Protein kinase, tyrosine

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121765 AG 825 - CAS 149092-50-2 - Calbiochem A potent, cell-premeable, reversible, substrate competitive, and selective inhibitor of HER2 (neu/ErbB2; IC₅₀ = 0.35 µM) relative to HER1 (IC₅₀= 19 µM) autophosphorylation. C₁₉H₁₅N₃O₃S₂
121767 AG 1024 - CAS 65678-07-1 - Calbiochem A cell-permeable, reversible, substrate competitive, and specific inhibitor of insulin-like growth factor-1 (IGF-1) and insulin receptor tyrosine kinase activity. C₁₄H₁₃BrN₂O
19-123-M Staurosporine Staurosporine Streptomyces is a potent, cell-permeable, reversible, ATP-competitive and broad spectrum inhibitor of protein kinases.  
197221 Bcr-abl Inhibitor - CAS 778270-11-4 - Calbiochem The Bcr-abl Inhibitor, also referenced under CAS 778270-11-4, controls the biological activity of Bcr-abl. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₈H₁₃F₃N₄O₂
197223 Bcr-abl Inhibitor II - CAS 607702-99-8 - Calbiochem The Bcr-abl Inhibitor II, also referenced under CAS 607702-99-8, controls the biological activity of Bcr-abl. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₆H₁₁F₂N₃OS₂
197224 Bcr-abl Inhibitor III, GNF-5 - Calbiochem The Bcr-abl Inhibitor III, GNF-5 controls the biological activity of Bcr-abl. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₀H₁₇F₃N₄O₃
203661-M Bruton's Tyrosine Kinase Inhibitor III - CAS 936563-87-0 - Calbiochem The Bruton's Tyrosine Kinase Inhibitor III, also referenced under CAS 936563-87-0, controls the biological activity of Bruton's Tyrosine Kinase. C₂₅H₂₄N₆O₂
203697 BPDQ - CAS 169205-87-2 - Calbiochem A cell-permeable, reversible, ATP-competitive, potent and specific inhibitor of the tyrosine kinase activity of the epidermal growth factor receptor (EGFR; IC₅₀ = 120 pM). C₁₄H₁₂BrN₅
203987 Butein - CAS 487-52-5 - Calbiochem A cell-permeable, reversible, substrate competitive, plant polyphenol that acts as a specific protein tyrosine kinase inhibitor. C₁₅H₁₂O₅
233100 CL-387,785 - CAS 194423-06-8 - Calbiochem A cell-permeable and irreversible inhibitor of EGF-receptor (EGFR) kinase activity in vivo (IC₅₀ = 250-490 pM) as well as EGF-stimulated autophosphorylation of tyrosine residues in the EGFR in vivo (IC₅₀ = 5 nM). C₁₈H₁₃BrN₄O
234490 PD 153035 - CAS 153436-54-5 - Calbiochem An extremely potent, cell-permeamble, reversible, ATP-competitive and specific inhibitor of the tyrosine kinase activity of the epidermal growth factor receptor (EGFR; IC₅₀ = 25 pM; Ki = 6 pM). C₁₆H₁₄BrN₃O₂
234491 InSolution™ PD 153035 - Calbiochem C₁₆H₁₄BrN₃O₂
234505 Compound 56 - CAS 171745-13-4 - Calbiochem A cell-permeable, reversible, ATP-competitive, highly potent and specific inhibitor of the tyrosine kinase activity of the epidermal growth factor receptor (IC₅₀ = 6 pM). C₁₈H₁₈BrN₃O₂
238590 Cucurbitacin I, Cucumis sativus L. - CAS 2222-07-3 - Calbiochem Cucurbitacin I, Cucumis sativus L., CAS 2222-07-3, is a cell-permeable anti-proliferative agent that acts as a potent and highly selective inhibitor of JAK/STAT3 signaling pathway., A cell-permeable and irreversible bitter triterpenoid compound (NCI identifier: NSC 521777) that displays anti-proliferative and antitumor properties both in vitro and in vivo. C₃₀H₄₂O₇
251600 Daidzein - CAS 486-66-8 - Calbiochem Inactive analog of Genistein. C₁₅H₁₀O₄
251650 Damnacanthal - CAS 477-84-9 - Calbiochem A cell-permeable, potent, reversible, and selective inhibitor of p56lck tyrosine kinase. C₁₆H₁₀O₅
260585 5ʹ-Deoxy-5ʹ-methylthioadenosine - CAS 2457-80-9 - Calbiochem A cell-permeable, reversible, and ATP-competitive naturally-occurring co-product of polyamine biosynthesis that acts as an endogenous substrate of methylthioadenosine phosphorylase (MTAP). C₁₁H₁₅N₅O₃S
324673 EGFR/ErbB-2 Inhibitor - CAS 179248-61-4 - Calbiochem The EGFR/ErbB-2 Inhibitor, also referenced under CAS 179248-61-4, controls the biological activity of EGFR/ErbB-2. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₃H₂₁N₃O₃
324674 EGFR Inhibitor - CAS 879127-07-8 - Calbiochem The EGFR Inhibitor, also referenced under CAS 879127-07-8, controls the biological activity of EGFR. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₁H₁₈F₃N₅O
