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Showing 1-23 of 23 results for "480959" within Papers
Balasubramanian Narasimhan et al.
Chemical & pharmaceutical bulletin, 54(8), 1067-1071 (2006-08-02)
A method consisting of quantitative structure-activity relationship (QSAR) (MLR) was developed to predict the hydrolytic rate constant of 37 benzoglycolamide ester prodrugs. The regression method was used as a calibration model for calculating the hydrolytic rate constant and investigating their
Fereidoon Daryaee et al.
European journal of medicinal chemistry, 44(1), 289-295 (2008-04-26)
On the basis of the structural similarity of N-substituted glycolamides with N-glycolyl muramic acid residues of the cell wall of Mycobacterium tuberculosis, a series of these compounds were designed and synthesized by the reaction of glycolic acid acetonide 1 (2,2-dimethyl-5-oxo-1,3-dioxolane)
Parmeshwari K Halen et al.
Mini reviews in medicinal chemistry, 9(1), 124-139 (2009-01-20)
Non-steroidal anti-inflammatory drugs (NSAIDs), commonly used for the treatment of chronic inflammatory diseases suffer from several undesired side effects, the most important being gastrointestinal (GI) irritation and ulceration. The prodrug designing is one of the several strategies used to overcome
Partial molal isothermal compressibility of glycine, DL-α-alanine, glycylglycine, glycolamide, and lactamide.
Yayanos AA.
The Journal of Physical Chemistry, 97(49), 13027-13028 (1993)
Sean D Reilly et al.
Chemical communications (Cambridge, England), 48(78), 9732-9734 (2012-08-24)
Complexation of Pu(IV) with TMDGA, TEDGA, and TODGA diglycolamide ligands was followed by vis-NIR spectroscopy. A crystal structure determination reveals that TMDGA forms a 1 : 3 homoleptic Pu(IV) complex with the nitrate anions forced into the outer coordination sphere.
P R Brown et al.
Journal of general microbiology, 133(6), 1527-1533 (1987-06-01)
A positive selection is described for isolating amidase-negative mutants from Pseudomonas aeruginosa strains. The method is based on the conversion, via amidase activity, of glycollamide to glycollate which is growth inhibitory. Three types of mutant were isolated on lactate medium
A K Bansal et al.
Drug development and industrial pharmacy, 27(1), 63-70 (2001-03-15)
Glycolamide esters of ibuprofen (I), namely, unsubstituted (II), N,N dimethyl (III), and N,N diethyl (IV), were synthesized and studied for different physicochemical, pharmacological, and toxicological properties. They were comparable with I in respect of anti-inflammatory and analgesic activity but did
Maneesh Kumar et al.
Journal of cellular biochemistry, 120(10), 18298-18308 (2019-07-17)
The arthropod-transmitted chikungunya virus has emerged as an epidemic menace that causes debilitating polyarthritis. With this life-threatening impact on humans, the possible treatment requires to cure the viral infectivity. But, devoid of any vaccine against the chikungunya virus (CHIKV), there
Yu-Cai He et al.
Applied biochemistry and biotechnology, 160(5), 1428-1440 (2009-04-01)
Alcaligenes sp. ECU0401 has been isolated from soil samples with high nitrilase activity against glycolonitrile using the enrichment culture technique. The preferred carbon/nitrogen sources and metal ions were sodium acetate, a composite of peptone and yeast extract, and Cu(2+), respectively.
H Ogata et al.
Biochimica et biophysica acta, 1119(2), 123-126 (1992-02-26)
Alkyl glycolamido phosphoric esters (P-O-CH2-CO-NH-(CH2)n-CH3) and alkyl monoglycolate phosphoric esters (P-O-CH2-CO-O-(CH2)n-CH3), which are analogs of the aldolase substrate fructose-1-phosphate, were synthesized and use for probing the active site of rabbit muscle aldolase. The inhibition constants (Ki) were affected by the
Samuel Bernardo-Bermejo et al.
