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CDP-alcohol hydrolase, a very efficient activity of the 5'-nucleotidase/UDP-sugar hydrolase encoded by the ushA gene of Yersinia intermedia and Escherichia coli. Isabel Alves-Pereira et al J. Bacteriol. 190, 6153-61, (2008)
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Mycobacterium tuberculosis acg gene is required for growth and virulence in vivo. Yanmin Hu et al PLoS ONE 6, e20958, (2011)
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Genetic and structural insights into the dissemination potential of the extremely broad-spectrum class A β-lactamase KPC-2 identified in an Escherichia coli strain and an Enterobacter cloacae strain isolated from the same patient in France. Stephanie Petrella et al Antimicrob. Agents Chemother. 52, 3725-36, (2008)
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Beta-lactam screening by specific residues of the OmpF eyelet. Stéphanie Vidal et al J. Med. Chem. 48, 1395-400, (2005)
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Three-dimensional quantitative structure-activity relationship analyses of beta-lactam antibiotics and tripeptides as substrates of the mammalian H+/peptide cotransporter PEPT1. Annegret Biegel et al J. Med. Chem. 48, 4410-9, (2005)
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Aqua mediated synthesis of substituted 2-amino-4H-chromenes and in vitro study as antibacterial agents. Mazaahir Kidwai et al Bioorg. Med. Chem. Lett. 15, 4295-8, (2005)
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Studies on synthesis and evaluation of quantitative structure-activity relationship of 5-[(3'-chloro-4',4'-disubstituted-2-oxoazetidinyl)(N-nitro)amino]-6-hydroxy-3-alkyl/aryl[1,3]azaphospholo[1,5-a]pyridin-1-yl-phosphorus dichlorides. Pratibha Sharma et al Bioorg. Med. Chem. Lett. 15, 937-43, (2005)
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Studies on synthesis and evaluation of quantitative structure-activity relationship of 10-methyl-6-oxo-5-arylazo-6,7-dihydro-5H-[1,3]azaphospholo[1,5-d][1,4]benzodiazepin-2-phospha-3-ethoxycarbonyl-1-phosphorus dichlorides. Ashok Kumar et al Bioorg. Med. Chem. Lett. 16, 2484-91, (2006)
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Synthesis and antibacterial evaluation of ureides of Baylis-Hillman derivatives. Somnath Nag et al Bioorg. Med. Chem. Lett. 16, 3824-8, (2006)
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Lactones from a brown alga endophytic fungus (No. ZZF36) from the South China Sea and their antimicrobial activities. Rui-yun Yang et al Bioorg. Med. Chem. Lett. 16, 4205-8, (2006)
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Naphtho[2,3-b][1,4]-thiazine-5,10-diones and 3-substituted-1,4-dioxo-1,4-dihydronaphthalen-2-yl-thioalkanoate derivatives: synthesis and biological evaluation as potential antibacterial and antifungal agents. Vishnu K Tandon et al Bioorg. Med. Chem. Lett. 16, 5883-7, (2006)
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A clinical drug library screen identifies astemizole as an antimalarial agent. Curtis R Chong et al Nat. Chem. Biol. 2, 415-6, (2006)
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Antibacterial nicotinamide adenine dinucleotide synthetase inhibitors: amide- and ether-linked tethered dimers with alpha-amino acid end groups. Sadanandan E Velu et al J. Med. Chem. 50, 2612-21, (2007)
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Optimizing cell permeation of an antibiotic resistance inhibitor for improved efficacy. Venturelli, A.; et al. J. Med. Chem. 50, 5644, (2007)
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Unexpected inhibition of peptidoglycan LD-transpeptidase from Enterococcus faecium by the beta-lactam imipenem. Jean-Luc Mainardi et al J. Biol. Chem. 282, 30414-22, (2007)
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Fatty acyl benzamido antibacterials based on inhibition of DnaK-catalyzed protein folding. Markus Liebscher et al J. Biol. Chem. 282, 4437-46, (2007)
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PTC124 targets genetic disorders caused by nonsense mutations. Ellen M Welch et al Nature 447, 87-91, (2007)
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Anti-mycobacterial activity of a bis-sulfonamide. Brendan L Wilkinson et al Bioorg. Med. Chem. Lett. 17, 1355-7, (2007)
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Synthesis of pseudopeptides based L-tryptophan as a potential antimicrobial agent. Jian Lv et al Bioorg. Med. Chem. Lett. 17, 1601-7, (2007)
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Synthesis and antimicrobial activity of some novel phenyl and benzimidazole substituted benzyl ethers. Ozden Ozel Güven et al Bioorg. Med. Chem. Lett. 17, 2233-6, (2007)
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New antifungal flavonoid glycoside from Vitex negundo. B Sathiamoorthy et al Bioorg. Med. Chem. Lett. 17, 239-42, (2007)
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Synthesis and evaluation of amphiphilic cationic quinine-derived for antibacterial activity against methicillin-resistant Staphylococcus aureus. Jian Lv et al Bioorg. Med. Chem. Lett. 17, 4102-6, (2007)
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Design, synthesis, and evaluation of efflux substrate-metal chelator conjugates as potential antimicrobial agents. Yanling Zhang et al Bioorg. Med. Chem. Lett. 17, 707-11, (2007)
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Synthesis and structure-antibacterial activity relationship investigation of isomeric 2,3,5-substituted perhydropyrrolo[3,4-d]isoxazole-4,6-diones. Hikmet Agirbas et al Bioorg. Med. Chem. 15, 2322-33, (2007)
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Identification of antitumour activity of novel derivatives of 8-aryl-2,6,7,8-tetrahydroimidazo[2,1-c][1,2,4]triazine-3,4-dione and 8-aryl-4-imino-2,3,7,8-tetrahydroimidazo[2,1-c][1,2,4]triazin-3(6H)-one. Krzysztof Sztanke et al Bioorg. Med. Chem. 15, 2837-49, (2007)
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Synthesis, characterization and antimicrobial activity of new aliphatic sulfonamide. Neslihan Ozbek et al Bioorg. Med. Chem. 15, 5105-9, (2007)
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Identification of antibacterial and antiviral activities of novel fused 1,2,4-triazine esters. Krzysztof Sztanke et al Bioorg. Med. Chem. 15, 5480-6, (2007)
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1-Acylthiosemicarbazides, 1,2,4-triazole-5(4H)-thiones, 1,3,4-thiadiazoles and hydrazones containing 5-methyl-2-benzoxazolinones: synthesis, analgesic-anti-inflammatory and antimicrobial activities. Umut Salgin-Gök?en et al Bioorg. Med. Chem. 15, 5738-51, (2007)
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Synthesis and antimicrobial activity of some new thiazolyl thiazolidine-2,4-dione derivatives. Oya Bozdağ-Dündar et al Bioorg. Med. Chem. 15, 6012-7, (2007)
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Utility of 6-amino-2-thiouracil as a precursor for the synthesis of bioactive pyrimidine derivatives. Nadia Ragab Mohamed et al Bioorg. Med. Chem. 15, 6227-35, (2007)
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Raman, FT-IR, NMR spectroscopic data and antimicrobial activity of bis[micro2-(benzimidazol-2-yl)-2-ethanethiolato-N,S,S-chloro-palladium(II)] dimer, [(micro2-CH2CH2NHNCC6H4)PdCl]2.C2H5OH complex. Naz M Aghatabay et al Eur. J. Med. Chem. 42, 1069-75, (2007)
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Synthesis and in vitro antimicrobial activity of new 2-[p-substituted-benzyl]-5-[substituted-carbonylamino]benzoxazoles. Betul Tekiner-Gulbas et al Eur. J. Med. Chem. 42, 1293-9, (2007)
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Synthesis, characterization and antimicrobial activity of Fe(II), Zn(II), Cd(II) and Hg(II) complexes with 2,6-bis(benzimidazol-2-yl) pyridine ligand. Naz M Aghatabay et al Eur. J. Med. Chem. 42, 205-13, (2007)
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Synthesis, antimicrobial, and anti-inflammatory activities of novel 2-(1-adamantyl)-5-substituted-1,3,4-oxadiazoles and 2-(1-adamantylamino)-5-substituted-1,3,4-thiadiazoles. Adnan A Kadi et al Eur. J. Med. Chem. 42, 235-42, (2007)
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Synthesis, in vitro antibacterial and antifungal evaluations of 2-amino-4-(1-naphthyl)-6-arylpyrimidines. N Ingarsal et al Eur. J. Med. Chem. 42, 517-20, (2007)
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Synthesis and antimicrobial evaluation of some new thiazole, thiazolidinone and thiazoline derivatives starting from 1-chloro-3,4-dihydronaphthalene-2-carboxaldehyde. Samir Bondock et al Eur. J. Med. Chem. 42, 948-54, (2007)
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Detection of a new SHV-type extended-spectrum beta-lactamase, SHV-31, in a Klebsiella pneumoniae strain causing a large nosocomial outbreak in The Netherlands. A Mazzariol et al Antimicrob. Agents Chemother. 51, 1082-4, (2007)
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Prevalence of plasmid-mediated quinolone resistance determinants QnrA, QnrB, and QnrS among clinical isolates of Enterobacter cloacae in a Taiwanese hospital. Jiunn-Jong Wu et al Antimicrob. Agents Chemother. 51, 1223-7, (2007)
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In vitro and in vivo antibacterial activities of heteroaryl isothiazolones against resistant gram-positive pathogens. Michael J Pucci et al Antimicrob. Agents Chemother. 51, 1259-67, (2007)
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Increased genome instability in Escherichia coli lon mutants: relation to emergence of multiple-antibiotic-resistant (Mar) mutants caused by insertion sequence elements and large tandem genomic amplifications. Hervé Nicoloff et al Antimicrob. Agents Chemother. 51, 1293-303, (2007)
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First report of plasmid-mediated qnrA1 in a ciprofloxacin-resistant Escherichia coli strain in Latin America. Mariana Castanheira et al Antimicrob. Agents Chemother. 51, 1527-9, (2007)
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First identification of Pseudomonas aeruginosa isolates producing a KPC-type carbapenem-hydrolyzing beta-lactamase. Maria Virginia Villegas et al Antimicrob. Agents Chemother. 51, 1553-5, (2007)
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Horizontal Gene Transfer of ftsI, Encoding Penicillin-Binding Protein 3, in Haemophilus influenzae. Sho Takahata, Takashi Ida, et. Al Antimicrob. Agents Chemother. 51, 1589 - 1595, (2007)
