Endothelin - Receptor Antagonists

Product #

Image

Product Name

Biochem/physiol Actions

Gene Symbol (ID)

Add to Cart

B150 BQ-123 ≥99%, lyophilized powder Selective ETA endothelin receptor antagonist.
human ... EDNRA(1909), EDNRB(1910)
rat ... Ednra(24326), Ednrb(50672)
B157 BQ-788 ≥95%, solid Selective ETB endothelin receptor antagonist.
human ... EDNRB(1910)
mouse ... EDNRB(13618)
rat ... EDNRB(50672)
J4250 JKC 302 ≥97% (HPLC) JKC-302 may be used as an endothelin receptor (eta) antagonist similar to JKC-301 and other cyclic D-amino acid containing pentapeptides.
 
K1513 Kendomycin from Streptomyces violaceoruber solid Potent endothelin receptor antagonist. Antiosteoporotic compound. Shows also remarkable antibacterial and cytotoxic activity. A putative cellular target for cytotoxicity has been identified: inhibition or altered regulation of the proteasome.
 
PZ0141 PD-156707 ≥98% (HPLC) PD-156707 is a selective endothelin receptor (ETA) antagonist.
 
S6377 Sulfisoxazole ≥99.0% Sulfisoxazole, a sulfonamide, is an antibacterial agent that acts by inhibiting the folic acid metabolism.1 It is also a non-selective endothelin antagonist. It is effective in the treatment of recurrent acute otitis media and also in rendering protection to retina against ischemic-like insults.2,3
rat ... Ednra(24326)