Acetylcholinesterase

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SML1569 Acotiamide dihydrochloride ≥98% (HPLC) Acotiamide is a potent, selective and reversible inhibitor of human and canine stomach-derived acetylcholinesterase (AChE). Acotiamide showed no affinity for dopamine D2 or serotonin 5-HT4 receptors but does have activity as a muscarinic antagonist. It acts as a prokinetic drug through acetylcholinesterase inhibition and muscarinic receptor antagonism, and has been used for the treatment of functional dyspepsia (FD) involving gastric motility dysfunction.
A3773 9-Amino-1,2,3,4-tetrahydroacridine hydrochloride hydrate ≥99%  
A9013 1,5-Bis(4-allyldimethylammoniumphenyl)pentan-3-one dibromide Selective acetylcholinesterase inhibitor.
W0641 W-84 dibromide ≥98% (HPLC), solid Potent allosteric modulator of M2 muscarinic acetylcholine receptors.
D0879 Diisopropylfluorophosphate Potent inhibitor of serine proteases such as trypsin and chymotrypsin, and of acetylcholinesterase; also inhibits cathepsin G, cholinesterase, coagulation factor Xa, leucocyte elastase, pancreatic elastase, tissue kallikrein, plasmin, subtilisin, and thrombin. Inhibition of acetylcholinesterase makes this compound especially toxic. Inhibits apoptosis induced by ricin and bacterial toxins.
E8375 Eserine Acetylcholinesterase inhibitor that crosses the blood-brain barrier and forms a carbamylated enzyme complex with acetyl cholinesterase that degrades slowly.
45710 Eserine ≥98.0% (N) Acetylcholinesterase inhibitor that crosses the blood-brain barrier and forms a carbamylated enzyme complex with acetyl cholinesterase that degrades slowly.
E8625 Eserine hemisulfate salt Acetylcholinesterase inhibitor that crosses the blood-brain barrier and forms a carbamylated enzyme complex with acetyl cholinesterase that degrades slowly.
G1660 Galanthamine hydrobromide from Lycoris sp. ≥94% (TLC) Cholinesterase inhibitor; reverses scopolamine-induced amnesia; antimyasthenic.
H5902 (−)-Huperzine A Acetylcholinesterase inhibitor; active enantiomer.
H5777 (±)-Huperzine A synthetic, ≥98% (TLC) Acetylcholinesterase inhibitor.
SML0033 Itopride hydrochloride ≥98% (HPLC) Itopride is an acetylcholinesterase (AChE) inhibitor and D2 dopamine receptor antagonist. Itopride is used as a gastroprokinetic agent.
N2001 Neostigmine bromide ≥98% (HPLC and titration), powder Reversible inhibitor of acetylcholinesterase that is similar to eserine, but does not cross the blood-brain barrier.
N2126 Neostigmine methyl sulfate Reversible inhibitor of acetylcholinesterase that is similar to eserine, but does not cross the blood-brain barrier.
P9797 Pyridostigmine bromide Acetylcholinesterase inhibitor.
SML0967 TAE-1 ≥98% (HPLC) TAE-1 is an inhibitor of amyloid-β fibril formation and aggregation. TAE-1 is a sym-triazine with dual activity against Alzheimer′s disease. TAE-1 inhibits cholinesterases AChE and BuChE with IC50 values of 0.3 and 3.9 μM. Studies using TAE-1 on differentiated human SH-SY5Y neuronal cells have suggested that it can stimulate synapse formation and promote the differentiation of human neurons, increasing neurite extension.