Imidazoline Binding Site Ligands

Product #	Description	Biochem/physiol Actions	Image	Add to Cart
A7127	Agmatine sulfate salt ≥97%, powder	Putative endogenous neurotransmitter at imidazoline receptors; displaces clonidine at α₂-adrenergic and at imidazoline receptors; blocks NMDA-activated ion channels in hippocampal neurons.		pricing

A9899	Antazoline hydrochloride	Imidazoline agonist; more potent than efaroxan in inducing insulin release from β cells; H₁ histamine receptor antagonist.		pricing

B154	BU224 hydrochloride solid	I₂ Imidazoline receptor antagonist.		pricing

B8433	BU99006 >91% (HPLC)	Irreversible I₂ imidazoline binding site ligand.		pricing

B4555	Benazoline oxalate salt solid	I₂imidazoline receptor agonist; has high affinity and selectivity for I₂ imidazoline receptors over α-adrenoceptors.		pricing

C223	Cirazoline hydrochloride solid	Selective α₁-adrenoceptor agonist; non-selective imidazoline binding site ligand		pricing

C7897	Clonidine hydrochloride solid	α₂-adrenoceptor agonist; I₁ imidazoline binding site ligand.		pricing

E3263	Efaroxan hydrochloride ≥98% (HPLC)	(+)-Isomer is a selective α-adrenoceptor antagonist; (−)-isomer is an imidazoline ligand that induces insulin secretion, mediated by the blockade of ATP-sensitive potassium channels in pancreatic β cells; I₁ imidazoline binding site antagonist.		pricing

I6138	Idazoxan hydrochloride	α₂-adrenoceptor antagonist; I₂ imidazoline receptor agonist; I₁ imidazoline receptor antagonist		pricing

M5685	Metrazoline solid	Potent and selective imidazoline binding site ligand		pricing

R134	Rilmenidine hemifumarate salt solid	Selective I₁ imidazoline receptor agonist.		pricing

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