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S5317 Sigma-Aldrich

SKF-95282 dimaleate salt

solid, >98% (HPLC)

Synonym: N-[3-[3-(1-Piperidinylmethyl)phenoxy]propyl]-2-benzothiazolamine, Zolantidine

  • CAS Number 104076-39-3

  • Empirical Formula (Hill Notation) C22H27N3OS · 2C4H4O4

  • Molecular Weight 613.68

  •  MDL number MFCD01862676

  •  PubChem Substance ID 24278066

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Description

Application

SKF 95282 dimaleate salt was one of the compounds tested for ability to cross gastrointestinal tract and blood-brain barrier by permeability assays.2

Biochem/physiol Actions

SKF 95282 is a benzthiazole derivative that potently inhibits histamine H2 receptor. It crosses the blood-brain barrier and inhibits the histamine-stimulated activity of adenylate cyclase in guinea pig brain.1

H2 Histamine receptor antagonist.

Features and Benefits

This compound is also offered as part of Sigma′s Library of Pharmacologically Active Compounds (LOPAC®1280), a biologically annotated collection of high-quality, ready-to-screen compounds. Click here to learn more.

This compound was developed by GlaxoSmithKline. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

Legal Information

Sold for research purposes under agreement from Glaxo­Smith­Kline

LOPAC is a registered trademark of Sigma-Aldrich Co. LLC

Safety & Documentation

Safety Information

RIDADR 
NONH for all modes of transport
WGK Germany 
3

Documents

Certificate of Analysis

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Milli-Q® Water Purification Solutions
Protocols & Articles
Peer-Reviewed Papers
15

References

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