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Serotonergics

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Image	Description	Biochem/physiol Actions	solubility	Product #
	(±)-2,5-Dimethoxy-4-bromoamphetamine hydrobromide	Hallucinogenic; 5-HT₂ serotonin receptor agonist.		D7412
	(±)-DOI hydrochloride ≥98% (HPLC), solid	(±)-DOI hydrochloride is a potent and selective 5-HT2 serotonin receptor agonist that crosses the blood-brain barrier, increases dopamine turnover and the treatment with DOI counteracted the expression of the nicotine-induced locomotor and neurochemical sensitization, but had no effect on nicotine-induced behavioral disinhibition. The responses to DOI provide evidence that of these receptors are abundant in the cortex, and show relatively lower levels in hippocampus and cerebellum.	ethanol: 2 mg/mL H₂O: 10 mg/mL	D101
	(R)(−)-DOI hydrochloride ≥98% (HPLC), solid	Potent and selective 5-HT₂ serotonin receptor agonist that crosses the blood-brain barrier; more potent enantiomer of ±-DOI hydrochloride.	ethanol: soluble H₂O: ≥20 mg/mL	D153
	1-(3-Chlorophenyl)piperazine hydrochloride	5-HT_2c serotonin receptor agonist; metabolite of trazodone.		125180
	Ketanserin (+)-tartrate salt >97%, solid	Selective 5-HT₂ serotonin receptor antagonist.	0.1 M HCl: 6 mg/mL DMSO: 52 mg/mL ethanol: 3.3 mg/mL	S006
	Pirenperone >97%, solid	5-HT₂ serotonin receptor antagonist.	0.1 M HCl: 11 mg/mL methanol: 2.5 mg/mL 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 5.0 mg/mL	P126
	S(−)-Cyanopindolol hemifumarate salt solid, ≥98% (HPLC)	5-HT_1A/1B serotonin receptor antagonist; β₃-adrenoceptor antagonist.	DMSO: >10 mg/mL	C238
	SB-206553 hydrochloride hydrate ≥98% (HPLC), solid	Potent 5-HT_2B/5-HT_2C serotonin receptor antagonist.	H₂O: >10 mg/mL	S180
	SB 242084 dihydrochloride hydrate ≥98% (HPLC), solid	Selective 5-HT_2c serotonin receptor antagonist; crosses the blood-brain barrier.	H₂O: ≥20 mg/mL	S8061
	VER-3323 hemifumarate salt >98% (HPLC), solid	5-HT_2C/ 5-HT_2B serotonin receptor agonist.	H₂O: 9 mg/mL, soluble	V1889
	α-Methylserotonin maleate salt ≥98% (HPLC), solid	5-HT₂ serotonin receptor agonist.	H₂O: >10 mg/mL	M110

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