324694 Emodin - CAS 518-82-1 - Calbiochem A cell-permeable, reversible, substrate competitive and potent p56lck tyrosine kinase inhibitor (IC₅₀ = 18.5 µM). C₁₅H₁₀O₅
324732 ErbB2 Inhibitor II - CAS 928207-02-7 - Calbiochem The ErbB2 Inhibitor II, also referenced under CAS 928207-02-7, controls the biological activity of ErbB2. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₅H₁₀N₄O
324832 EGFR Inhibitor II, BIBX1382 - CAS 196612-93-8 - Calbiochem The EGFR Inhibitor II, BIBX1382, also referenced under CAS 196612-93-8, controls the biological activity of EGFR. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₈H₁₉ClFN₇ • 2HCl • 2H₂O
324833-M EGFR Inhibitor III - CAS 733009-42-2 - Calbiochem The EGFR Inhibitor III, also referenced under CAS 733009-42-2, controls the biological activity of EGFR. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₆H₁₀Cl₃FN₄O
324840 EGFR/ErbB-2/ErbB-4 Inhibitor - CAS 881001-19-0 - Calbiochem The EGFR/ErbB-2/ErbB-4 Inhibitor, also referenced under CAS 881001-19-0, controls the biological activity of EGFR/ErbB-2/ErbB-4. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₇H₁₁ClFN₅O•2.5H₂O
324841-M EGF/FGF/PDGF Receptor Tyrosine Kinase Inhibitor - CAS 1135256-66-4 - Calbiochem The EGF/FGF/PDGF Receptor Tyrosine Kinase Inhibitor controls the biological activity of EGF/FGF/PDGF Receptor Tyrosine Kinase. Primarily used for Phosphorylation & Dephosphorylation applications. C₁₈H₁₈Cl₂N₆O
324842 EGFR/ErbB-2/ErbB-4 Inhibitor II - CAS 944341-54-2 - Calbiochem The EGFR/ErbB-2/ErbB-4 Inhibitor II, also referenced under CAS 944341-54-2, controls the biological activity of EGFR/ErbB-2/ErbB-4. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₄H₂₇ClN₆O₃ • HCl
324877 Focal Adhesion Kinase Inhibitor I - CAS 4506-66-5 - Calbiochem The Focal Adhesion Kinase Inhibitor I, also referenced under CAS 4506-66-5, controls the biological activity of Foca Adhesion Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₆H₁₀N₄ • 4HCl
341607 FGF/VEGF Receptor Tyrosine Kinase Inhibitor, PD173074 - CAS 219580-11-7 - Calbiochem The FGF/VEGF Receptor Tyrosine Kinase Inhibitor, PD173074 controls the biological activity of FGF/VEGF Receptor Tyrosine Kinase. Primarily used for Phosphorylation & Dephosphorylation applications. C₂₈H₄₁N₇O₃
341608 FGF Receptor Tyrosine Kinase Inhibitor - CAS 192705-79-6 - Calbiochem The FGF Receptor Tyrosine Kinase Inhibitor, also referenced under CAS 192705-79-6, controls the biological activity of FGF Receptor Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₀H₂₄N₆O₃
341609 FGF Receptor Tyrosine Kinase Inhibitor IV, NP603 - CAS 949164-80-1 - Calbiochem The FGF Receptor Tyrosine Kinase Inhibitor IV, NP603 controls the biological activity of FGF Receptor Tyrosine KInase. Primarily used for Phosphorylation & Dephosphorylation applications. C₂₆H₂₆N₂O₅
341610 FGF/PDGF/VEGF RTK Inhibitor - CAS 144335-37-5 - Calbiochem The FGF/PDGF/VEGF RTK Inhibitor, also referenced under CAS 144335-37-5, controls the biological activity of FGF/PDGF/VEGF RTK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₆H₁₁N₃O₂
343020 Flt-3 Inhibitor - CAS 301305-73-7 - Calbiochem The Flt-3 Inhibitor, also referenced under CAS 301305-73-7, controls the biological activity of Flt-3. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₈H₂₀N₂O₄S
343021 Flt-3 Inhibitor II - CAS 896138-40-2 - Calbiochem The Flt-3 Inhibitor II, also referenced under CAS 896138-40-2, controls the biological activity of Flt-3. C₁₇H₁₂N₂O₃
343022 Flt-3 Inhibitor III - CAS 852045-46-6 - Calbiochem The Flt-3 Inhibitor III, also referenced under CAS 852045-46-6, controls the biological activity of Flt-3. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₁H₂₃N₃OS
343023 Flt3 Inhibitor IV - CAS 819058-89-4 - Calbiochem The Flt3 Inhibitor IV, also referenced under CAS 819058-89-4, controls the biological activity of Flt3. C₁₃H₁₂N₄
344036-M cFMS Receptor Tyrosine Kinase Inhibitor - CAS 870483-87-7 - Calbiochem The cFMS Receptor Tyrosine Kinase Inhibitor, also referenced under CAS 870483-87-7, controls the biological activity of cFMS. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₀H₂₂N₄O₃