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Antibiotic Susceptibility Profile of Bifidobacteria as Affected by Oxgall, Acid, and Hydrogen Peroxide Stress. E. Kheadr, N. Dabour, et al. Antimicrob. Agents Chemother. 51, 169-174, (2007)
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Spread of extended-spectrum beta-lactamase CTX-M-producing escherichia coli clinical isolates in community and nosocomial environments in Portugal. Nuno Mendonça et al Antimicrob. Agents Chemother. 51, 1946-55, (2007)
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Time-kill and synergism studies of ceftobiprole against Enterococcus faecalis, including beta-lactamase-producing and vancomycin-resistant isolates. Cesar A Arias et al Antimicrob. Agents Chemother. 51, 2043-7, (2007)
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Polyamine effects on antibiotic susceptibility in bacteria. Dong-Hyeon Kwon et al Antimicrob. Agents Chemother. 51, 2070-7, (2007)
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PhoU is a persistence switch involved in persister formation and tolerance to multiple antibiotics and stresses in Escherichia coli. Yongfang Li et al Antimicrob. Agents Chemother. 51, 2092-9, (2007)
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Identification of the novel narrow-spectrum beta-lactamase SCO-1 in Acinetobacter spp. from Argentina. Laurent Poirel et al Antimicrob. Agents Chemother. 51, 2179-84, (2007)
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SCO-1, a novel plasmid-mediated class A beta-lactamase with carbenicillinase characteristics from Escherichia coli. C C Papagiannitsis et al Antimicrob. Agents Chemother. 51, 2185-8, (2007)
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Biochemical characterization of PER-2 and genetic environment of blaPER-2. Pablo Power et al Antimicrob. Agents Chemother. 51, 2359-65, (2007)
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Enterobacteriaceae bloodstream infections: presence of integrons, risk factors, and outcome. George L Daikos et al Antimicrob. Agents Chemother. 51, 2366-72, (2007)
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Transferable resistance to aminoglycosides by methylation of G1405 in 16S rRNA and to hydrophilic fluoroquinolones by QepA-mediated efflux in Escherichia coli. Bruno Périchon et al Antimicrob. Agents Chemother. 51, 2464-9, (2007)
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Ampicillin-resistant non-beta-lactamase-producing Haemophilus influenzae in Spain: recent emergence of clonal isolates with increased resistance to cefotaxime and cefixime. Silvia García-Cobos et al Antimicrob. Agents Chemother. 51, 2564-73, (2007)
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Characterization of an integron carrying blaIMP-1 and a new aminoglycoside resistance gene, aac(6')-31, and its dissemination among genetically unrelated clinical isolates in a Brazilian hospital. Rodrigo E Mendes et al Antimicrob. Agents Chemother. 51, 2611-4, (2007)
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Cytoplasmic-membrane anchoring of a class A beta-lactamase and its capacity in manifesting antibiotic resistance. Maxim Suvorov et al Antimicrob. Agents Chemother. 51, 2937-42, (2007)
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Identification and characterization of a new metallo-beta-lactamase, IND-5, from a clinical isolate of Chryseobacterium indologenes. Mariagrazia Perilli et al Antimicrob. Agents Chemother. 51, 2988-90, (2007)
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Novel complex class 1 integron bearing an ISCR1 element in an Escherichia coli isolate carrying the blaCTX-M-14 gene. Il Kwon Bae et al Antimicrob. Agents Chemother. 51, 3017-9, (2007)
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First characterization of heterogeneous resistance to imipenem in invasive nontypeable Haemophilus influenzae isolates. Marina Cerquetti et al Antimicrob. Agents Chemother. 51, 3155-61, (2007)
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Cloning, nucleotide sequencing, and analysis of the AcrAB-TolC efflux pump of Enterobacter cloacae and determination of its involvement in antibiotic resistance in a clinical isolate. Astrid Pérez et al Antimicrob. Agents Chemother. 51, 3247-53, (2007)
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New plasmid-mediated fluoroquinolone efflux pump, QepA, found in an Escherichia coli clinical isolate. Kunikazu Yamane et al Antimicrob. Agents Chemother. 51, 3354-60, (2007)
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In vitro activity of telavancin against gram-positive clinical isolates recently obtained in Europe. W T M Jansen et al Antimicrob. Agents Chemother. 51, 3420-4, (2007)
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Colistin methanesulfonate against multidrug-resistant Acinetobacter baumannii in an in vitro pharmacodynamic model. Lisa A Kroeger et al Antimicrob. Agents Chemother. 51, 3431-3, (2007)
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Can the Etest correctly determine the MICs of beta-lactam and cephalosporin antibiotics for beta-lactamase-negative ampicillin-resistant Haemophilus influenzae? Dewan Sakhawat Billal et al Antimicrob. Agents Chemother. 51, 3463-4, (2007)
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Pharmacokinetics of penicillin G in infants with a gestational age of less than 32 weeks. Anouk E Muller et al Antimicrob. Agents Chemother. 51, 3720-5, (2007)
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Genetic characteristics and clonal dissemination of beta-lactamase-negative ampicillin-resistant Haemophilus influenzae strains isolated from the upper respiratory tract of patients in Japan. Muneki Hotomi et al Antimicrob. Agents Chemother. 51, 3969-76, (2007)
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Prevalence and expression of the plasmid-mediated quinolone resistance determinant qnrA1. Xiaogang Xu et al Antimicrob. Agents Chemother. 51, 4105-10, (2007)
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The PhoQ-activating potential of antimicrobial peptides contributes to antimicrobial efficacy and is predictive of the induction of bacterial resistance. Jason Kindrachuk et al Antimicrob. Agents Chemother. 51, 4374-81, (2007)
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Biochemical Characterization of SFC-1, a class A carbapenem-hydrolyzing beta-lactamase. Fátima Fonseca et al Antimicrob. Agents Chemother. 51, 4512-4, (2007)
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Development of colistin-dependent Acinetobacter baumannii-Acinetobacter calcoaceticus complex. Joshua S Hawley et al Antimicrob. Agents Chemother. 51, 4529-30, (2007)
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Diversity of ampicillin resistance genes and antimicrobial susceptibility patterns in Haemophilus influenzae strains isolated in Korea. In-Suk Kim et al Antimicrob. Agents Chemother. 51, 453-60, (2007)
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Contribution of target gene mutations and efflux to decreased susceptibility of Salmonella enterica serovar typhimurium to fluoroquinolones and other antimicrobials. Sheng Chen et al Antimicrob. Agents Chemother. 51, 535-42, (2007)
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Substrate competition studies using whole-cell accumulation assays with the major tripartite multidrug efflux pumps of Escherichia coli. Christopher A Elkins et al Antimicrob. Agents Chemother. 51, 923-9, (2007)
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Antimicrobial arylcoumarins from Asphodelus microcarpus. Hesham R El-Seedi et al J. Nat. Prod. 70, 118-20, (2007)
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Disrupting antibiotic resistance propagation by inhibiting the conjugative DNA relaxase. Scott A Lujan et al Proc. Natl. Acad. Sci. U. S. A. 104, 12282-7, (2007)
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Water-soluble pleuromutilin derivative with excellent in vitro and in vivo antibacterial activity against gram-positive pathogens. Yoshimi Hirokawa et al J. Med. Chem. 51, 1991-4, (2008)
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Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1. Gustav Ahlin et al J. Med. Chem. 51, 5932-42, (2008)
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Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors. Lourdes Santana et al J. Med. Chem. 51, 6740-51, (2008)
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Antimicrobial activities of the bromophenols from the red alga Odonthalia corymbifera and some synthetic derivatives. Ki-Bong Oh et al Bioorg. Med. Chem. Lett. 18, 104-8, (2008)
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Synthesis and biological evaluation of novel 1,3,5-triazine derivatives as antimicrobial agents. Chunhui Zhou et al Bioorg. Med. Chem. Lett. 18, 1308-11, (2008)
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Synthesis and antimicrobial activity of beta-lactam-bile acid conjugates linked via triazole. Namdev S Vatmurge et al Bioorg. Med. Chem. Lett. 18, 2043-7, (2008)
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Substituted 3-((Z)-2-(4-nitrophenyl)-2-(1H-tetrazol-5-yl) vinyl)-4H-chromen-4-ones as novel anti-MRSA agents: synthesis, SAR, and in-vitro assessment. Santosh D Diwakar et al Bioorg. Med. Chem. Lett. 18, 4678-81, (2008)
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Design and synthesis of 3-pyrazolyl-thiophene, thieno[2,3-d]pyrimidines as new bioactive and pharmacological activities. H N Hafez et al Bioorg. Med. Chem. Lett. 18, 5222-7, (2008)
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Inhibition of Candida albicans isocitrate lyase activity by sesterterpene sulfates from the tropical sponge Dysidea sp. Dongha Lee et al Bioorg. Med. Chem. Lett. 18, 5377-80, (2008)
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Synthesis and antimicrobial activity of 2-alkenylchroman-4-ones, 2-alkenylthiochroman-4-ones and 2-alkenylquinol-4-ones. Nicole Hoettecke et al Bioorg. Med. Chem. 16, 10319-25, (2008)
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2-Heteroarylimino-5-benzylidene-4-thiazolidinones analogues of 2-thiazolylimino-5-benzylidene-4-thiazolidinones with antimicrobial activity: synthesis and structure-activity relationship. Paola Vicini et al Bioorg. Med. Chem. 16, 3714-24, (2008)
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Bioactive alkenylphenols from Piper obliquum. Carola Valdivia et al Bioorg. Med. Chem. 16, 4120-6, (2008)
