Benzofurans

Benzofuran (coumarone), a heterocyclic compound consisting of fused benzene and furan rings, has been identified as a privileged structure in medicinal chemistry. Benzofuran derviatives have shown biological activities ranging from antifungal and antimicrobial to antagonists for the H3 receptor and angiotensin II. A diversity of synthetic routes can be applied to the synthesis of benzofurans. The presence of a halogen allows these reagents to be used as substrates in various coupling reactions, including Suzuki-Miyaura cross-coupling reactions.

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New Reagents for Selective Metalation, Deprotonation, and Additions

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CDS016824 3-bromo-1-benzofuran AldrichCPR C8H5BrO
761796 5-Bromobenzofuran 97% C8H5BrO
303453 3-Bromo-2-coumaranone 95% C8H5BrO2
647187 5-Bromophthalide 97% C8H5BrO2
CDS014530 5-bromo-2,3-dihydrobenzo[b]furan-7-sulfonyl chloride AldrichCPR C8H6BrClO3S
CDS003452 5-iodo-2,3-dihydrobenzo[b]furan AldrichCPR C8H7IO
CBR01411 2,3-Dihydro-1-benzofuran-3-amine hydrochloride AldrichCPR C8H10ClNO
CDS015785 5-bromo-1-benzofuran-2-carbaldehyde AldrichCPR C9H5BrO2
CDS014745 1-benzofuran-5-carbonyl chloride AldrichCPR C9H5ClO2
CDS006351 5-chlorobenzofuran-2-carboxylic acid AldrichCPR C9H5ClO3
CDS015544 5-bromo-2,3-dihydrobenzo[b]furan-7-carbonyl chloride AldrichCPR C9H6BrClO2
CDS014119 5-bromo-2,3-dihydrobenzo[b]furan-7-carbaldehyde AldrichCPR C9H7BrO2
CDS013862 7-bromo-2,3-dihydro-1-benzofuran-5-carbaldehyde AldrichCPR C9H7BrO2
CDS015015 5-bromo-2,3-dihydrobenzofuran-7-carboxylic acid AldrichCPR C9H7BrO3
CDS014415 2,3-dihydro-1-benzofuran-5-carbonyl chloride AldrichCPR C9H7ClO2
CBR00813 (2-Methyl-1-benzofuran-7-yl)amine hydrochloride AldrichCPR C9H10ClNO
CBR00712 (2-Methyl-2,3-dihydro-1-benzofuran-5-yl)amine hydrobromide AldrichCPR C9H12BrNO
CDS016941 1-(1-benzofuran-5-yl)-2-bromo-1-ethanone AldrichCPR C10H7BrO2
CDS000927 1-(5-Bromo-1-benzofuran-2-yl)ethanone AldrichCPR C10H7BrO2
CDS010818 5-bromo-3-methyl-1-benzofuran-2-carboxylic acid AldrichCPR C10H7BrO3
CBR00224 5-Bromo-7-methoxy-1-benzofuran-2-carboxylic acid AldrichCPR C10H7BrO4
CDS011618 5-chloro-3-methyl-benzofuran-2-carboxylic acid AldrichCPR C10H7ClO3
CDS011454 7-chloro-3-methylbenzofuran-2-carboxylic acid AldrichCPR C10H7ClO3
CDS010624 5-fluoro-3-methyl-1-benzofuran-2-carboxylic acid AldrichCPR C10H7FO3
CDS012516 2-bromo-1-(2,3-dihydro-1-benzofuran-5-yl)ethanone AldrichCPR C10H9BrO2
CDS002610 2-Methyl-2,3-dihydro-1-benzofuran-5-carbonyl chloride AldrichCPR C10H9ClO2
CDS019204 1-(5-Chloro-benzofuran-2-yl)-ethylamine AldrichCPR C10H10ClNO
CDS017733 1-(5-bromo-7-methoxy-1-benzofuran-2-yl)-1-ethanone AldrichCPR C11H9BrO3
CDS009805 (5-chloro-6-methyl-1-benzofuran-3-yl)acetic acid AldrichCPR C11H9ClO3
CDS009809 7-chloro-3,5-dimethyl-2-benzofurancarboxylic acid AldrichCPR C11H9ClO3
748536 Ethyl 5-chlorobenzofuran-3-carboxylate 95% C11H9ClO3
768472 4-Bromodibenzofuran 97% C12H7BrO
CDS014029 2-(2,3-dihydro-1-benzofuran-5-yl)thiazole-4-carbonyl chloride AldrichCPR C12H8ClNO2S
550132 3-Amino-2-(4-bromobenzoyl)-6-nitrobenzofuran 97% C15H9BrN2O4
550159 3-Amino-2-(4-chlorobenzoyl)-6-nitrobenzofuran 97% C15H9ClN2O4
CDS018493 2-(4-chlorobenzoyl)-1-benzofuran-5-carbaldehyde AldrichCPR C16H9ClO3