344037 cFMS Receptor Inhibitor II - CAS 959860-85-6 - Calbiochem The cFMS Receptor Inhibitor II, also referenced under CAS 959860-85-6, controls the biological activity of cFMS. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₃H₂₀N₄O
344038 cFMS Receptor Inhibitor III - CAS 959861-21-3 - Calbiochem The cFMS Receptor Inhibitor III, also referenced under CAS 959861-21-3, controls the biological activity of cFMS. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₅H₂₃N₃O₃S
344039 cFMS Receptor Inhibitor IV - CAS 959626-45-0 - Calbiochem The cFMS Receptor Inhibitor IV, also referenced under CAS 959626-45-0, controls the biological activity of cFMS. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₂H₂₆N₄O₂
344041 InSolution™ cFMS Receptor Tyrosine Kinase Inhibitor - Calbiochem The InSolution™ cFMS Receptor Tyrosine Kinase Inhibitor controls the biological activity of cFMS Receptor Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₀H₂₂N₄O₃
345805 Geldanamycin, Streptomyces hygroscopicus - CAS 30562-34-6 - Calbiochem A benzoquinoid antibiotic that inhibits p60c-src tyrosine kinase and c-myc gene expression in murine lymphoblastoma cells. C₂₉H₄₀N₂O₉
345834 Genistein, Soybean - CAS 446-72-0 - Calbiochem A cell-permeable, reversible, substrate competitive inhibitor of protein tyrosine kinases, including autophosphorylation of epidermal growth factor receptor kinase (IC₅₀ = 2.6 µM). C₁₅H₁₀O₅
345836 Genistin - CAS 529-59-9 - Calbiochem An isoflavone glycoside found in soy-based food products. C₂₁H₂₀O₁₀
371806 GTP-14564 - CAS 34823-86-4 - Calbiochem A cell-permeable, reversible, and ATP-competitive tricyclic benzofurano-indazolo compound that acts as a potent and specific inhibitor of class III receptor tyrosine kinases. C₁₅H₁₀N₂O
375670 Herbimycin A, Streptomyces sp. - CAS 70563-58-5 - Calbiochem A potent and cell-permeable protein tyrosine kinase inhibitor. C₃₀H₄₂N₂O₉
397100 HNMPA-(AM)₃ - CAS 120944-03-8 - Calbiochem A cell-permeable analog of HNMPA that yields the parent compound upon cleavage by cytosolic esterases. C₂₀H₂₃O₁₀P
402087 7BIO - CAS 916440-85-2 - Calbiochem A cell-permeable 6-BIO structural isomer that acts as an ATP-competitive inhibitor of Flt3 and a caspase-independent, non-apoptotic cell death inducer. C₁₆H₁₀BrN₃O₂
407247 IGF-1R Inhibitor, PPP - CAS 477-47-4 - Calbiochem IGF-1R Inhibitor, PPP, CAS 477-47-4, is a cell-permeable, substrate competitive, reversible, potent, and specific inhibitor of IGF-1R both in vitro (IC50 = 1 nM in cell-free kinase assay) & in vivo., The IGF-1R Inhibitor, PPP, also referenced under CAS 477-47-4, controls the biological activity of IGF-1R. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₂H₂₂O₈
407248 IGF-1R Inhibitor II, PQ401 - CAS 196868-63-0 - Calbiochem The IGF-1R Inhibitor II, also referenced under CAS 196868-63-0, controls the biological activity of IGF-1R. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₈H₁₆ClN₃O₂
420139 JAK2 Inhibitor IV - CAS 1110502-30-1 - Calbiochem The JAK2 Inhibitor IV, also referenced under CAS 1110502-30-1, controls the biological activity of JAK2. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₇H₂₀N₄O₂S
428150 Lavendustin A - CAS 125697-92-9 - Calbiochem A cell-permeable, reversible, and substrate competitive inhibitor of EGF receptor tyrosine kinase and p60c-src with little effect on protein kinase A or protein kinase C. C₂₁H₁₉NO₆
428201 LDN-211904 - Calbiochem LDN-211904 modulates the biological activity of EphB3 receptor tyrosine kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₁H₂₁ClN₄O₅
428205-M Lck Inhibitor - CAS 213743-31-8 - Calbiochem The Lck Inhibitor, also referenced under CAS 213743-31-8, controls the biological activity of Lck. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₃H₂₂N₄O
428206 Lck Inhibitor II - CAS 918870-43-6 - Calbiochem The Lck Inhibitor II, also referenced under CAS 918870-43-6, controls the biological activity of Lck. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₄H₂₆N₆O₃
428207 Lck Inhibitor III - CAS 1188890-30-3 - Calbiochem The Lck Inhibitor III, also referenced under CAS 1188890-30-3, controls the biological activity of Lck. C₂₅H₂₈N₆O₃ • H₂O
