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Showing 1-14 of 14 results for "09658" within Papers
Development of Two Synthetic Approaches to an APJ Receptor Agonist Containing a Tetra-ortho-Substituted Biaryl Pyridone
Goldfogel, M. J., et al.
Organic Process Research & Development, 26, 3, 624-634 (2022)
Progress towards the synthesis of piperazimycin A: synthesis of the non-proteogenic amino acids and elaboration into dipeptides
Kennedy JP and Lindsley CW
Tetrahedron Letters, 51(18), 2493-2496 (2010)
Ayman El-Faham, et al
European Journal of Organic Chemistry, 19, 3641-3649 (2010)
Judit Tulla-Puche et al.
Bioconjugate chemistry, 19(10), 1968-1971 (2008-09-23)
Prodrugs are increasingly used as delivery vehicles for pharmaceutical agents that present solubility and/or pharmacokinetic/metabolic issues. In the course of the development of prodrugs for the antitumoral agent thiocoraline, standard coupling reagents and procedures failed to provide the desired target
J. Phillip Kennedy and Craig W. Lindsley
Tetrahedron Letters, 51, 2493-2496 (2010)
N, N, N′, N′-Tetramethylchloroformamidinium hexafluorophosphate (TCFH), a powerful coupling reagent for bioconjugation
Tulla-Puche J, et al.
Bioconjugate Chemistry, 19(10), 1968-1971 (2008)
Ayman El-Faham et al.
Chemistry (Weinheim an der Bergstrasse, Germany), 15(37), 9404-9416 (2009-07-22)
We describe a new family of uronium-type coupling reagents that differ in their iminium moieties and leaving groups. The presence of the morpholino group in conjunction with an oxime derivative--especially ethyl 2-cyano-2-(hydroxyimino)acetate (Oxyma)--had a marked influence on the solubilities, stabilities
J. Habermann et al.
J. Prakt. Chem./Chem.-Ztg., 340, 233-233 (1998)
COMU: a safer and more effective replacement for benzotriazole-based uronium coupling reagents
El-Faham A, et al.
Chemistry?A European Journal , 15(37), 9404-9416 (2009)
L.A. Carpino et al.
Journal of the American Chemical Society, 117, 5401-5401 (1995)
An Efficient Second-Generation Manufacturing Process for the pan-RAF Inhibitor Belvarafenib
Zell, D., et al.
Organic Process Research & Development, 25, 10, 2338-2350 (2021)
A novel family of onium salts based upon isonitroso meldrum's acid proves useful as peptide coupling reagents
El-Faham A, et al.
European Journal of Organic Chemistry, 2010(19), 3641-3649 (2010)
Anita K Kovács et al.
Frontiers in chemistry, 6, 120-120 (2018-05-05)
A general strategy for the synthesis of N-peptide-6-amino-D-luciferin conjugates has been developed. The applicability of the strategy was demonstrated with the preparation of a known substrate, N-Z-Asp-Glu-Val-Asp-6-amino-D-luciferin (N-Z-DEVD-aLuc). N-Z-DEVD-aLuc was obtained via a hybrid liquid/solid phase synthesis method, in which
Rapid Development of a Commercial Process for Linrodostat, an Indoleamine 2,3-Dioxygenase (IDO) Inhibitor
Fraunhoffer, K.J., et al.
Organic Process Research & Development, 23, 11, 2482-2498 (2019)
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