Didoron Esters

 
ChemFilesTitle Vol. 2, No. 1
Products for Suzuki Coupling

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Introduction / Boronic Acids / Boronic Acids Esters / Diboron Esters / Prolines & Pyroglutamates
Transition-Metal Catalysts / Palladium Scavengers / Large-Scale Suzuki Coupling / Reference Books

Diboron Esters

The following diboron esters are versatile reagents that couple with organic triflates2 and halides3 to give the corresponding boronic esters, which are readily converted to arylboronic acids. This route and the subsequent Suzuki coupling reaction can be run under mild conditions, thus permitting the use of cyano-,ester-, carbonyl-, and nitro-substituted aryl rings. The wide variety of arylboronic acids available via these diboron esters also makes this class of compounds suitable for solid-phase combinatorial studies.4,5

 

51,880-8

C10H20B2O4

1g; 5g

47,328-6

C12H8B2O4

1g; 5g

52,568-5

C12H24B2O4

1g; 5g

47,329-4

C12H24B2O4

1g; 5g

52,716-5

C16H24B2O12

1g; 5g

52,714-9

C20H32B2O4

1g; 5g

52,713-0

C20H32B2O4

1g; 5g

 

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