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Hetero-Diels-Alder reaction of 1,3-bis(trimethylsilyloxy)-1,3-butadienes with arylsulfonylcyanides. Synthesis and antimicrobial activity of 4-hydroxy-2-(arylsulfonyl)pyridines. Ibrar Hussain et al Bioorg. Med. Chem. 16, 9898-903, (2008)
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Synthesis, potent anti-staphylococcal activity and QSARs of some novel 2-anilinobenzazoles. Seçkin Ozden et al Eur. J. Med. Chem. 43, 1390-402, (2008)
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Synthesis and antimicrobial activity of some new heterocycles incorporating antipyrine moiety. Samir Bondock et al Eur. J. Med. Chem. 43, 2122-9, (2008)
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Synthesis and biological evaluation of diversely substituted indolin-2-ones. Fadoua Bouchikhi et al Eur. J. Med. Chem. 43, 2316-22, (2008)
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Synthesis, determination of the lipophilicity, anticancer and antimicrobial properties of some fused 1,2,4-triazole derivatives. Krzysztof Sztanke et al Eur. J. Med. Chem. 43, 404-19, (2008)
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Synthesis and biological evaluation of some thiazolyl and thiadiazolyl derivatives of 1H-pyrazole as anti-inflammatory antimicrobial agents. Adnan A Bekhit et al Eur. J. Med. Chem. 43, 456-63, (2008)
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Induction of L1 and L2 beta-lactamases of Stenotrophomonas maltophilia. Rouh-Mei Hu et al Antimicrob. Agents Chemother. 52, 1198-200, (2008)
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Genetic and biochemical characterization of OXA-63, a new class D beta-lactamase from Brachyspira pilosicoli BM4442. Djalal Meziane-Cherif et al Antimicrob. Agents Chemother. 52, 1264-8, (2008)
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Convergent in vivo and in vitro selection of ceftazidime resistance mutations at position 167 of CTX-M-3 beta-lactamase in hypermutable Escherichia coli strains. Marina N Stepanova et al Antimicrob. Agents Chemother. 52, 1297-301, (2008)
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Induction of L1 and L2 beta-lactamase production in Stenotrophomonas maltophilia is dependent on an AmpR-type regulator. Aki Okazaki et al Antimicrob. Agents Chemother. 52, 1525-8, (2008)
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Carbapenem-resistant Acinetobacter baumannii isolates from Tunisia producing the OXA-58-like carbapenem-hydrolyzing oxacillinase OXA-97. Laurent Poirel et al Antimicrob. Agents Chemother. 52, 1613-7, (2008)
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Synergy between polyethylenimine and different families of antibiotics against a resistant clinical isolate of Pseudomonas aeruginosa. Hayssam Khalil et al Antimicrob. Agents Chemother. 52, 1635-41, (2008)
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In vitro activities of the Rx-01 oxazolidinones against hospital and community pathogens. Laura Lawrence et al Antimicrob. Agents Chemother. 52, 1653-62, (2008)
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Comparison of antimicrobial resistance profiles among extended-spectrum-beta-lactamase-producing and acquired AmpC beta-lactamase-producing Escherichia coli isolates from Canadian intensive care units. Patricia J Baudry et al Antimicrob. Agents Chemother. 52, 1846-9, (2008)
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Comparison of the efficacies of oral beta-lactams in selection of Haemophilus influenzae transformants with mutated ftsI genes. Sho Takahata et al Antimicrob. Agents Chemother. 52, 1880-3, (2008)
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Emergence of Serratia marcescens, Klebsiella pneumoniae, and Escherichia coli Isolates possessing the plasmid-mediated carbapenem-hydrolyzing beta-lactamase KPC-2 in intensive care units of a Chinese hospital. Jia Chang Cai et al Antimicrob. Agents Chemother. 52, 2014-8, (2008)
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Methicillin-resistant Staphylococcus saprophyticus isolates carrying staphylococcal cassette chromosome mec have emerged in urogenital tract infections. Masato Higashide et al Antimicrob. Agents Chemother. 52, 2061-8, (2008)
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Biochemical characterization of metallo-beta-lactamase VIM-11 from a Pseudomonas aeruginosa clinical strain. Patricia Marchiaro et al Antimicrob. Agents Chemother. 52, 2250-2, (2008)
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Fitness trade-offs in blaTEM evolution. Joanna E Mroczkowska et al Antimicrob. Agents Chemother. 52, 2340-5, (2008)
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Comparative surveillance study of telavancin activity against recently collected gram-positive clinical isolates from across the United States. Deborah C Draghi et al Antimicrob. Agents Chemother. 52, 2383-8, (2008)
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Low beta-lactamase-negative ampicillin-resistant Haemophilus influenzae strains are best detected by testing amoxicillin susceptibility by the broth microdilution method. Silvia García-Cobos et al Antimicrob. Agents Chemother. 52, 2407-14, (2008)
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Functional diversity among metallo-beta-lactamases: characterization of the CAR-1 enzyme of Erwinia carotovora. Magdalena Stoczko et al Antimicrob. Agents Chemother. 52, 2473-9, (2008)
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Identification of a novel multidrug efflux pump of Mycobacterium tuberculosis. Olga Danilchanka et al Antimicrob. Agents Chemother. 52, 2503-11, (2008)
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In vitro activity of telavancin against resistant gram-positive bacteria. Kevin M Krause et al Antimicrob. Agents Chemother. 52, 2647-52, (2008)
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Role of global regulators and nucleotide metabolism in antibiotic tolerance in Escherichia coli. Sonja Hansen et al Antimicrob. Agents Chemother. 52, 2718-26, (2008)
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Mechanism and fitness costs of PR-39 resistance in Salmonella enterica serovar Typhimurium LT2. Maria Pränting et al Antimicrob. Agents Chemother. 52, 2734-41, (2008)
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Antimicrobial susceptibilities of geographically diverse clinical human isolates of Leptospira. Roseanne A Ressner et al Antimicrob. Agents Chemother. 52, 2750-4, (2008)
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Discovery and characterization of QPT-1, the progenitor of a new class of bacterial topoisomerase inhibitors. Alita A Miller et al Antimicrob. Agents Chemother. 52, 2806-12, (2008)
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First molecular characterization of group B streptococci with reduced penicillin susceptibility. Kouji Kimura et al Antimicrob. Agents Chemother. 52, 2890-7, (2008)
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Kinetic characterization of VIM-7, a divergent member of the VIM metallo-beta-lactamase family. Ørjan Samuelsen et al Antimicrob. Agents Chemother. 52, 2905-8, (2008)
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Point mutation in the group B streptococcal pbp2x gene conferring decreased susceptibility to beta-lactam antibiotics. Samira Dahesh et al Antimicrob. Agents Chemother. 52, 2915-8, (2008)
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In vitro activity of tigecycline against multidrug-resistant Acinetobacter baumannii and selection of tigecycline-amikacin synergy. Ellen S Moland et al Antimicrob. Agents Chemother. 52, 2940-2, (2008)
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Characterization of the carbapenem-hydrolyzing oxacillinase oxa-58 in an Acinetobacter genospecies 3 clinical isolate. Sara Marti et al Antimicrob. Agents Chemother. 52, 2955-8, (2008)
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In vitro profiling of ceftaroline against a collection of recent bacterial clinical isolates from across the United States. Yigong Ge et al Antimicrob. Agents Chemother. 52, 3398-407, (2008)
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Characterization of the new metallo-beta-lactamase VIM-13 and its integron-borne gene from a Pseudomonas aeruginosa clinical isolate in Spain. Carlos Juan et al Antimicrob. Agents Chemother. 52, 3589-96, (2008)
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Molecular and biochemical characterization of SHV-56, a novel inhibitor-resistant beta-lactamase from Klebsiella pneumoniae. Véronique Dubois et al Antimicrob. Agents Chemother. 52, 3792-4, (2008)
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Genetic basis of multidrug resistance in Acinetobacter baumannii clinical isolates at a tertiary medical center in Pennsylvania. Jennifer M Adams-Haduch et al Antimicrob. Agents Chemother. 52, 3837-43, (2008)
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A plasmid-borne blaOXA-58 gene confers imipenem resistance to Acinetobacter baumannii isolates from a Lebanese hospital. Raffaele Zarrilli et al Antimicrob. Agents Chemother. 52, 4115-20, (2008)
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KHM-1, a novel plasmid-mediated metallo-beta-lactamase from a Citrobacter freundii clinical isolate. Jun-ichiro Sekiguchi et al Antimicrob. Agents Chemother. 52, 4194-7, (2008)
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In vitro activity of ceftaroline against Streptococcus pneumoniae isolates exhibiting resistance to penicillin, amoxicillin, and cefotaxime. Asunción Fenoll et al Antimicrob. Agents Chemother. 52, 4209-10, (2008)
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Genetic heterogeneity in pbp genes among clinically isolated group B Streptococci with reduced penicillin susceptibility. Noriyuki Nagano et al Antimicrob. Agents Chemother. 52, 4258-67, (2008)
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Replication of Colonic Crohn's Disease Mucosal Escherichia coli Isolates within Macrophages and Their Susceptibility to Antibiotics. Sreedhar Subramanian et al Antimicrob. Agents Chemother. 52, 427-34, (2008)
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In vitro activities of doripenem, a new broad-spectrum carbapenem, against recently collected clinical anaerobic isolates, with emphasis on the Bacteroides fragilis group. David R Snydman et al Antimicrob. Agents Chemother. 52, 4492-6, (2008)
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Genetic and biochemical characterization of CAD-1, a chromosomally encoded new class A penicillinase from Carnobacterium divergens. Djalal Meziane-Cherif et al Antimicrob. Agents Chemother. 52, 551-6, (2008)
