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Others

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Biochem/physiol Actions
CAS Number
Product #
16,17-Epoxy-21-acetoxypregnenolone ≥98% 28444-97-5 E4625
16-Dehydropregnenolone acetate ≥95% 979-02-2 D4875
16-Methylene-17α-hydroxypregnenolone 3-acetate 15369-66-1 M8626
17α-Hydroxypregnenolone 387-79-1 H5002
3α,12α-Dihydroxy-5β-pregnan-20-one 3,12-diacetate 15991-93-2 P5902
3α,21-Dihydroxy-5α-pregnan-20-one ≥95% Positive allosteric modulator of GABAA receptors.
567-02-2 P2016
5α-Pregnan-3α-ol-11,20-dione powder, ≥98% (TLC) Synthetic steroid compound alphaxalone (AFX) - 5α-Pregnan-3α-ol-11,20-dione- is a neurosteroid that directly activates and potentiates GABAA receptor-activated membrane current (IGABA). It acts as a positive allosteric modulator of the GABAA receptor; anesthetic. The alpha subunit subtype of GABAA determines the efficacy, but not the potency, of AFX neuroactive steroid to potentiate IGABA.
P5052
5α-Pregnan-3α-ol-20-one solid Positive allosteric modulator of GABAA chloride channel.
516-54-1 P8887
5α-Pregnan-3β-ol-20-one 3β-acetate ≥98% 906-83-2 P8004
CGP-13501 ≥98% (HPLC), solid Positive allosteric modulator of GABAB receptors.
C0987
CGP-7930 >98% (HPLC), solid Positive allosteric modulator of GABAB receptors.
C0862
Dehydroisoandrosterone 3-sulfate sodium salt dihydrate ≥98%, powder Dehydroisoandrosterone 3-sulfate sodium salt dihydrate is a negative allosteric modulator of GABAA receptors.
78590-17-7 D5297
GS39783 ≥98% (HPLC), powder Positive allosteric modulator of GABAB receptors
G5919
Guvacine hydrochloride ≥97% (NMR), solid GABA uptake inhibitor.
6027-91-4 G007
NCS-356 sodium salt hydrate solid, ≥98% (HPLC) γ-Hydroxybutyrate (GHB) receptor agonist.
430440-66-7 N4034
NCS-382 hydrate solid, ≥98% (HPLC) γ-Hydroxybutyrate (GHB) receptor antagonist; anti­convulsant.
N4159
NO-711 hydrochloride solid, ≥98% (HPLC) Potent and selective GABA uptake inhibitor that crosses the blood-brain barrier.
145645-62-1 N142
Nipecotic acid 98% 498-95-3 211672
Pregnenolone sulfate sodium salt Neurosteroid that antagonizes the GABAA receptor chloride channel.
P162
γ-Hydroxybutyric acid sodium salt Endogenous GABA analog that induces absence-like seizures. It blocks dopamine release by blocking impulse flow in dopaminergic neurons.
502-85-2 H3635

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