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P2278 Sigma

1,3-Dimethyl-8-phenylxanthine

crystalline

Synonym: 8-Phenyltheophylline

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Properties

Related Categories Adenosines/P2 Nucleotide Receptor - Antagonists, Adenosines/P2 Nucleotide Receptors (Purinergics), Antagonists, Bioactive Small Molecule Alphabetical Index, Bioactive Small Molecules,
InChI Key   PJFMAVHETLRJHJ-UHFFFAOYSA-N
form   crystalline
potency   86 nM Ki for A1 receptors
color   off-white to light yellow
mp   >300 °C(lit.)
solubility   H2O: slightly soluble
  aqueous base: moderately soluble (Solutions should be stored at 4 °C.)
  ethanol: moderately soluble (Solutions should be stored at 4 °C.)
Gene Information   human ... ADORA1(134), ADORA2B(136), ADORA3(140)
rat ... Adora1(29290), Adora2a(25369), Adora2b(29316)

Description

Biochem/physiol Actions

Selective A1 adenosine receptor antagonist.

Packaging

1 g in glass bottle

100 mg in glass bottle

Features and Benefits

This compound is also offered as part of Sigma′s Library of Pharmacologically Active Compounds (LOPAC®1280), a biologically annotated collection of high-quality, ready-to-screen compounds. Click here to learn more.

Legal Information

LOPAC is a registered trademark of Sigma-Aldrich Co. LLC

Price and Availability


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Safety & Documentation

Safety Information

RIDADR 
NONH for all modes of transport
WGK Germany 
3
RTECS 
UO8445700
Protocols & Articles
Peer-Reviewed Papers
15

References

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