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Combined real-time PCR and pyrosequencing strategy for objective, sensitive, specific, and high-throughput identification of reduced susceptibility to penicillins in Neisseria meningitidis. Sara Thulin et al Antimicrob. Agents Chemother. 52, 753-6, (2008)
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RmtC 16S rRNA methyltransferase in Australia. Zhiyong Zong et al Antimicrob. Agents Chemother. 52, 794-5, (2008)
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E240V substitution increases catalytic efficiency toward ceftazidime in a new natural TEM-type extended-spectrum beta-lactamase, TEM-149, from Enterobacter aerogenes and Serratia marcescens clinical isolates. Mariagrazia Perilli et al Antimicrob. Agents Chemother. 52, 915-9, (2008)
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Reduced Susceptibility of Proteus mirabilis to triclosan. David J Stickler et al Antimicrob. Agents Chemother. 52, 991-4, (2008)
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Bioactive 5alpha-pregnane-type steroidal alkaloids from Sarcococca hookeriana. Krishna P Devkota et al J. Nat. Prod. 71, 1481-4, (2008)
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Scalarane sesterterpenes from the sponge Smenospongia sp. Jueun Song et al J. Nat. Prod. 71, 1866-71, (2008)
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Sesterterpenoids from the sponge Sarcotragus sp. Nan Wang et al J. Nat. Prod. 71, 551-7, (2008)
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Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds. R Scott Obach et al Drug Metab. Dispos. 36, 1385-405, (2008)
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Physicochemical determinants of human renal clearance. Manthena V S Varma et al J. Med. Chem. 52, 4844-52, (2009)
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Discovery of new inhibitors of resistant Streptococcus pneumoniae penicillin binding protein (PBP) 2x by structure-based virtual screening. Laurence Miguet et al J. Med. Chem. 52, 5926-36, (2009)
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Coordination Chemistry Based Approach to Lipophilic Inhibitors of 1-Deoxy-D-xylulose-5-phosphate Reductoisomerase Deng, L.; et al. J. Med. Chem. 52, 6539-6542, (2009)
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Synthesis and antimicrobial activities of halogenated bis(hydroxyphenyl)methanes. Ki-Bong Oh et al Bioorg. Med. Chem. Lett. 19, 945-8, (2009)
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Synthesis and antimicrobial evaluation of some new substituted purine derivatives. Meral Tunçbilek et al Bioorg. Med. Chem. 17, 1693-700, (2009)
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Design, synthesis, antimicrobial activity and molecular modeling studies of novel benzofuroxan derivatives against Staphylococcus aureus. Salomão Dória Jorge et al Bioorg. Med. Chem. 17, 3028-36, (2009)
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Synthesis and antimicrobial activity of 4-hydroxy-4-(pyridyl)alk-3-en-2-ones. Abdolmajid Riahi et al Bioorg. Med. Chem. 17, 4323-6, (2009)
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Guide to Receptors and Channels (GRAC), 4th Edition. Br. J. Pharmacol. 158 Suppl 1, S1-254, (2009)
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Synthesis and in vitro antimicrobial activity of some novel substituted benzimidazole derivatives having potent activity against MRSA. Meral Tunçbilek et al Eur. J. Med. Chem. 44, 1024-33, (2009)
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Synthesis of some new 1,2,4-triazoles, their Mannich and Schiff bases and evaluation of their antimicrobial activities. Hacer Bayrak et al Eur. J. Med. Chem. 44, 1057-66, (2009)
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Synthesis, characterization and antimicrobial activity of Co(II), Zn(II) and Cd(II) complexes with N-benzyloxycarbonyl-S-phenylalanine. Dragana Miti? et al Eur. J. Med. Chem. 44, 1537-44, (2009)
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Synthesis, antimicrobial and cytotoxic activities of some 5-arylidene-4-thioxo-thiazolidine-2-ones. Frederico L Gouveia et al Eur. J. Med. Chem. 44, 2038-43, (2009)
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Synthesis and evaluation of some new benzimidazole derivatives as potential antimicrobial agents. K F Ansari et al Eur. J. Med. Chem. 44, 2294-9, (2009)
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Physicochemical and biological characterization of novel macrocycles derived from o-phthalaldehyde. P Muralidhar Reddy et al Eur. J. Med. Chem. 44, 2621-5, (2009)
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Synthesis and antimicrobial studies of novel methylene bridged benzisoxazolyl imidazo[2,1-b][1,3,4]thiadiazole derivatives. Ravi S Lamani et al Eur. J. Med. Chem. 44, 2828-33, (2009)
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Synthesis of some new 1,3,4-thiadiazol-2-ylmethyl-1,2,4-triazole derivatives and investigation of their antimicrobial activities. Ahmet Demirbas et al Eur. J. Med. Chem. 44, 2896-903, (2009)
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Mono and bis-6-arylbenzimidazo[1,2-c]quinazolines: a new class of antimicrobial agents. Rondla Rohini et al Eur. J. Med. Chem. 44, 3330-9, (2009)
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Synthesis, Raman, FT-IR, NMR spectroscopic data and antimicrobial activity of mixed aza-oxo-thia macrocyclic compounds. Naz Mohammed Aghatabay et al Eur. J. Med. Chem. 44, 365-72, (2009)
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A facile one-pot green synthesis and antibacterial activity of 2-amino-4H-pyrans and 2-amino-5-oxo-5,6,7,8-tetrahydro-4H-chromenes. Dalip Kumar et al Eur. J. Med. Chem. 44, 3805-9, (2009)
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Synthesis, physicochemical properties and antimicrobial activity of some new benzimidazole derivatives. K F Ansari et al Eur. J. Med. Chem. 44, 4028-33, (2009)
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Synthesis, characterization and in vitro antimicrobial activity of novel 2-thioxo-4-thiazolidinones and 4,4'-bis(2-thioxo-4-thiazolidinone-3-yl)diphenylsulfones. Mohamed S A El-Gaby et al Eur. J. Med. Chem. 44, 4148-52, (2009)
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Synthesis of some new 1,2,4-triazoles starting from isonicotinic acid hydrazide and evaluation of their antimicrobial activities. Hacer Bayrak et al Eur. J. Med. Chem. 44, 4362-6, (2009)
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Synthesis and antibacterial activity of some new thiazole and thiophene derivatives. A M Khalil et al Eur. J. Med. Chem. 44, 4434-40, (2009)
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Synthesis and antibacterial activity of some new heterocycles incorporating phthalazine. A M Khalil et al Eur. J. Med. Chem. 44, 4448-54, (2009)
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Synthesis, characterization and antibacterial activity of 2-[1-(5-chloro-2-methoxy-phenyl)-5-methyl-1H-pyrazol-4-yl]-5-(substituted-phenyl)-[1,3,4]oxadiazoles. Neithnadka Premsai Rai et al Eur. J. Med. Chem. 44, 4522-7, (2009)
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Synthesis, Raman, FT-IR, NMR spectroscopic characterization, antimicrobial activity, cytotoxicity and DNA binding of new mixed aza-oxo-thia macrocyclic compounds. Naz M Aghatabay et al Eur. J. Med. Chem. 44, 4681-9, (2009)
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Synthesis, characterization and evaluation of antibacterial activity of some thiazolo[3,2-b][1,2,4]triazole incorporating diphenylsulfone moieties. Stefania-Felicia Barbuceanu et al Eur. J. Med. Chem. 44, 4752-7, (2009)
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Widespread dissemination of aminoglycoside resistance genes armA and rmtB in Klebsiella pneumoniae isolates in Taiwan producing CTX-M-type extended-spectrum beta-lactamases. Ling Ma et al Antimicrob. Agents Chemother. 53, 104-11, (2009)
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Multiple regulatory pathways associated with high-level ciprofloxacin and multidrug resistance in Salmonella enterica serovar enteritidis: involvement of RamA and other global regulators. Edel O'Regan et al Antimicrob. Agents Chemother. 53, 1080-7, (2009)
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Genetic variability among ampC genes from acinetobacter genomic species 3. Alejandro Beceiro et al Antimicrob. Agents Chemother. 53, 1177-84, (2009)
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Effect of DNase and antibiotics on biofilm characteristics. George V Tetz et al Antimicrob. Agents Chemother. 53, 1204-9, (2009)
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Antimicrobial Activity of Prulifloxacin Tested against a Worldwide Collection of Gastroenteritis-Producing Pathogens, Including Those Causing Traveler's Diarrhea Fritsche, T. R.; Biedenbach, D. J., et al. Antimicrob. Agents Chemother. 53, 1221-1224, (2008)
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Carbapenem resistance among Pseudomonas aeruginosa strains from India: evidence for nationwide endemicity of multiple metallo-beta-lactamase clones (VIM-2, -5, -6, and -11 and the newly characterized VIM-18). Mariana Castanheira et al Antimicrob. Agents Chemother. 53, 1225-7, (2009)
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Contribution of vraSR and graSR point mutations to vancomycin resistance in vancomycin-intermediate Staphylococcus aureus. Longzhu Cui et al Antimicrob. Agents Chemother. 53, 1231-4, (2009)
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CMY-31 and CMY-36 cephalosporinases encoded by ColE1-like plasmids. A Zioga et al Antimicrob. Agents Chemother. 53, 1256-9, (2009)
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Activities of dalbavancin against a worldwide collection of 81,673 gram-positive bacterial isolates. Douglas J Biedenbach et al Antimicrob. Agents Chemother. 53, 1260-3, (2009)
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Contribution of oxidative damage to antimicrobial lethality. Xiuhong Wang et al Antimicrob. Agents Chemother. 53, 1395-402, (2009)
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Antibiotic susceptibility and characteristics of Neisseria meningitidis isolates from the African meningitis belt, 2000 to 2006: phenotypic and genotypic perspectives. Sara Thulin Hedberg et al Antimicrob. Agents Chemother. 53, 1561-6, (2009)
