Cyclin-Dependent Kinase (CDK)

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126870 Alsterpaullone - CAS 237430-03-4 - Calbiochem A cell-permeable, potent, reversible, and ATP competitive inhibitor of GSK-3β (IC₅₀ = 4 nM) and Cdk1/cyclin B (IC₅₀ = 35 nM).
126871 Alsterpaullone, 2-Cyanoethyl - CAS 852529-97-0 - Calbiochem A cell-permeable and reversible Alsterpaullone derivative that acts as a highly potent, ATP-competitive, selective inhibitor of Cdk1/cyclin B and GSK-3β.
128125 Aloisine A - CAS 496864-16-5 - Calbiochem A cell-permeable pyrrolo-pyrazine compound that exerts anti-proliferative effects.
164640 Aminopurvalanol A - CAS 220792-57-4 - Calbiochem A cell-permeable 2,6,9-trisubstituted purine analog that displays anti-mitotic as well as anti-tumor properties.
203881 CR8, (R)-Isomer - CAS 294646-77-8 - Calbiochem A cell-permeable (R)-DRF053 analog that acts as an ATP-binding pocket-targeting CDK/CK1 dual-specific inhibitor.
203882-M CR8, (S)-Isomer - CAS 1084893-56-0 - Calbiochem A cell-permeable (R)-DRF053 analog that acts as an ATP-binding pocket-targeting CDK/CK1 dual-specific inhibitor.
203988 Butyrolactone I - CAS 87414-49-1 - Calbiochem A cell-permeable and highly selective inhibitor of cyclin-dependent protein kinases (Cdks) that inhibits cell cycle progression at the G₁/S and G₂/M transitions.
217695 Cdk1 Inhibitor - CAS 220749-41-7 - Calbiochem The Cdk1 Inhibitor, also referenced under CAS 220749-41-7, controls the biological activity of Cdk1. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
217697-M Cdk1 Inhibitor III The Cdk1 Inhibitor III, also referenced under CAS 440362-74-3, controls the biological activity of Cdk1. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
217699 Cdk1 Inhibitor IV, RO-3306 - Calbiochem RO-3306 is a cell-permeable, potent and ATP-competitive inhibitor of Cdk1 (Ki = 35 nM and 110 nM for Cdk1/B1 and Cdk1/A, respectively).
217707 Cdc7/Cdk9 Inhibitor - CAS 845714-00-3 - Calbiochem The Cdc7/Cdk9 Inhibitor, also referenced under CAS 845714-00-3, controls the biological activity of Cdc7/Cdk9. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
217713 Cdk1/2 Inhibitor II, NU6102 - CAS 444722-95-6 - Calbiochem The Cdk1/2 Inhibitor II, NU6102, also referenced under CAS 444722-95-6, controls the biological activity of Cdk1/2. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
217714 Cdk1/2 Inhibitor III - CAS 443798-55-8 - Calbiochem The Cdk1/2 Inhibitor III, also referenced under CAS 443798-55-8, controls the biological activity of Cdk1/2. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
217720 Cdk1/5 Inhibitor - CAS 40254-90-8 - Calbiochem The Cdk1/5 Inhibitor, also referenced under CAS 40254-90-8, controls the biological activity of Cdk1/5. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
217721 InSolution™ Cdk1 Inhibitor IV, RO-3306 - Calbiochem The InSolution™ Cdk1 Inhibitor IV, RO-3306 controls the biological activity of Cdk1. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
219445 Cdk2 Inhibitor II - CAS 222035-13-4 - Calbiochem The Cdk2 Inhibitor II, also referenced under CAS 222035-13-4, controls the biological activity of Cdk2. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
219457 Cdk Inhibitor, p35 - CAS 471270-60-7 - Calbiochem The Cdk Inhibitor, p35, also referenced under CAS 471270-60-7, controls the biological activity of Cdk. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
219477 Cdk4 Inhibitor II, NSC 625987 - CAS 141992-47-4 - Calbiochem The Cdk4 Inhibitor II, NSC 625987, also referenced under CAS 141992-47-4, controls the biological activity of Cdk4. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