435300 LFM-A13 - CAS 62004-35-7 - Calbiochem A potent, cell-permeable, reversible, substrate competitive, and specific inhibitor of Bruton's Tyrosine Kinase (BTK; IC₅₀ = 17.2 µM for human BTK in vitro and IC₅₀ = 2.5 µM for recombinant BTK). C₁₁H₈Br₂N₂O₂
445835-M Mer RTK Inhibitor, UNC569 - Calbiochem Mer RTK Inhibitor, UNC569, 1350547-65-7 is a potent, reversible and ATP-competitive inhibitor of Mer receptor tyrosine kinase (IC50 = 2.9 nM; Ki = 4.3 nM). C₂₂H₂₉FN₆
448101 Met Kinase Inhibitor - CAS 658084-23-2 - Calbiochem The Met Kinase Inhibitor, also referenced under CAS 658084-23-2, controls the biological activity of Met Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₈H₃₀ClN₅O₄S
448103 Met/Flt-3/VEGFR2 Tyrosine Kinase Inhibitor - CAS 888719-03-7 - Calbiochem The Met/Flt-3/VEGFR2 Tyrosine Kinase Inhibitor controls the biological activity of Met/Flt-3/VEGFR2 Tyrosine Kinase. Primarily used for Phosphorylation & Dephosphorylation applications. C₂₅H₁₆F₂N₄O₃
448104 c-Met/RON Dual Kinase Inhibitor - CAS 913376-84-8 - Calbiochem The c-Met/RON Dual Kinase Inhibitor, also referenced under CAS 913376-84-8, controls the biological activity of c-Met/RON. C₃₁H₂₉FN₄O₅
448105 c-Met Kinase Inhibitor III - Calbiochem The c-Met Kinase Inhibitor III controls the biological activity of c-Met. C₂₁H₁₇Cl₂FN₂O₂
448106 Met Kinase Inhibitor VI, SGX523 - CAS 1022150-57-7 - Calbiochem The Met Kinase Inhibitor VI, SGX523, also referenced under CAS 1022150-57-7, controls the biological activity of Met Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₈H₁₃N₇S
481909 Niclosamide - CAS 50-65-7 - Calbiochem A salicylanilide anthelmintic drug that acts as a potent and selective Stat3- and Wnt-signaling pathway inhibitor. C₁₃H₈Cl₂N₂O₄
5.04595 Bcr-abl Inhibitor IV, Imatinib - CAS 220127-57-1 - Calbiochem C₂₉H₃₁N₇O • CH₃SO₃H
513001 InSolution™ PD 98059 - CAS 167869-21-8 - Calbiochem InSolution™ PD 98059, CAS 167869-21-8, is a 5 mg/ml solution in DMSO. A a cell-permeable, selective & reversible inhibitor of MAP Kinase Kinase (MEK). C₁₆H₁₃NO₃
513028 PD 166285 - CAS 212391-63-4 - Calbiochem A cell-permeable, orally bioavailable, ATP-competitive, broad-spectrum tyrosine kinase inhibitor that suppresses angiogenesis both in vitro and in vivo. C₂₆H₂₇Cl₂N₅O₂ • 2HCl
513033 PD 168393 - CAS 194423-15-9 - Calbiochem PD 168393, CAS 194423-15-9, is a cell-permeable, potent, selective, irreversible, ATP-competitive inhibitor of EGF receptor (EGFR) tyrosine kinase activity (IC50 = 700 pM)., A potent, cell-permeable, irreversible, ATP-competitive and selective inhibitor of EGF receptor (EGFR) tyrosine kinase activity (IC₅₀ = 700 pM). C₁₇H₁₃BrN₄O
513035 PD 158780 - CAS 171179-06-9 - Calbiochem A potent, cell-permeable, reversible, ATP-competitive inhibitor of the EGFR tyrosine kinase activity (IC₅₀ = 8 pM). C₁₄H₁₂BrN₅
513036 InSolution™ PD 158780 - CAS 171179-06-9 - Calbiochem C₁₄H₁₂BrN₅
513040-M PD 174265 - CAS 216163-53-0 - Calbiochem A potent, cell-permeable, reversible, ATP-competitive and selective inhibitor of EGF receptor (EGFR) tyrosine kinase activity (IC₅₀ = 450 pM). C₁₇H₁₅BrN₄O
521231 PDGFR Tyrosine Kinase Inhibitor II - CAS 249762-74-1 - Calbiochem The PDGFR Tyrosine Kinase Inhibitor II, also referenced under CAS 249762-74-1, controls the biological activity of PDGFR Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₁H₁₈N₂O₃
521232 PDGFR Tyrosine Kinase Inhibitor III - CAS 205254-94-0 - Calbiochem C₂₇H₂₇N₅O₄
521233 PDGFR Tyrosine Kinase Inhibitor IV - CAS 627518-40-5 - Calbiochem C₁₈H₁₆FN₃O₂
521234 PDGFR Tyrosine Kinase Inhibitor V - CAS 347155-76-4 - Calbiochem The PDGFR Tyrosine Kinase Inhibitor V, also referenced under CAS 347155-76-4, controls the biological activity of PDGFR Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₆H₂₃N₃O₄S • 3H₂O
521235 PDGFR Tyrosine Kinase Inhibitor VI, SU6668 - CAS 210644-62-5 - Calbiochem The PDGFR Tyrosine Kinase Inhibitor VI, SU6668, also referenced under CAS 210644-62-5, controls the biological activity of PDGFR Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₈H₁₈N₂O₃
