Vol . 2, No. 4
Unnatural Amino Acids II

The latest Update on New Tools for Drug Discovery
Click here to download PDF version. (688 KB)

 


Introduction / Cyclic Amino Acids / Diamino Acids / ß-Amino Acids and Homo Amino Acids
Alanine Derivatives / Phenylalanine Boronic Acids / Proline and Pyroglutamine Derivatives
Other Amino Acid Building Blocks / Coupling Reagents / Preloaded Resins
Preloaded Resins

Wang Resin
PS crosslinked with 1% DVB
100-200 mesh; *200-400 mesh
~0.4-0.8 mmol/g resin
packages: 1 g, 5 g

Tentagel® S PHB Resin
POE grafted to low crosslinked
PS matrix ; particle size: 90 mm
~0.1-0.3 mmol/g resin
packages: 1 g, 5 g

2-chlorotrityl Resin
PS crosslinked with 1% DVB
100-200 mesh; * 200-400 mesh
~0.6-1.2 mmol/g resin
packages: 1g, 5g

Tentagel® STrt Resin
POE grafted to low crosslinked
PS matrix; particle size: 90 mm
~0.1-0.3 mmol/g resin
packages: 1 g, 5 g

  Wang Resin Tentagel® S PHB Resin 2-Chlorotrityl Resin Tentagel® STrt Resin
  Cat. #   Residue Cat. #   Residue Cat. #   Residue Cat. #  Residue
Ala 47644  Fmoc-Ala- 86367  Fmoc-Ala- 80929  H-Ala- 86408  Fmoc-Ala-
Arg 47362  Fmoc-Arg(Pbf)-
47665  Fmoc-Arg(Pmc)-
86381  Fmoc-Arg(Pbf)-
86369  Fmoc-Arg(Pmc)-
88619  H-Arg(Pbf)-
72859  H-Arg(Pmc)-
86442  Fmoc-Arg(Pbf)-
86411  Fmoc-Arg(Pmc)-
Asn 47388  Fmoc-Asn(Trt)- 86378  Fmoc-Asn(Trt)- 94636  H-Asn(Trt)- 86412  Fmoc-Asn(Trt)-
Asp 47646*  Fmoc-Asp(OtBu)- 86379  Fmoc-Asp(OtBu)- 92368  H-Asp(OtBu)- 86413  Fmoc-Asp(OtBu)-
Cys 47613*  Fmoc-Cys(Acm)-
47651*  Fmoc-Cys(StBu)-
18606   Fmoc-Cys(Trt)-
86383  Fmoc-Cys(Acm)-
86384  Fmoc-Cys(tBu)-
86385  Fmoc-Cys(S-tBu)-
86386  Fmoc-Cys(Trt)-

90254  H-Cys(Trt)-
86414  Fmoc-Cys(Acm)-
86415  Fmoc-Cys(tBu)-
86416  Fmoc-Cys(S-tBu)-
86417  Fmoc-Cys(Trt)-
Gln 47402   Fmoc-Gln(Trt)- 86388  Fmoc-Gln(Trt)- 95256  H-Gln(Trt)- 86419  Fmoc-Gln(Trt)-
Glu 47658*  Fmoc-Glu(OtBu)- 86389  Fmoc-Glu(OtBu)- 82201  H-Glu(OtBu)- 86421  Fmoc-Glu(tBu)-
Gly 47659*  Fmoc-Gly- 86391  Fmoc-Gly- 92681  H-Gly- 86422  Fmoc-Gly-
His 42237   Fmoc-His(Trt)- 86392  Fmoc-His(Trt)-   86423  Fmoc-His(Trt)-
Ile 47661*  Fmoc-Ile- 86393  Fmoc-Ile- 82914  H-Ile- 86424  Fmoc-Ile-
Leu 47662*  Fmoc-Leu- 86394  Fmoc-Leu- 82938  H-Leu- 86425  Fmoc-Leu-
Lys 47647*  Fmoc-Lys(Boc)- 86395  Fmoc-Lys(Boc)-   86426  Fmoc-Lys(Boc)-
Met 47663*  Fmoc-Met-
47338   Fmoc-D-Met-
86396  Fmoc-Met- 76215  H-Met- 86427  Fmoc-Met-
Phe 7666*   Fmoc-Phe-
47379  Fmoc-D-Phe-
86399  Fmoc-Phe-   86431  Fmoc-Phe-
Pro 47667*  Fmoc-Pro- 86401  Fmoc-Pro- 94077  H-Pro- 86433  Fmoc-Pro-
Ser 47648*  Fmoc-Ser(tBu)-
47403   Fmoc-Ser(Trt)-
86402  Fmoc-Ser(tBu)- 73571  H-Ser(tBu)- 86434  Fmoc-Ser(tBu)-
Thr 47652*  Fmoc-Thr(tBu)- 86403  Fmoc-Thr(tBu)- 72574  H-Thr(tBu)- 86435  Fmoc-Thr(tBu)-
Trp 55606   Fmoc-Trp(Boc)-
47668*  Fmoc-Trp-
86418  Fmoc-Trp(Boc)-
86404  Fmoc-Trp-
80539  H-Trp(Boc)-
86436  Fmoc-Trp-
86443  Fmoc-Trp(Boc)-
47404  Fmoc-D-Trp-
Tyr 47654*  Fmoc-Tyr(tBu)- 86405  Fmoc-Tyr(tBu)- 71025  H-Tyr(tBu)- 86437  Fmoc-Tyr(tBu)-
Val 47669*  Fmoc-Val-
47407   Fmoc-D-Val-
86406  Fmoc-Val- 86557  H-Val- 86438  Fmoc-Val-
*200-400 mesh