219478 Cdk4 Inhibitor III - CAS 265312-55-8 - Calbiochem The Cdk4 Inhibitor III, also referenced under CAS 265312-55-8, controls the biological activity of Cdk4. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
219491 Cdk/Crk Inhibitor - CAS 784211-09-2 - Calbiochem The Cdk/Crk Inhibitor, also referenced under CAS 784211-09-2, controls the biological activity of Cdk/Crk. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
219492 Cdk4/6 Inhibitor IV - CAS 359886-84-3 - Calbiochem The Cdk4/6 Inhibitor IV, also referenced under CAS 359886-84-3, controls the biological activity of Cdk4/6. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
219494 Cdk/CKI Inhibitor, (R)-DRF053 - CAS 1186647-87-9 - Calbiochem The Cdk/CKI Inhibitor, (R)-DRF053, also referenced under CAS 1186647-87-9, controls the biological activity of Cdk/CKI. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
219503 Cdk4 Inhibitor V - CAS 943746-57-4 - Calbiochem The Cdk4 Inhibitor V, also referenced under CAS 943746-57-4, controls the biological activity of Cdk4. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
219511 Cdc2-Like Kinase Inhibitor IV, KH-CB19 - Calbiochem The Cdc2-Like Kinase Inhibitor IV, KH-CB19 controls the biological activity of Cdc2-Like KInase. This small molecule/inhibitor is primarily used for Cell Structure applications.
238803 Cdk2 Inhibitor III - CAS 199986-75-9 - Calbiochem The Cdk2 Inhibitor III, also referenced under CAS 199986-75-9, controls the biological activity of Cdk2. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
238804 Cdk2 Inhibitor IV, NU6140 - CAS 444723-13-1 - Calbiochem The Cdk2 Inhibitor IV, NU6140, also referenced under CAS 444723-13-1, controls the biological activity of Cdk2. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
238806 Cdk2/9 Inhibitor - CAS 507487-89-0 - Calbiochem The Cdk2/9 Inhibitor, also referenced under CAS 507487-89-0, controls the biological activity of Cdk2/9. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
238811 Cdk9 Inhibitor II - CAS 140651-18-9 - Calbiochem The Cdk9 Inhibitor II, also referenced under CAS 140651-18-9, controls the biological activity of Cdk9. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
341251 Fascaplysin, Synthetic - CAS 114719-57-2 - Calbiochem A cell-permeable red pigment, originally isolated from marine sponge, that acts as a potent, ATP-competitive inhibitor of Cdk4/D1 (IC₅₀ = 0.35 µM).
361552 InSolution™ GSK-3 Inhibitor IX - CAS 667463-62-9 - Calbiochem The InSolution™ GSK-3 Inhibitor IX, also referenced under CAS 667463-62-9, controls the biological activity of GSK-3. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
402081 Indirubin Derivative E804 - CAS 854171-35-0 - Calbiochem A cell-permeable indirubin derivative (IDR) that blocks the Src-Stat3 signaling pathway and displays anti-tumor properties.
402085 Indirubin-3ʹ-monoxime - CAS 160807-49-8 - Calbiochem A potent, reversible, and ATP-compatible inhibitor of GSK-3β (glycogen synthase kinase 3β), Cdk1 (cyclin-dependent kinase1) and Cdk5 (IC₅₀ = 22 nM, 180 nM, and 100 nM, respectively).
402086 Indirubin-3ʹ-monoxime, 5-Iodo- - CAS 331467-03-9 - Calbiochem A highly potent cell-permeable and reversible inhibitor of glycogen synthase kinase-3β (GSK-3β; IC₅₀ = 9 nM).
402088 Indirubin-3ʹ-monoxime-5-sulphonic Acid - CAS 331467-05-1 - Calbiochem A potent, reversible, and selective inhibitor of Cdk1 (IC₅₀ = 5 nM) and Cdk5 (IC₅₀ = 7 nM) and glycogen synthase kinase-3β (GSK-3β; IC₅₀ = 80 nM).