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blaCTX-M genes in escherichia coli strains from Croatian Hospitals are located in new (blaCTX-M-3a) and widely spread (blaCTX-M-3a and blaCTX-M-15) genetic structures. Elzbieta Literacka et al Antimicrob. Agents Chemother. 53, 1630-5, (2009)
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New plasmid-mediated quinolone resistance gene, qnrC, found in a clinical isolate of Proteus mirabilis. Minghua Wang et al Antimicrob. Agents Chemother. 53, 1892-7, (2009)
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Novel plasmid-encoded ceftazidime-hydrolyzing CTX-M-53 extended-spectrum beta-lactamase from Salmonella enterica serotypes Westhampton and Senftenberg. Benoît Doublet et al Antimicrob. Agents Chemother. 53, 1944-51, (2009)
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Antianaerobic activity of sulopenem compared to six other agents. Lois M Ednie et al Antimicrob. Agents Chemother. 53, 2163-70, (2009)
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Potency and bactericidal activity of iclaprim against recent clinical gram-positive isolates. Helio S Sader et al Antimicrob. Agents Chemother. 53, 2171-5, (2009)
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Antimicrobial susceptibility and mechanisms of resistance in Shigella and Salmonella isolates from children under five years of age with diarrhea in rural Mozambique. Inácio Mandomando et al Antimicrob. Agents Chemother. 53, 2450-4, (2009)
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Capsular type and antibiotic resistance in Streptococcus agalactiae isolates from patients, ranging from newborns to the elderly, with invasive infections. Somay Yamagata Murayama et al Antimicrob. Agents Chemother. 53, 2650-3, (2009)
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Antibiotic susceptibility of Waddlia chondrophila in Acanthamoeba castellanii amoebae. Geneviève Goy et al Antimicrob. Agents Chemother. 53, 2663-6, (2009)
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Genotypic versus phenotypic characterization, with respect to beta-lactam susceptibility, of Haemophilus influenzae isolates exhibiting decreased susceptibility to beta-lactam resistance markers. David Sevillano et al Antimicrob. Agents Chemother. 53, 267-70, (2009)
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Study of the in vitro activities of rifaximin and comparator agents against 536 anaerobic intestinal bacteria from the perspective of potential utility in pathology involving bowel flora. S M Finegold et al Antimicrob. Agents Chemother. 53, 281-6, (2009)
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First report of plasmid-mediated quinolone resistance determinant qnrS1 in an Escherichia coli strain of animal origin in Italy. Marina Cerquetti et al Antimicrob. Agents Chemother. 53, 3112-4, (2009)
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First detection of plasmid-encoded blaOXY beta-lactamase. J J González-López et al Antimicrob. Agents Chemother. 53, 3143-6, (2009)
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Reduced susceptibility to cefepime among Escherichia coli clinical isolates producing novel variants of CMY-2 beta-lactamase. Yohei Doi et al Antimicrob. Agents Chemother. 53, 3159-61, (2009)
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Detection of the pandemic O25-ST131 human virulent Escherichia coli CTX-M-15-producing clone harboring the qnrB2 and aac(6')-Ib-cr genes in a dog. Constança Pomba et al Antimicrob. Agents Chemother. 53, 327-8, (2009)
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Emergence of high levels of extended-spectrum-beta-lactamase-producing gram-negative bacilli in the Asia-Pacific region: data from the Study for Monitoring Antimicrobial Resistance Trends (SMART) program, 2007. Stephen P Hawser et al Antimicrob. Agents Chemother. 53, 3280-4, (2009)
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Beta-lactamase-mediated beta-lactam resistance in Campylobacter species: prevalence of Cj0299 (bla OXA-61) and evidence for a novel beta-Lactamase in C. jejuni. Deborah J Griggs et al Antimicrob. Agents Chemother. 53, 3357-64, (2009)
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Characterization of pABVA01, a plasmid encoding the OXA-24 carbapenemase from Italian isolates of Acinetobacter baumannii. Marco Maria D'Andrea et al Antimicrob. Agents Chemother. 53, 3528-33, (2009)
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Inhibition of intracellular growth of Salmonella enterica serovar Typhimurium in tissue culture by antisense peptide-phosphorodiamidate morpholino oligomer. Georgi M Mitev et al Antimicrob. Agents Chemother. 53, 3700-4, (2009)
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In vitro activities of telavancin and six comparator agents against anaerobic bacterial isolates. Sydney M Finegold et al Antimicrob. Agents Chemother. 53, 3996-4001, (2009)
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Role of porins in the susceptibility of Mycobacterium smegmatis and Mycobacterium chelonae to aldehyde-based disinfectants and drugs. Zuzana Svetlíková et al Antimicrob. Agents Chemother. 53, 4015-8, (2009)
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Antimicrobial activities of piperacillin-tazobactam against Haemophilus influenzae isolates, including beta-lactamase-negative ampicillin-resistant and beta-lactamase-positive amoxicillin-clavulanate-resistant isolates, and mutations in their quinolone resistance-determining regions. Yoichi Hirakata et al Antimicrob. Agents Chemother. 53, 4225-30, (2009)
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Cotransfer of antibiotic resistance genes and a hylEfm-containing virulence plasmid in Enterococcus faecium. Cesar A Arias et al Antimicrob. Agents Chemother. 53, 4240-6, (2009)
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AI-2/LuxS is involved in increased biofilm formation by Streptococcus intermedius in the presence of antibiotics. Nibras A Ahmed et al Antimicrob. Agents Chemother. 53, 4258-63, (2009)
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IND-6, a highly divergent IND-type metallo-beta-lactamase from Chryseobacterium indologenes strain 597 isolated in Burkina Faso. Boukaré Zeba et al Antimicrob. Agents Chemother. 53, 4320-6, (2009)
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Complete nucleotide sequences of plasmids pEK204, pEK499, and pEK516, encoding CTX-M enzymes in three major Escherichia coli lineages from the United Kingdom, all belonging to the international O25:H4-ST131 clone. Neil Woodford et al Antimicrob. Agents Chemother. 53, 4472-82, (2009)
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In vitro activities of panduratin A against clinical Staphylococcus strains. Yaya Rukayadi et al Antimicrob. Agents Chemother. 53, 4529-32, (2009)
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Emergence of Klebsiella pneumoniae ST258 with KPC-2 in Poland. Anna Baraniak et al Antimicrob. Agents Chemother. 53, 4565-7, (2009)
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Induction of multidrug resistance mechanism in Escherichia coli biofilms by interplay between tetracycline and ampicillin resistance genes. Thithiwat May et al Antimicrob. Agents Chemother. 53, 4628-39, (2009)
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Comparative in vitro activity profile of oritavancin against recent gram-positive clinical isolates. Francis F Arhin et al Antimicrob. Agents Chemother. 53, 4762-71, (2009)
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Combined inactivation of lon and ycgE decreases multidrug susceptibility by reducing the amount of OmpF porin in Escherichia coli. Valérie Duval et al Antimicrob. Agents Chemother. 53, 4944-8, (2009)
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OXA-143, a novel carbapenem-hydrolyzing class D beta-lactamase in Acinetobacter baumannii. Paul G Higgins et al Antimicrob. Agents Chemother. 53, 5035-8, (2009)
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Characterization of a new metallo-beta-lactamase gene, bla(NDM-1), and a novel erythromycin esterase gene carried on a unique genetic structure in Klebsiella pneumoniae sequence type 14 from India. Dongeun Yong et al Antimicrob. Agents Chemother. 53, 5046-54, (2009)
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Effects of subinhibitory concentrations of antibiotics on colonization factor expression by moxifloxacin-susceptible and moxifloxacin-resistant Clostridium difficile strains. Cécile Denève et al Antimicrob. Agents Chemother. 53, 5155-62, (2009)
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High prevalence of plasmid-mediated quinolone resistance determinants qnr, aac(6')-Ib-cr, and qepA among ceftiofur-resistant Enterobacteriaceae isolates from companion and food-producing animals. Junying Ma et al Antimicrob. Agents Chemother. 53, 519-24, (2009)
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Mutational upregulation of a resistance-nodulation-cell division-type multidrug efflux pump, SdeAB, upon exposure to a biocide, cetylpyridinium chloride, and antibiotic resistance in Serratia marcescens. Hideaki Maseda et al Antimicrob. Agents Chemother. 53, 5230-5, (2009)
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Variations in amino acid composition of antisense peptide-phosphorodiamidate morpholino oligomer affect potency against Escherichia coli in vitro and in vivo. Brett L Mellbye et al Antimicrob. Agents Chemother. 53, 525-30, (2009)
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Susceptibilities of 23 Desulfovibrio isolates from humans. Ken-ichi Nakao et al Antimicrob. Agents Chemother. 53, 5308-11, (2009)
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Novel chimeric beta-lactamase CTX-M-64, a hybrid of CTX-M-15-like and CTX-M-14 beta-lactamases, found in a Shigella sonnei strain resistant to various oxyimino-cephalosporins, including ceftazidime. Yukiko Nagano et al Antimicrob. Agents Chemother. 53, 69-74, (2009)
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Prevalence of sulfonamide resistance genes in bacterial isolates from manured agricultural soils and pig slurry in the United Kingdom. K G Byrne-Bailey et al Antimicrob. Agents Chemother. 53, 696-702, (2009)
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Isolation of VanB-type Enterococcus faecalis strains from nosocomial infections: first report of the isolation and identification of the pheromone-responsive plasmids pMG2200, Encoding VanB-type vancomycin resistance and a Bac41-type bacteriocin, and pMG2201, encoding erythromycin resistance and cytolysin (Hly/Bac). Bo Zheng et al Antimicrob. Agents Chemother. 53, 735-47, (2009)