521236 PDGFR/VEGFR2 Tyrosine Kinase Inhibitor, 5-Br SU6668 - CAS 251356-32-8 - Calbiochem The PDGFR/VEGFR2 Tyrosine Kinase Inhibitor, 5-Br SU6668 controls the biological activity of PDGFR/VEGFR2 Tyrosine Kinase. Primarily used for Phosphorylation & Dephosphorylation applications. C₁₈H₁₇BrN₂O₃
521237 PDGFR Tyrosine Kinase Inhibitor VII - CAS 251356-45-3 - Calbiochem The PDGFR Tyrosine Kinase Inhibitor VII, also referenced under CAS 251356-45-3, controls the biological activity of PDGFR Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₄H₂₂N₂O₃
521276 PDK1 Inhibitor II - CAS 850717-64-5 - Calbiochem The PDK1 Inhibitor II, also referenced under CAS 850717-64-5, controls the biological activity of PDK1. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₅H₁₄N₄O₂
527948 Piceatannol - CAS 10083-24-6 - Calbiochem A cell-permeable, substrate competitive and reversible plant metabolite that inhibits the activity of rat liver protein kinase A catalytic subunit (IC₅₀ = 3 µM), PKC (IC₅₀ = 8 µM), MLCK (IC₅₀ = 12 µM). C₁₄H₁₂O₄
529573 PP2 - CAS 172889-27-9 - Calbiochem PP2, CAS 172889-27-9, is a potent, reversible, ATP-competitive, inhibitor of the Src family of protein tyrosine kinases (IC₅₀ = 4, 5, 5, &100 nM for p56lck, p59fynT, Hck, & Src, respectively). C₁₅H₁₆ClN₅
529574 PP3 - CAS 5334-30-5 - Calbiochem PP3, CAS 5334-30-5, is a negative control for the Src family protein tyrosine kinase inhibitor PP2 (Cat. No. 529573). However, it inhibits the activity of EGFR kinase (IC50 = 2.7 µM)., A negative control for the Src family protein tyrosine kinase inhibitor PP2. However, it inhibits the activity of EGFR kinase (IC₅₀ = 2.7 µM). C₁₁H₉N₅
529576 InSolution™ PP2 - Calbiochem InSolution™ PP2, 172889-27-9, is a 10 mM solution of PP2 (Cat. No. 529573) in DMSO. A potent, reversible, ATP-competitive, inhibitor of the Src family of protein tyrosine kinases. C₁₅H₁₆ClN₅
529579 PP1 Analog - CAS 221243-82-9 - Calbiochem C₁₉H₁₉N₅
529581 PP1 Analog II, 1NM-PP1 - CAS 221244-14-0 - Calbiochem PP1 Analog II, CAS 221244-14-0, is a cell-permeable PP1 analog that acts as a potent, reversible, selective, ATP-competitive inhibitor of mutant over wild-type kinases. C₂₀H₂₁N₅
529584 PTK/PI 3-K/mTOR Inhibitor, PP121 - CAS 1092788-83-4 - Calbiochem The PTK/PI 3-K/mTOR Inhibitor, PP121, also referenced under CAS 1092788-83-4, controls the biological activity of PTK/PI 3-K/mTOR. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₇H₁₇N₇
529605-M InSolution™ PP1 Analog - CAS 221243-82-9 - Calbiochem A potent, reversible, ATP-competitive, and cell-permeable inhibitor of Src-family tyrosine kinases that is >800 times more selective for the I338G mutant v-Src compared to wild-type v-Src. C₁₉H₁₉N₅
5.38169 Motesanib, Diphosphate - CAS 857876-30-3 - Calbiochem A cell-permeable, highly potent, ATP-competitive multi-kinase inhibitor (IC₅₀ = 2, 3, 6, 8 nM for VEGFR1, VEGFR2, VEGFR3, and Kit, respectively). C₂₂H₂₃N₅O.2H₃PO₄
539571 InSolution™ Src Inhibitor, PP1 - Calbiochem The InSolution™ Src Inhibitor, PP1 controls the biological activity of Src. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₆H₁₉N₅
539644 UCN-01 A cell-permeable Staurosporine derived anticancer agent that reversibly and ATP-competitively inhibits several protein kinases. C₂₈H₂₆N₄O₄
539648 Staurosporine, N-Benzoyl A cell-permeable Staurosporine derivative that displays antitumor properties. C₃₅H₃₀N₄O₄
553400 Radicicol, Diheterospora chlamydosporia - CAS 12772-57-5 - Calbiochem C₁₈H₁₇ClO₆
567805 Src Kinase Inhibitor I - CAS 179248-59-0 - Calbiochem The Src Kinase Inhibitor I, also referenced under CAS 179248-59-0, controls the biological activity of Src Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₂H₁₉N₃O₃
567806 Src Kinase Inhibitor II - CAS 459848-35-2 - Calbiochem The Src Kinase Inhibitor II, also referenced under CAS 459848-35-2, controls the biological activity of Src Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₂H₂₀N₄O₃S
567809-M Src Inhibitor, PP1 - CAS 172889-26-8 - Calbiochem The Src Inhibitor PP1, also referenced under CAS 172889-26-8, controls the biological activity of Src. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₆H₁₉N₅
569615-M Stem-Cell Factor/c-Kit Inhibitor, ISCK03 - CAS 945526-43-2 - Calbiochem The Stem-Cell Factor/c-Kit Inhibitor, ISCK03, also referenced under CAS 945526-43-2, controls the biological activity of Stem-Cell Factor/c-Kit. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₉H₂₁N₃O₂S
