 |
GW5074 |
G6416 |
| Protein kinase, tyrosine |
Amiloride hydrochloride hydrate |
A7410 |
| Protein kinase, tyrosine |
Chelerythrine chloride |
C2932 |
| Protein kinase, tyrosine |
Daidzein |
D7802 |
| Protein kinase, tyrosine |
Herbimycin A from Streptomyces hygroscopicus |
H6649 |
| Protein kinase, tyrosine |
Lavendustin A |
L2400 |
| Protein kinase, tyrosine |
Lavendustin C |
L1289 |
| Protein kinase, tyrosine |
Quercetin dihydrate |
Q0125 |
| Protein kinase, tyrosine |
ST638 solid >99% |
S5139 |
| Protein kinase, tyrosine ; competitive inhibitor of ATP |
Genistein |
G6649 |
| Protein kinase, tyrosine ; competitive inhibitor of ATP |
Genistein |
G6776 |
| Protein kinase, tyrosine blocks production of TNF-alpha |
Tyrphostin AG 126 |
T9177 |
| Protein kinase, tyrosine blocks production of TNF-alpha |
Tyrphostin AG 1288 |
T9302 |
| Protein kinase, tyrosine p56lck |
Damnacanthal |
D6309 |
| Protein kinase, tyrosine Syk, p40 and p56 |
Piceatannol |
P0453 |
| Protein kinase, tyrosine, EGF receptor |
Daphnetin |
D5564 |
| Protein kinase, tyrosine, EGF receptor |
2,5-Dihydroxycinnamic acid methyl ester |
D2667 |
| Protein kinase, tyrosine, EGF receptor |
Geldanamycin from Streptomyces hygroscopicus |
G3381 |
| Protein kinase, tyrosine, EGF receptor |
GW583340 dihydrochloride solid ³97% (HPLC) |
G3545 |
| Protein kinase, tyrosine, EGF receptor |
SU 4312 >99 % (HPLC) |
S8567 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin 1 |
T7040 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin 23 |
T7165 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin 25 |
T7290 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin 46 |
T7415 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin 47 |
T7540 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin 51 |
T7665 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin 63 |
T7790 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin A9 |
T-182 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 1007 |
T5943 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 1024 |
T6068 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 1112 |
T6193 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 112 |
T6943 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 1478 |
T4182 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 34 |
T6318 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 494 |
T4318 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 527 |
T4443 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 528 |
T4568 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 537 |
T4693 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 555 |
T4818 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 556 |
T4943 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 658 |
T5068 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 698 |
T5193 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 825 |
T5443 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 835 |
T5568 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 974 |
T5818 |
| Protein kinase, tyrosine, EGF receptor |
Tyrphostin AG 1433 |
T5317 |
| Protein kinase, tyrosine, EGF receptor |
SU 5416 >98 % (HPLC) |
|