Journal of chromatography. A, 1596, 124-133 (2019-03-18)
Diabetes mellitus is a major health concern nowadays. It is estimated that 40% of diabetics are affected by diabetic nephropathy, one of the complications derived from high glucose blood levels which can lead to chronic loss of kidney function. It
A Study of the Diffusion of Glycolamide in Water at 25? with the Gouy Interference Method.
Dunlop PJ and Gosting LJ.
Journal of the American Chemical Society, 75(20), 5073-5075 (1953)
R Ruhela et al.
Talanta, 85(2), 1217-1220 (2011-07-06)
A precise, sensitive and selective method for the spectrophotometric determination of palladium (II) using N,N,N',N'-tetra(2-ethylhexyl) thiodiglycolamide T(2EH)TDGA as an extractant is described. Palladium (II) forms yellow colored complex with T(2EH)TDGA which exhibits an absorption maximum at ∼ 300 nm. The
Prasanta K Mohapatra et al.
Inorganic chemistry, 52(5), 2533-2541 (2013-02-12)
Diglycolamide-functionalized calix[4]arenes (C4DGAs) with varying structural modifications were evaluated for actinide complexation from their extraction behavior toward actinide ions such as UO2(2+), Pu(4+), PuO2(2+), and Am(3+) in the room temperature ionic liquid (RTIL) 1-n-octyl-3-methylimidazolium bis(trifluoromethane)sulfonamide (C8mimNTf2). The formation constants were
Peter C Burgers et al.
European journal of mass spectrometry (Chichester, England), 18(2), 149-159 (2012-05-30)
Early combined computational and experimental studies by J.K. Terlouw c.s. in Refs. 1-3 propose that low-energy methyl carbamate ions, NH(2)COOCH(3)(•+) (MC-1), rearrange into distonic ions NH(2)C(OH)OCH(2)(•+) and hydrogen-bridged radical cations [NH(2)C=O--H--OCH(2)](•+) (MC-5) en route to the observed losses of HCO(•)
Jeffrey C Pelletier et al.
Bioorganic & medicinal chemistry, 16(13), 6617-6640 (2008-05-31)
Antagonism of the gonadotropin releasing hormone (GnRH) receptor has shown positive clinical results in numerous reproductive tissue disorders such as endometriosis, prostate cancer and others. Traditional therapy has been limited to peptide agonists and antagonists. Recently, small molecule GnRH antagonists
New facile synthesis of phosphoglycolohydroxamic acid and other phosphoglycolic acid derivatives.
Weber P, et al.
Tetrahedron Letters, 44(50), 9047-9049 (2003)
Yuji Sasaki et al.
Analytical sciences : the international journal of the Japan Society for Analytical Chemistry, 21(10), 1171-1175 (2005-11-08)
In order to evaluate the extraction property of new extractants, diglycolamide (DGA) compounds, we investigated the maximum extraction of di-, tri-, and tetravalent metal ions using nitric acid and n-dodecane. The limits of metal concentration (LOC) for Ca(II), Nd(III) and
J F Gilmer et al.
Chemico-biological interactions, 157-158, 317-319 (2005-11-04)
Butyrylcholinesterase [EC 3.1.1.8] present widely in mammalian tissue does not have a precisely defined biological function or known endogenous substrate. However, it plays an important role in the detoxification of certain xenobiotics and is an established vector for the systemic
The Heats of Dilution of Aqueous Solutions of Glycine and Glycolamide, and Other Thermodynamic Properties of Glycine at 25?1,2.
Gucker Jr FT, et al.
Journal of the American Chemical Society, 62(10), 2698-2704 (1940)
Activity data for aqueous glycolamide solutions at 25?.
Stokes RH.
Transactions of the Faraday Society, 50, 565-567 (1954)
On the conformational equilibrium of glycolamide: A free jet millimetre-wave spectroscopy and computational study.
Maris A.
Physical Chemistry Chemical Physics, 6(10), 2611-2616 (2004)
Alan C Cheng et al.
Scientific reports, 8(1), 7570-7570 (2018-05-17)
Small molecules and antibodies each have advantages and limitations as therapeutics. Here, we present for the first time to our knowledge, the structure-guided design of "chemibodies" as small molecule-antibody hybrids that offer dual recognition of a single target by both
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