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Identification of a novel trimethoprim resistance gene, dfrK, in a methicillin-resistant Staphylococcus aureus ST398 strain and its physical linkage to the tetracycline resistance gene tet(L). Kristina Kadlec et al Antimicrob. Agents Chemother. 53, 776-8, (2009)
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Codetection of blaOXA-23-like gene (blaOXA-133) and blaOXA-58 in Acinetobacter radioresistens: report from the SENTRY antimicrobial surveillance program. Rodrigo E Mendes et al Antimicrob. Agents Chemother. 53, 843-4, (2009)
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IncA/C plasmid-mediated florfenicol resistance in the catfish pathogen Edwardsiella ictaluri. Timothy J Welch et al Antimicrob. Agents Chemother. 53, 845-6, (2009)
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Naturally occurring Class A ss-lactamases from the Burkholderia cepacia complex. Laurent Poirel et al Antimicrob. Agents Chemother. 53, 876-82, (2009)
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Pyrosequencing using the single-nucleotide polymorphism protocol for rapid determination of TEM- and SHV-type extended-spectrum beta-lactamases in clinical isolates and identification of the novel beta-lactamase genes blaSHV-48, blaSHV-105, and blaTEM-155. C Hal Jones et al Antimicrob. Agents Chemother. 53, 977-86, (2009)
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Bioactive constituents of the stem bark of Mitrephora glabra. Chen Li et al J. Nat. Prod. 72, 1949-53, (2009)
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Glionitrin A, an antibiotic-antitumor metabolite derived from competitive interaction between abandoned mine microbes. Hyun Bong Park et al J. Nat. Prod. 72, 248-52, (2009)
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Limazepines A-F, pyrrolo[1,4]benzodiazepine Antibiotics from an Indonesian Micrococcus sp. Serge Fotso et al J. Nat. Prod. 72, 690-5, (2009)
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Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination. Manthena V S Varma et al J. Med. Chem. 53, 1098-108, (2010)
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Antimicrobial selaginellin derivatives from Selaginella pulvinata. Yuan Cao et al Bioorg. Med. Chem. Lett. 20, 2456-60, (2010)
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Synthesis and antimicrobial activity of novel fluorine containing 4-(substituted-2-hydroxybenzoyl)-1H-pyrazoles and pyrazolyl benzo[d]oxazoles. Amol V Gadakh et al Bioorg. Med. Chem. Lett. 20, 5572-6, (2010)
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Bernthsen synthesis, antimicrobial activities and cytotoxicity of acridine derivatives. Mehul M Patel et al Bioorg. Med. Chem. Lett. 20, 6324-6, (2010)
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Bromophenols as Candida albicans isocitrate lyase inhibitors. Ki-Bong Oh et al Bioorg. Med. Chem. Lett. 20, 6644-8, (2010)
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Synthetic analogs of indole-containing natural products as inhibitors of sortase A and isocitrate lyase. Lee, Y.-J.; et al. Bioorg. Med. Chem. Lett. 20, 6882, (2010)
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Efflux-mediated bis-indole resistance in Staphylococcus aureus reveals differential substrate specificities for MepA and MepR. Timothy J Opperman et al Bioorg. Med. Chem. 18, 2123-30, (2010)
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Synthesis, anticonvulsant and antimicrobial activities of some new 2-acetylnaphthalene derivatives. Arzu Karakurt et al Bioorg. Med. Chem. 18, 2902-11, (2010)
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Novel 4-thiazolidinone derivatives as potential antifungal and antibacterial drugs. Kouatli Omar et al Bioorg. Med. Chem. 18, 426-32, (2010)
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Novel antimicrobial peptides that exhibit activity against select agents and other drug resistant bacteria. Divakaramenon Venugopal et al Bioorg. Med. Chem. 18, 5137-47, (2010)
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Identification of novel bacterial histidine biosynthesis inhibitors using docking, ensemble rescoring, and whole-cell assays. S T Henriksen et al Bioorg. Med. Chem. 18, 5148-56, (2010)
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The chemical synthesis and antibiotic activity of a diverse library of 2-aminobenzimidazole small molecules against MRSA and multidrug-resistant A. baumannii. Robert W Huigens et al Bioorg. Med. Chem. 18, 663-74, (2010)
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Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species. Denis Fourches et al Chem. Res. Toxicol. 23, 171-83, (2010)
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Antimicrobial study of newly synthesized 6-substituted indolo[1,2-c]quinazolines. Rondla Rohini et al Eur. J. Med. Chem. 45, 1200-5, (2010)
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Synthesis and antimicrobial activities of some new thiazole and pyrazole derivatives based on 4,5,6,7-tetrahydrobenzothiophene moiety. M A Gouda et al Eur. J. Med. Chem. 45, 1338-45, (2010)
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An eco-friendly synthesis and antimicrobial activities of dihydro-2H-benzo- and naphtho-1,3-oxazine derivatives. Bijoy P Mathew et al Eur. J. Med. Chem. 45, 1502-7, (2010)
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Synthesis and study of some new 1,3-isoindoledione derivatives as potential antibacterial agents. A M Khalil et al Eur. J. Med. Chem. 45, 1552-9, (2010)
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Synthesis and antimicrobial of new anthraquinone derivatives incorporating pyrazole moiety. M A Gouda et al Eur. J. Med. Chem. 45, 1843-8, (2010)
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Synthesis, spectroscopic and biological studies on the new symmetric Schiff base derived from 2,6-diformyl-4-methylphenol with N-aminopyrimidine. Mehmet Sönmez et al Eur. J. Med. Chem. 45, 1935-40, (2010)
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Design, synthesis, characterization, and antibacterial activity of {5-chloro-2-[(3-substitutedphenyl-1,2,4-oxadiazol-5-yl)-methoxy]-phenyl}-(phenyl)-methanones. Neithnadka Premsai Rai et al Eur. J. Med. Chem. 45, 2677-82, (2010)
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New 6-amino-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazines and [1,2,4]triazolo[3,4-b] [1,3,4]thiadiazin-6-ones: synthesis, characterization and antibacterial activity evaluation. Gabriela Laura Almajan et al Eur. J. Med. Chem. 45, 3191-5, (2010)
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Synthesis, antibacterial activity evaluation and QSAR studies of novel dispiropyrrolidines. K Karthikeyan et al Eur. J. Med. Chem. 45, 3446-52, (2010)
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Synthesis, characterization, in vitro and molecular docking studies of new 2,5-dichloro thienyl substituted thiazole derivatives for antimicrobial properties. Balladka Kunhanna Sarojini et al Eur. J. Med. Chem. 45, 3490-6, (2010)
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Synthesis of substituted thieno[2,3-d]pyrimidine-2,4-dithiones and their S-glycoside analogues as potential antiviral and antibacterial agents. Hend N Hafez et al Eur. J. Med. Chem. 45, 4026-34, (2010)
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A study of cytotoxicity of novel chlorokojic acid derivatives with their antimicrobial and antiviral activities M. D. Aytemir and B. Oezcelik, Eur. J. Med. Chem. 45, 4089-4095, (2010)
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Pharmacological evaluation and characterizations of newly synthesized 1,2,4-triazoles. Navin B Patel et al Eur. J. Med. Chem. 45, 4293-9, (2010)
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Synthesis of some 3-substituted amino-4,5-tetramethylene thieno[2,3-d][ 1,2,3]-triazin-4(3H)-ones as potential antimicrobial agents. Janardhanan Saravanan et al Eur. J. Med. Chem. 45, 4365-9, (2010)
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Cyclization of some carbothioamide derivatives containing antipyrine and triazole moieties and investigation of their antimicrobial activities. Hacer Bayrak et al Eur. J. Med. Chem. 45, 4726-32, (2010)
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Synthesis, antimicrobial and anti-inflammatory activities of novel 5-(1-adamantyl)-1,3,4-thiadiazole derivatives. Adnan A Kadi et al Eur. J. Med. Chem. 45, 5006-11, (2010)
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Design, synthesis and in vitro evaluation of antitubercular and antimicrobial activity of some novel pyranopyrimidines. Nimesh R Kamdar et al Eur. J. Med. Chem. 45, 5056-63, (2010)
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Synthesis of some new S-triazine based chalcones and their derivatives as potent antimicrobial agents. Anjani Solankee et al Eur. J. Med. Chem. 45, 510-8, (2010)
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Synthesis of new pyrrolo[2,3-d]pyrimidine derivatives as antibacterial and antifungal agents. Khalid Mohammed Hassan Hilmy et al Eur. J. Med. Chem. 45, 5243-50, (2010)
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Synthesis and biological evaluation of some thiazolylpyrazole derivatives as dual anti-inflammatory antimicrobial agents. Adnan A Bekhit et al Eur. J. Med. Chem. 45, 6027-38, (2010)
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Synthesis and antimicrobial evaluation of some fused heterocyclic [1,2,4]triazolo[3,4-b][1,3,4]thiadiazole derivatives. Gabriela Laura Almajan et al Eur. J. Med. Chem. 45, 6139-46, (2010)
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Neural computational prediction of oral drug absorption based on CODES 2D descriptors. A Guerra et al Eur. J. Med. Chem. 45, 930-40, (2010)
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Single nucleotide polymorphism analysis of the major tripartite multidrug efflux pump of Escherichia coli: functional conservation in disparate animal reservoirs despite exposure to antimicrobial chemotherapy. Christopher A Elkins et al Antimicrob. Agents Chemother. 54, 1007-15, (2010)
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Antimicrobial susceptibilities of multidrug-resistant Campylobacter jejuni and C. coli strains: in vitro activities of 20 antimicrobial agents. Mirva Lehtopolku et al Antimicrob. Agents Chemother. 54, 1232-6, (2010)
