Protein Kinase Inhibitors

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A4970 N-Acetyl-O-phosphono-Tyr-Glu Dipentylamide Potent dipeptide inhibitor of pp60c-src SH2 domain.
A6833 Arg-Lys-Arg-Ser-Arg-Ala-Glu lyophilized powder  
A4308 Autocamtide 2-related inhibitory peptide ≥97% (HPLC), lyophilized powder Potent inhibitor of calmodulin-depentent protein kinase II.
B3056 Bisindolylmaleimide II ≥97% (Mixture of 2 isomers) Inhibitor of protein kinase C.
B3306 Bisindolylmaleimide IV ≥98% (TLC), solid Inhibitor of protein kinase C.
B3681 Bisindolylmaleimide VII 96% (TLC), solid Selective inhibitor of protein kinase C.
B3931 Bisindolylmaleimide X hydrochloride ≥90%, solid Selective inhibitor of protein kinase C.
B4056 Bisindolylmaleimide XI hydrochloride ≥98% (TLC), solid Selective inhibitor of protein kinase C.
B6292 GF 109203X hydrochloride ≥95% Inhibitor of protein kinase C; potent inhibitor of GSK-3.
M7795 rac-2-Methoxy-3-hexadecanamido-1-propylphosphocholine ≥90% Protein kinase C inhibitor.
P6062 Protein Kinase A Inhibitor Fragment 6-22 amide ≥97% (HPLC) Potent inhibitor of cAMP-dependent protein kinase (PKA) (Ki = 2.5 nM); derived from the active portion of the heat-stable PKA inhibitor protein PKI.
P3115 Protein Kinase C Inhibitor, Myristoylated ≥7.5 mg/mL (peptide and counter ion), ≥95% (Minimum peptide content 70%, HPLC), aqueous solution (neutral pH) Protein Kinase C Inhibitor, Myristoylated is a cell permeable, specific inhibitor of calcium and phospholipid-dependent Protein Kinase C.
P1614 Protein kinase Cζ pseudosubstrate, myristoyl trifluoroacetate salt ≥90% (HPLC) Cell permeable protein kinase C (PKC) ζ inhibitor.
P0393 Protein Kinase Inhibitor from porcine heart 1-3 inhibitor U/μg protein, lyophilized powder These proteins bind to the catalytic subunit of cyclic-AMP dependent protein kinase, displacing the regulatory subunit and inhibiting phosphorylating activity. The cyclic-AMP binding capacity of the regulatory subunit is enhanced. Many other proteins exhibit this enhancement ability, too (Brostrom, C.O. and Kon, C., Anal. Biochem., 58, 459 [1974]).
P0300 Protein Kinase Inhibitor from rabbit ≥85% (HPLC) Inhibitor of c-AMP-dependent protein kinase
These proteins bind to the catalytic subunit of cyclic-AMP dependent protein kinase, displacing the regulatory subunit and inhibiting phosphorylating activity. The cyclic-AMP binding capacity of the regulatory subunit is enhanced.