570100 Ste11 MAPKKK Activation Inhibitor - CAS 331662-51-2 - Calbiochem The Ste11 MAPKKK Activation Inhibitor, also referenced under CAS 331662-51-2, controls the biological activity of Ste11 MAPKKK. C₁₆H₁₃Cl₂N₃O₂
572630 SU5402 - CAS 215543-92-3 - Calbiochem SU5402, CAS 215543-92-3, is a cell-permeable, reversible, and ATP-competitive inhibitor of the tyrosine kinase activity of FGFR1 (IC₅₀ = 10-20 µM in the presence of 1 mM ATP). C₁₇H₁₆N₂O₃
572632-M SU5614 - CAS 186611-56-3 - Calbiochem A potent, cell-permeable, reversible, ATP-competitive, and selective inhibitor of VEGF (Flk-1; IC₅₀ = 1.2 µM) and PDGF (IC₅₀ = 2.9 µM) receptor tyrosine kinases. C₁₅H₁₃N₂OCl
572635 SU6656 - CAS 330161-87-0 - Calbiochem SU6656, CAS 330161-87-0, is a cell-permeable, potent, reversible, ATP-competitive inhibitor of Src (IC50 = 280 nM). Also inhibits Fyn (IC50 = 170 nM), Yes (IC50 = 20 nM), and Lyn (IC50 = 130 nM)., A potent, cell-permeable, reversible, and ATP-competitive Src family kinase inhibitor. C₁₉H₂₁N₃O₃S
572636 InSolution™ SU6656 - Calbiochem C₁₉H₂₁N₃O₃S
572660 SU11652 - CAS 326914-10-7 - Calbiochem A cell-permeable pyrrole-indolinone compound that acts as a potent, reversible, and ATP-competitive tyrosine kinase receptor and angiogenic inhibitor. C₂₂H₂₇ClN₄O₂
572888-M SU1498 - Calbiochem SU1498, CAS 168835-82-3, is a potent, reversible, ATP-competitive and selective inhibitor of Flk-1 kinase (IC50 = 700 nM)., A potent, reversible, ATP-competitive and selective inhibitor of Flk-1 kinase (IC₅₀ = 700 nM), a vascular endothelial growth factor (VEGF) receptor kinase. C₂₅H₃₀N₂O₂
574711 Syk Inhibitor - CAS 622387-85-3 - Calbiochem The Spleen Tyrosine Kinase Inhibitor, also referenced under CAS 622387-85-3, controls the biological activity of Spleen Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₈H₁₅N₃O₃S
574712 Syk Inhibitor II - CAS 227449-73-2 - Calbiochem The Syk Inhibitor II, also referenced under CAS 227449-73-2, controls the biological activity of Syk. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₄H₁₅F₃N₆O • 2HCl•2H₂O
574714 Syk Inhibitor IV, BAY 61-3606 - CAS 732938-37-8 - Calbiochem Syk Inhibitor IV, BAY 61-3606, CAS 732938-37-8, is a cell-permeable, potent, ATP-competitive, reversible, and highly selective inhibitor of Syk tyrosine kinase activity (IC50 = 10 nM)., The Syk Inhibitor IV, BAY 61-3606, also referenced under CAS 732938-37-8, controls the biological activity of Syk. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₀H₁₈N₆O₃ • HCl • H₂O
574715 Syk Inhibitor V - Calbiochem The Syk Inhibitor V controls the biological activity of Syk. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₀H₂₃N₅O₂S
581810 (-)-Terreic Acid, Synthetic - CAS 121-40-4 - Calbiochem A cell-permeable quinone epoxide antibiotic that acts as a reversible, substrate competitive, and selective inhibitor of Bruton's tyrosine kinase catalytic activity (BTK; IC₅₀ = 10 µM and 3 µM for the basal and activation levels). C₇H₆O₄
612085 Tie2 Kinase Inhibitor - CAS 948557-43-5 - Calbiochem The Tie2 Kinase Inhibitor, also referenced under CAS 948557-43-5, controls the biological activity of Tie2 Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₆H₂₁N₃O₂S
648450-M TrkA Inhibitor - CAS 388626-12-8 - Calbiochem The TrkA Inhibitor, also referenced under CAS 388626-12-8, controls the biological activity of TrkA. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₅H₁₃N₃O₃S
648451 Trk Inhibitor III, GNF-5837 - CAS 1033769-28-6 - Calbiochem The Trk Inhibitor III, GNF-5837 controls the biological activity of Trk. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₈H₂₁F₄N₅O₂
655200 TX-1123 - CAS 157397-06-3 - Calbiochem A cell-permeable, reversible, and substrate-competitive arylidene-cyclopentenedione derived tyrphostin that acts as an inhibitor for Src, eEF2-K, and PKA, and EGFR-K/PKC at much higher concentrations. C₂₀H₂₄O₃
657021 Tyrosine Kinase Inhibitor Set II - Calbiochem The Tyrosine Kinase Inhibitor Set II controls the biological activity of Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.  