445820 Meriolin 2 - Calbiochem Meriolin 2 primarily used in Inhibition.
445821 Meriolin 3 - CAS 954143-48-7 - Calbiochem A cell-permeable, ATP site-targeting azaindolopyrimidine compound that is reported to inhibit kinase activity.
495620 Olomoucine - CAS 101622-51-9 - Calbiochem A purine derivative that acts as a potent, reversible and selective inhibitor of p34cdk1/cyclin B and related kinases.
495621 Olomoucine II - CAS 500735-47-7 - Calbiochem A cell-permeable 2,6,9-trisubstituted purine analog that acts as a potent, reversible, and ATP-competitive inhibitor of Cdk1/B.
495624 InSolution™ Olomoucine - Calbiochem
539644 UCN-01 A cell-permeable Staurosporine derived anticancer agent that reversibly and ATP-competitively inhibits several protein kinases.
540500 Purvalanol A - CAS 212844-53-6 - Calbiochem A potent, cell-permeable, reversible, and selective inhibitor of cyclin-dependent kinases.
557360 Roscovitine - CAS 186692-46-6 - Calbiochem Roscovitine, CAS 186692-46-6, is a potent, reversible, and selective inhibitor of CDKs. Displays 10 to 20 fold greater potency for p34cdk1, p33cdk2, and p33cdk5 relative to Olomoucine., A potent, reversible, and selective inhibitor of Cdks that exhibits about 10-fold greater efficacy towards p34-cdk1 and p33-cdk2 and 20-fold greater efficacy towards p33-cdk5 relative to Olomoucine.
557362 Roscovitine, (S)-Isomer - CAS 186692-45-5 - Calbiochem The (S)-enantiomer of the potent cyclin-dependent kinase (Cdk) inhibitor Roscovitine.
557364 InSolution™ Roscovitine - Calbiochem
572650 SU9516 - CAS 666837-93-0 - Calbiochem A cell-permeable 3-substituted indolinone compound that displays anti-proliferative and proapoptotic properties in tumor cells.
681500 WHI-P180 A potent inhibitor of lgE-mediated mast cell responses to allergens in vitro and in vivo.
A4847 Alsterpaullone ≥98% (HPLC), powder
SML1855 AZD5438 ≥97% (HPLC) New
B0435 Bohemine ≥95% (HPLC), powder
C3242 CDKi hydrochloride ≥98% (HPLC), solid
SML1352 CINK4 ≥95% (HPLC)
C3249 CR8 ≥95% (HPLC)
F3055 Flavopiridol hydrochloride hydrate ≥98% (HPLC), powder
G7791 GW8510 solid
I0404 Indirubin-3′-oxime ≥98% (HPLC), solid
SML1225 Indisulam ≥98% (HPLC)
I0763 N9-Isopropylolomoucine ≥98% (HPLC)
K3888 Kenpaullone ≥98%
SML0559 LDN193189 hydrochloride ≥98% (HPLC)
SML1036 LDN-193594 ≥98% (HPLC)
SML0064 MBX-102 ≥98% (HPLC)
M5824 MBX-102 acid ≥98% (HPLC), powder
M5443 mC2p solid
M5318 mC2p-NLS solid
N0915 NSC43067 ≥98% (HPLC)
N7287 NU-1025 ≥97% (HPLC), solid
N4286 NU2058 >98% (HPLC)
N4411 NU6027 ≥98% (HPLC)
SML1323 NU6140 ≥98% (HPLC)
O0886 Olomoucine ≥98% (HPLC)
O3264 Olomoucine II ≥97% (HPLC), powder
PZ0199 PD 0332991 isethionate ≥98% (HPLC)
PZ0178 PHA 767491 hydrochloride ≥98% (HPLC)
SML0498 PNU112455A ≥98% (HPLC)
P5234 Purvalanol B ≥97% (HPLC), solid
P4484 Purvalanol A ≥98% (HPLC), powder
SML1254 R547 ≥98% (HPLC)
R7772 Roscovitine ≥98% (TLC)
S1693 SU 9516 ≥98% (HPLC), crystalline