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Penicillin sulfone inhibitors of class D beta-lactamases. Sarah M Drawz et al Antimicrob. Agents Chemother. 54, 1414-24, (2010)
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Haemophilus influenzae clinical isolates with plasmid pB1000 bearing blaROB-1: fitness cost and interspecies dissemination. Alvaro San Millan et al Antimicrob. Agents Chemother. 54, 1506-11, (2010)
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Genetic and biochemical characterization of TRU-1, the endogenous class C beta-lactamase from Aeromonas enteropelogenes. Filomena De Luca et al Antimicrob. Agents Chemother. 54, 1547-54, (2010)
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Proteus mirabilis pmrI, an RppA-regulated gene necessary for polymyxin B resistance, biofilm formation, and urothelial cell invasion. Sin-Sien Jiang et al Antimicrob. Agents Chemother. 54, 1564-71, (2010)
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PER-6, an extended-spectrum beta-lactamase from Aeromonas allosaccharophila. Delphine Girlich et al Antimicrob. Agents Chemother. 54, 1619-22, (2010)
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Transfer of plasmid-mediated CTX-M-9 from Salmonella enterica serotype Virchow to Enterobacteriaceae in human flora-associated rats treated with cefixime. S Faure et al Antimicrob. Agents Chemother. 54, 164-9, (2010)
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Kinetic parameters of efflux of penicillins by the multidrug efflux transporter AcrAB-TolC of Escherichia coli. Siew Ping Lim et al Antimicrob. Agents Chemother. 54, 1800-6, (2010)
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Genetic basis of multidrug resistance in Acinetobacter clinical isolates in Taiwan. Yu-Chi Lin et al Antimicrob. Agents Chemother. 54, 2078-84, (2010)
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KPC-producing extreme drug-resistant Klebsiella pneumoniae isolate from a patient with diabetes mellitus and chronic renal failure on hemodialysis in South Korea. Ji-Young Rhee et al Antimicrob. Agents Chemother. 54, 2278-9, (2010)
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Characterization of DIM-1, an integron-encoded metallo-beta-lactamase from a Pseudomonas stutzeri clinical isolate in the Netherlands. Laurent Poirel et al Antimicrob. Agents Chemother. 54, 2420-4, (2010)
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Emergence of ciprofloxacin-nonsusceptible Streptococcus pyogenes isolates from healthy children and pediatric patients in Portugal. Renato Pires et al Antimicrob. Agents Chemother. 54, 2677-80, (2010)
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Substrate selectivity and a novel role in inhibitor discrimination by residue 237 in the KPC-2 beta-lactamase. Krisztina M Papp-Wallace et al Antimicrob. Agents Chemother. 54, 2867-77, (2010)
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Antimicrobial resistance among respiratory pathogens in Spain: latest data and changes over 11 years (1996-1997 to 2006-2007). Emilio Pérez-Trallero et al Antimicrob. Agents Chemother. 54, 2953-9, (2010)
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In vitro activity of the aminoglycoside antibiotic arbekacin against Acinetobacter baumannii-calcoaceticus isolated from war-wounded patients at Walter Reed Army Medical Center. Michael J Zapor et al Antimicrob. Agents Chemother. 54, 3015-7, (2010)
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Susceptibility of gram-negative pathogens isolated from patients with complicated intra-abdominal infections in the United States, 2007-2008: results of the Study for Monitoring Antimicrobial Resistance Trends (SMART). Daryl J Hoban et al Antimicrob. Agents Chemother. 54, 3031-4, (2010)
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Incidence and antimicrobial susceptibility of Escherichia coli and Klebsiella pneumoniae with extended-spectrum beta-lactamases in community- and hospital-associated intra-abdominal infections in Europe: results of the 2008 Study for Monitoring Antimicrobial Resistance Trends (SMART). Stephen P Hawser et al Antimicrob. Agents Chemother. 54, 3043-6, (2010)
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Novel chromosome-encoded CTX-M-78 beta-lactamase from a Kluyvera georgiana clinical isolate as a putative origin of CTX-M-25 subgroup. María Margarita Rodríguez et al Antimicrob. Agents Chemother. 54, 3070-1, (2010)
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Mutational analysis of VIM-2 reveals an essential determinant for metallo-beta-lactamase stability and folding. Luisa Borgianni et al Antimicrob. Agents Chemother. 54, 3197-204, (2010)
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Novel ambler class A carbapenem-hydrolyzing beta-lactamase from a Pseudomonas fluorescens isolate from the Seine River, Paris, France. Delphine Girlich et al Antimicrob. Agents Chemother. 54, 328-32, (2010)
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Identification of the novel dfrK-carrying transposon Tn559 in a porcine methicillin-susceptible Staphylococcus aureus ST398 strain. Kristina Kadlec et al Antimicrob. Agents Chemother. 54, 3475-7, (2010)
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Extended-spectrum cephalosporinase in Acinetobacter baumannii. José-Manuel Rodríguez-Martínez et al Antimicrob. Agents Chemother. 54, 3484-8, (2010)
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N-acetylcysteine-mediated modulation of bacterial antibiotic susceptibility. Manish Goswami et al Antimicrob. Agents Chemother. 54, 3529-30, (2010)
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Fitness costs and stability of a high-level ciprofloxacin resistance phenotype in Salmonella enterica serotype enteritidis: reduced infectivity associated with decreased expression of Salmonella pathogenicity island 1 genes. Edel O'Regan et al Antimicrob. Agents Chemother. 54, 367-74, (2010)
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Optimized Nile Red efflux assay of AcrAB-TolC multidrug efflux system shows competition between substrates. Jürgen A Bohnert et al Antimicrob. Agents Chemother. 54, 3770-5, (2010)
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Different classes of antibiotics differentially influence shiga toxin production. Colleen Marie McGannon et al Antimicrob. Agents Chemother. 54, 3790-8, (2010)
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In vitro activity of tebipenem, a new oral carbapenem antibiotic, against beta-lactamase-nonproducing, ampicillin-resistant Haemophilus influenzae. Kozue Kishii et al Antimicrob. Agents Chemother. 54, 3970-3, (2010)
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Plasmid-mediated resistance to cephalosporins in Salmonella enterica serovar Typhi. Masatomo Morita et al Antimicrob. Agents Chemother. 54, 3991-2, (2010)
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In vitro antimicrobial activity and mutant prevention concentration of colistin against Acinetobacter baumannii. Yun Cai et al Antimicrob. Agents Chemother. 54, 3998-9, (2010)
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Contribution of BlaA and BlaB beta-lactamases to antibiotic susceptibility of Yersinia enterocolitica biovar 1B. Zachary W Bent et al Antimicrob. Agents Chemother. 54, 4000-2, (2010)
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Prevalence and dissemination of oqxAB in Escherichia coli isolates from animals, farmworkers, and the environment. Jingjing Zhao et al Antimicrob. Agents Chemother. 54, 4219-24, (2010)
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High-resolution crystal structure of the subclass B3 metallo-beta-lactamase BJP-1: rational basis for substrate specificity and interaction with sulfonamides. Jean-Denis Docquier et al Antimicrob. Agents Chemother. 54, 4343-51, (2010)
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Origin and molecular evolution of the determinant of methicillin resistance in staphylococci. Sae Tsubakishita et al Antimicrob. Agents Chemother. 54, 4352-9, (2010)
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The ABC transporter AnrAB contributes to the innate resistance of Listeria monocytogenes to nisin, bacitracin, and various beta-lactam antibiotics. Barry Collins et al Antimicrob. Agents Chemother. 54, 4416-23, (2010)
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ampG gene of Pseudomonas aeruginosa and its role in ?-lactamase expression. Ying Zhang et al Antimicrob. Agents Chemother. 54, 4772-9, (2010)
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Comparative biochemical and computational study of the role of naturally occurring mutations at Ambler positions 104 and 170 in GES ?-lactamases. Stathis D Kotsakis et al Antimicrob. Agents Chemother. 54, 4864-71, (2010)
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A mecA-negative strain of methicillin-resistant Staphylococcus aureus with high-level ?-lactam resistance contains mutations in three genes. Ritu Banerjee et al Antimicrob. Agents Chemother. 54, 4900-2, (2010)
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Antimicrobial resistance testing of verocytotoxin-producing Escherichia coli and first description of TEM-52 extended-spectrum ?-lactamase in serogroup O26. Glenn Buvens et al Antimicrob. Agents Chemother. 54, 4907-9, (2010)
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In vivo selection of a missense mutation in adeR and conversion of the novel blaOXA-164 gene into blaOXA-58 in carbapenem-resistant Acinetobacter baumannii isolates from a hospitalized patient. Paul G Higgins et al Antimicrob. Agents Chemother. 54, 5021-7, (2010)
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Interplay between drug efflux and antioxidants in Escherichia coli resistance to antibiotics. Girija Dhamdhere et al Antimicrob. Agents Chemother. 54, 5366-8, (2010)
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Nonclonal emergence of colistin-resistant Klebsiella pneumoniae isolates from blood samples in South Korea. Ji-Yoeun Suh et al Antimicrob. Agents Chemother. 54, 560-2, (2010)
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Antimicrobial resistance in Haemophilus influenzae respiratory tract isolates in Korea: results of a nationwide acute respiratory infections surveillance. Songmee Bae et al Antimicrob. Agents Chemother. 54, 65-71, (2010)
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Efficacy of clarithromycin against experimentally induced pneumonia caused by clarithromycin-resistant Haemophilus influenzae in mice. Shigeki Nakamura et al Antimicrob. Agents Chemother. 54, 757-62, (2010)
