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370654 Millipore

PKG Inhibitor - Calbiochem

The PKG Inhibitor controls the biological activity of PKG. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

Synonym: Protein Kinase G Inhibitor, RKRARKE

  • Empirical Formula (Hill Notation) C38H74N18O10

  • Molecular Weight 943.11

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Properties

Related Categories Biochemicals and Reagents, Enzyme Inhibitors, Enzyme Inhibitors by Enzyme, Enzymes, Inhibitors, and Substrates, P to Q,
packaging   1 mg in Plastic ampoule (370654-1MG)
feature productdata solubility   H₂O (1 mg/ml)
brand family   Calbiochem
form   Lyophilized
primary target Ki   86 µM against protein kinase G
purity   ≥95% by HPLC
storage conditions   Hygroscopic
  Ok to freeze
shipped in   ambient
storage conditions   -20C

Description

Biochem/physiol Actions

Cell permeable: no

Product does not compete with ATP.

Reversible: yes

General description

A more specific, reversible, and substrate competitive inhibitor of protein kinase G (Ki = 86 µM) relative to protein kinase A (Ki = 550 µM). Sequence corresponds to a non-phosphorylatable analog (Ser32 to Ala32) of histone H2B (amino acids 29-35).

A specific, reversible, and substrate competitive inhibitor of PKG (Ki = 86 µM) relative to PKA (Ki = 550 µM). Sequence corresponds to a non-phosphorylatable analog (Ser32 to Ala32) of histone H2B (amino acids 29-35).

Other Notes

Glass, D.B., et al. 1983. Biochem. J.213, 159.

Packaging

Yes

Warning

Standard Handling (A)

Sequence

H-Arg-Lys-Arg-Ala-Arg-Lys-Glu-OH

Safety & Documentation

Safety Information

Safety Information for this product is unavailable at this time.

Documents

Certificate of Analysis

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Protocols & Articles
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