658390 AG 9 - CAS 2826-26-8 - Calbiochem An inactive compound that can be used as a negative control for inhibition of EGFR (IC₅₀ >1250 µM for EGFR kinase). C₁₁H₈N₂O
658395 AG 18 - CAS 118409-57-7 - Calbiochem A broad-spectrum protein tyrosine kinase inhibitor. C₁₀H₆N₂O₂
658400 AG 82 - CAS 118409-58-8 - Calbiochem A cell-permeable, reversible, and competitive inhibitor of substrate binding on protein tyrosine kinases. C₁₀H₆N₂O₃
658401 AG 490 - CAS 133550-30-8 - Calbiochem A cell-permeable, reversible, substrate competitive, and potent inhibitor of epidermal growth factor receptor kinase autophosphorylation (IC₅₀ = 100 nM). C₁₇H₁₄N₂O₃
658403 AG 538 - CAS 133550-18-2 - Calbiochem A potent, cell-premeable, reversible, and competitive inhibitor of IGF-1 receptor kinase (IC₅₀ = 400 nM). C₁₆H₁N₁₁O₅
658411 InSolution™ AG490 - Calbiochem C₁₇H₁₄N₂O₃
658425 AG 17 - CAS 10537-47-0 - Calbiochem Anti-proliferative agent that acts as a selective inhibitor of the platelet-derived growth factor receptor tyrosine kinase (IC₅₀ = 500 nM). C₁₈H₂₂N₂O
658460 AG 879 - CAS 148741-30-4 - Calbiochem A cell-permeable, reversible, and substrate competitive inhibitor of nerve growth factor (NGF)-dependent p140c-trk tyrosine phosphorylation (EC₅₀ = 10 µM) as well as NGF-induced phospholipase C-γ1 phosphorylation. C₁₈H₂₄N₂OS
658548 InSolution™ AG 1478 - CAS 175178-82-2 - Calbiochem C₁₆H₁₄ClN₃O₂
658550 AG 1295 - CAS 71897-07-9 - Calbiochem A cell-permeable, reversible, ATP-competitive, and selective inhibitor of platelet-derived growth factor (PDGF) receptor kinase (IC₅₀ = 500 nM) and PDGF-dependent DNA synthesis (IC₅₀ = 2.5 µM) in Swiss/3T3 cells. C₁₆H₁₄N₂
658551 AG 1296 - CAS 146535-11-7 - Calbiochem A cell-permeable, reversible, and ATP-competitive, inhibitor of PDGF receptor kinase and blocks signaling of human PDGF α-receptors and β-receptors. C₁₆H₁₄N₂O₂
658552 AG 1478 - CAS 175178-82-2 - Calbiochem AG 1478, CAS 175178-82-2, is a cell-permeable, potent, selective, reversible & ATP-competitive inhibitor of EGF receptor kinase (IC50 = 3 nM vs 100 µM for HER2-neu and PDGF receptor kinase)., A cell-permeable, reversible, ATP-competitive, highly potent and selective inhibitor of epidermal growth factor receptor kinase versus HER2-neu and platelet-derived growth factor receptor kinase. C₁₆H₁₄ClN₃O₂
676480 VEGFR2 Kinase Inhibitor I - CAS 15966-93-5 - Calbiochem The VEGFR2 Kinase Inhibitor I, also referenced under CAS 15966-93-5, controls the biological activity of VEGFR2 Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₈H₁₈N₂O₃
676481 VEGFR Tyrosine Kinase Inhibitor II - CAS 269390-69-4 - Calbiochem The VEGFR Tyrosine Kinase Inhibitor II, also referenced under CAS 269390-69-4, controls the biological activity of VEGFR Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₉H₁₆ClN₃O
676483 VEGFR Tyrosine Kinase Inhibitor IV - CAS 475108-18-0 - Calbiochem The VEGFR Tyrosine Kinase Inhibitor IV, also referenced under CAS 475108-18-0, controls the biological activity of VEGFR Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₂H₁₉ClN₄O₅ • H₂O
676484 VEGFR2 Kinase Inhibitor VI, Ki8751 - CAS 228559-41-9 - Calbiochem The VEGFR2 Kinase Inhibitor VI, Ki8751, also referenced under CAS 228559-41-9, controls the biological activity of VEGFR2 Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₄H₁₈F₃N₃O₄