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Transferable quinolone resistance in Vibrio cholerae. Hong Bin Kim et al Antimicrob. Agents Chemother. 54, 799-803, (2010)
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Inhibitor resistance in the KPC-2 beta-lactamase, a preeminent property of this class A beta-lactamase. Krisztina M Papp-Wallace et al Antimicrob. Agents Chemother. 54, 890-7, (2010)
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Identification of a plasmid-borne resistance gene cluster comprising the resistance genes erm(T), dfrK, and tet(L) in a porcine methicillin-resistant Staphylococcus aureus ST398 strain. Kristina Kadlec et al Antimicrob. Agents Chemother. 54, 915-8, (2010)
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Interaction of ceftobiprole with the low-affinity PBP 5 of Enterococcus faecium. Xavier Henry et al Antimicrob. Agents Chemother. 54, 953-5, (2010)
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Discorhabdins from the Korean marine sponge Sceptrella sp. Ju-Eun Jeon et al J. Nat. Prod. 73, 258-62, (2010)
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Design and synthesis of potent Gram-negative specific LpxC inhibitors. U Faruk Mansoor et al Bioorg. Med. Chem. Lett. 21, 1155-61, (2011)
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Sargachromanols as inhibitors of Na+/K+ ATPase and isocitrate lyase. Soon-Chun Chung et al Bioorg. Med. Chem. Lett. 21, 1958-61, (2011)
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Exploration of antimicrobial and antioxidant potential of newly synthesized 2,3-disubstituted quinazoline-4(3H)-ones. Ashok Kumar et al Bioorg. Med. Chem. Lett. 21, 4353-7, (2011)
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3-[Benzimidazo- and 3-[benzothiadiazoleimidazo-(1,2-c)quinazolin-5-yl]-2H-chromene-2-ones as potent antimicrobial agents. B Suresh Kuarm et al Bioorg. Med. Chem. Lett. 21, 524-7, (2011)
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Microwave assisted synthesis and antimicrobial evaluation of new fused pyran derivatives bearing 2-morpholinoquinoline nucleus. Jigar A Makawana et al Bioorg. Med. Chem. Lett. 21, 6166-9, (2011)
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Synthesis and antimicrobial activity of brominated resorcinol dimers. Elise Bouthenet et al Bioorg. Med. Chem. Lett. 21, 7142-5, (2011)
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A new antifungal briarane diterpenoid from the gorgonian Junceella juncea Pallas. Y L N Murthy et al Bioorg. Med. Chem. Lett. 21, 7522-5, (2011)
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Synthesis and evaluation of anti-tubercular activity of new dithiocarbamate sugar derivatives. Yasuhiro Horita et al Bioorg. Med. Chem. Lett. 21, 899-903, (2011)
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Thiazole-based chalcones as potent antimicrobial agents. Synthesis and biological evaluation. K Liaras et al Bioorg. Med. Chem. 19, 3135-40, (2011)
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Synthesis of some new [1,2,4]triazolo[3,4-b][1,3,4]thiadiazines and [1,2,4]triazolo[3,4-b][1,3,4] thiadiazoles starting from 5-nitro-2-furoic acid and evaluation of their antimicrobial activity. Sahar M I Badr et al Bioorg. Med. Chem. 19, 4506-12, (2011)
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Fragmental modeling of hPepT2 and analysis of its binding features by docking studies and pharmacophore mapping. Alessandro Pedretti et al Bioorg. Med. Chem. 19, 4544-51, (2011)
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Novel benzofuroxan derivatives against multidrug-resistant Staphylococcus aureus strains: design using Topliss' decision tree, synthesis and biological assay. Salomão Dória Jorge et al Bioorg. Med. Chem. 19, 5031-8, (2011)
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Synthesis, molecular modeling and preliminary biological evaluation of a set of 3-acetyl-2,5-disubstituted-2,3-dihydro-1,3,4-oxadiazole as potential antibacterial, anti-Trypanosoma cruzi and antifungal agents. Marina Ishii et al Bioorg. Med. Chem. 19, 6292-301, (2011)
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Novel (E)-1-(4-methyl-2-(alkylamino)thiazol-5-yl)-3-arylprop-2-en-1-ones as potent antimicrobial agents. K Liaras et al Bioorg. Med. Chem. 19, 7349-56, (2011)
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Synthesis, biopharmaceutical characterization, antimicrobial and antioxidant activities of 1-(4'-O-?-D-glucopyranosyloxy-2'-hydroxyphenyl)-3-aryl-propane-1,3-diones. Javed Sheikh et al Eur. J. Med. Chem. 46, 1390-9, (2011)
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Applications of 2-arylhydrazononitriles in synthesis: preparation of new indole containing 1,2,3-triazole, pyrazole and pyrazolo[1,5-a]pyrimidine derivatives and evaluation of their antimicrobial activities. Haider Behbehani et al Eur. J. Med. Chem. 46, 1813-20, (2011)
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Identification of novel potential antibiotics for tuberculosis by in silico structure-based drug screening. Yuya Izumizono et al Eur. J. Med. Chem. 46, 1849-56, (2011)
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Synthesis and antimicrobial activity of thiosemicarbazides, s-triazoles and their Mannich bases bearing 3-chlorophenyl moiety. Tomasz Plech et al Eur. J. Med. Chem. 46, 241-8, (2011)
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Synthesis of 2-aziridinyl phosphonates by modified Gabriel-Cromwell reaction and their antibacterial activities. Özdemir Doğan et al Eur. J. Med. Chem. 46, 2485-9, (2011)
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Synthesis, antitumor and antimicrobial activities of 4-(4-chlorophenyl)-3-cyano-2-(?-O-glycosyloxy)-6-(thien-2-yl)-nicotinonitrile. Hassan A El-Sayed et al Eur. J. Med. Chem. 46, 2948-54, (2011)
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Synthesis and identification of ?-aryloxyquinolines and their pyrano[3,2-c]chromene derivatives as a new class of antimicrobial and antituberculosis agents. Divyesh C Mungra et al Eur. J. Med. Chem. 46, 4192-200, (2011)
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1,3-Dihydro-2H-indol-2-ones derivatives: design, synthesis, in vitro antibacterial, antifungal and antitubercular study. Tarunkumar Nanjibhai Akhaja et al Eur. J. Med. Chem. 46, 5573-9, (2011)
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Synthesis and structure-activity relationship of 2-thiopyrimidine-4-one analogs as antimicrobial and anticancer agents. Supaluk Prachayasittikul et al Eur. J. Med. Chem. 46, 738-42, (2011)
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Synthesis of 4H-chromene, coumarin, 12H-chromeno[2,3-d]pyrimidine derivatives and some of their antimicrobial and cytotoxicity activities. Nermien M Sabry et al Eur. J. Med. Chem. 46, 765-72, (2011)
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Genetic context and biochemical characterization of the IMP-18 metallo-beta-lactamase identified in a Pseudomonas aeruginosa isolate from the United States. Luisa Borgianni et al Antimicrob. Agents Chemother. 55, 140-5, (2011)
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Roles of residues Cys69, Asn104, Phe160, Gly232, Ser237, and Asp240 in extended-spectrum beta-lactamase Toho-1. Akiko Shimizu-Ibuka et al Antimicrob. Agents Chemother. 55, 284-90, (2011)
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Inhibition of bacterial multidrug resistance by celecoxib, a cyclooxygenase-2 inhibitor. Arunasree M Kalle et al Antimicrob. Agents Chemother. 55, 439-42, (2011)
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Verrucamides A-D, antibacterial cyclopeptides from Myrothecium verrucaria. Xianwei Zou et al J. Nat. Prod. 74, 1111-6, (2011)
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Sesterterpenes from the tropical sponge Coscinoderma sp. Jaemin Bae et al J. Nat. Prod. 74, 1805-11, (2011)
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Biologically active arborinane-type triterpenoids and anthraquinones from Rubia yunnanensis. Jun-Ting Fan et al J. Nat. Prod. 74, 2069-80, (2011)
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In Vitro Antibacterial Activity of Sphaeropsidins and Chemical Derivatives toward Xanthomonas oryzae pv. oryzae, the Causal Agent of Rice Bacterial Blight. Antonio Evidente et al J. Nat. Prod. 74, 2520-5, (2011)
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Comazaphilones A-F, azaphilone derivatives from the marine sediment-derived fungus Penicillium commune QSD-17. Shu-Shan Gao et al J. Nat. Prod. 74, 256-61, (2011)
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Antimicrobial isopropenyl-dihydrofuranoisoflavones from Crotalaria lachnophora. Maurice Ducret Awouafack et al J. Nat. Prod. 74, 272-8, (2011)
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N-hydroxypyridones, phenylhydrazones, and a quinazolinone from Isaria farinosa. Cheng Ma et al J. Nat. Prod. 74, 32-7, (2011)
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Scalarane sesterterpenes from the sponge Hyatella sp. Ju-eun Jeon et al J. Nat. Prod. 74, 847-51, (2011)
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Translating Clinical Findings into Knowledge in Drug Safety Evaluation - Drug Induced Liver Injury Prediction System (DILIps). Zhichao Liu et al PLoS Comput. Biol. 7, e1002310, (2011)
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Bioactive lipids from the sponge Spirastrella abata. Kyoung Hwa Jang et al Bioorg. Med. Chem. Lett. 22, 1078-81, (2012)
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Synthesis of novel sulfonamide-1,2,4-triazoles, 1,3,4-thiadiazoles and 1,3,4-oxadiazoles, as potential antibacterial and antifungal agents. Biological evaluation and conformational analysis studies. P Zoumpoulakis et al Bioorg. Med. Chem. 20, 1569-83, (2012)
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Studies on the synthesis and antibacterial activity of 3,6-disubstituted 1,2,4-triazolo[3,4-b]1,3,4-thiadiazoles. Tomasz Plech et al Eur. J. Med. Chem. 47, 580-4, (2012)
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Synthesis and evaluation of anti-tubercular and antibacterial activities of new 4-(2,6-dichlorobenzyloxy)phenyl thiazole, oxazole and imidazole derivatives. Part 2. Xiaoyun Lu et al Eur. J. Med. Chem. 49C, 164-71, (2012)
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Merck 14,586
Corp MSDS 1 (1), 247:A / RegBook 1 (2), 2065:H / Sax 6, 201 / Sigma FT-IR 1 (1), 619:A / Structure Index 1, 328:A:3