676485 VEGFR2 Kinase Inhibitor II - CAS 288144-20-7 - Calbiochem The VEGFR2 Kinase Inhibitor II, also referenced under CAS 288144-20-7, controls the biological activity of VEGFR2 Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₇H₁₅BrN₂O
676487 VEGFR2 Kinase Inhibitor III - CAS 204005-46-9 - Calbiochem The VEGFR2 Kinase Inhibitor III, also referenced under CAS 204005-46-9, controls the biological activity of VEGFR2 Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₅H₁₄N₂O
676492 VEGFR3 Kinase Inhibitor, MAZ51 - CAS 163655-37-6 - Calbiochem VEGFR3 Kinase Inhibitor, MAZ51, CAS 163655-37-6, is a cell-permeable, reversible, ATP-competitive inhibitor of VEGF receptor tyrosine kinase. Blocks VEGF-C & VEGF-D-induced phosphorylation of VEGFR-3., The VEGFR3 Kinase Inhibitor, MAZ51, also referenced under CAS 163655-37-6, controls the biological activity of VEGFR3 Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₁H₁₈N₂O
676493 VEGF Inhibitor, Flt₂₋₁₁ - Calbiochem The VEGF Inhibitor, Flt2-11 controls the biological activity of VEGF. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₆₁H₁₀₄N₁₄O₁₅
676494 VEGF Inhibitor, Je-11 - Calbiochem The VEGF Inhibitor, Je-11 controls the biological activity of VEGF. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₈₈H₂₇₃N₄₉O₅₇
676495 VEGF Inhibitor, V1 - Calbiochem The VEGF Inhibitor, V1 controls the biological activity of VEGF. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₄₀H₆₁N₁₁O₉
676496 VEGF Inhibitor, CBO-P11 - Calbiochem VEGF Inhibitor, CBO-P11, is a macrocyclic peptide derived from residues 79-93 of VEGF. Mediates VEGF binding to VEGFR-2. Blocks VEGF165 binding to VEGFR1 and 2 (IC50 = 700 nM & 1.3 µM, respectively)., The VEGF Inhibitor, CBO-P11 controls the biological activity of VEGF. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₉₀H₁₄₀N₂₈O₂₂S
676500-M VEGFR2/Flt3/c-Kit Inhibitor - CAS 796967-10-7 - Calbiochem The VEGFR2/Flt3/c-Kit Inhibitor, also referenced under CAS 796967-10-7, controls the biological activity of VEGFR2/Flt3/c-Kit. This small molecule/inhibitor is primarily used for Activators/Inducers applications. C₂₁H₁₉N₅O
676501 VEGFR Tyrosine Kinase Inhibitor V - Calbiochem The VEGFR Tyrosine Kinase Inhibitor V controls the biological activity of VEGFR Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₅H₂₂N₂O₄ • HCl • H₂O
676503 VEGFR/Tie-2/PDGFR Tyrosine Kinase Inhibitor - Calbiochem The VEGFR/Tie-2/PDGFR Tyrosine Kinase Inhibitor controls the biological activity of VEGFR/Tie-2/PDGFR. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₂₁H₁₅F₄N₅O₂
676504 VEGFR Tyrosine Kinase Inhibitor VI, AAL-993 - CAS 269390-77-4 - Calbiochem The VEGFR Tyrosine Kinse Inhibitor VI, ALL-993, also referenced under CAS 269390-77-4, controls the biological activity of VEGFR Tyrosine Kinase. This small molecule/inhibitor is primarily used for Cancer applications. C₂₀H₁₆F₃N₃O
676505 VEGFR2 Kinase Inhibitor VII, SKLB1002 - Calbiochem The VEGFR2 Kinase Inhibitor VII, SKLB1002 controls the biological activity of VEGFR2 Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. C₁₃H₁₂N₄O₂S₂
A7410 Amiloride hydrochloride hydrate ≥98% (TLC), powder C6H8ClN7O · HCl · xH2O
C2932 Chelerythrine chloride ≥95% (TLC), powder C21H18ClNO4
D7802 Daidzein ≥98%, synthetic C15H10O4
H6649 Herbimycin A from Streptomyces hygroscopicus ≥95% (HPLC), powder C30H42N2O9
L1289 Lavendustin C ≥97%, solid C14H13NO5