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SML0342 Sigma

TFM-4AS-1

≥98% (HPLC)

Synonym: (4aR,6aS,7S,11aR)-1,4a,6a-Trimethyl-2-oxo-N-[2-(trifluoromethyl)phenyl]-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11atetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxamide

  • CAS Number 188589-61-9

  • Empirical Formula (Hill Notation) C27H33F3N2O2

  • Molecular Weight 474.56

  •  PubChem Substance ID 329825347

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Properties

Related Categories Androgen, Bioactive Small Molecule Alphabetical Index, Bioactive Small Molecules, Cell Biology, Cell Signaling and Neuroscience,
InChI Key   YFBLEKKYWFJKBP-HNXMFXTHSA-N
assay   ≥98% (HPLC)
form   powder
color   white to beige
solubility   DMSO: >5 mg/mL
storage temp.   2-8°C

Description

Packaging

5, 25 mg in glass bottle

Biochem/physiol Actions

TFM-4AS-1 is a potent SARM (Selective Androgen Receptor Modulator). TFM-4AS-1 is a partial agonist of AR. The compound promotes the buildup of bone and muscle mass while having reduced effects on reproductive organs and sebaceous glands. The compound also is an inhibitor of rat 5 α-reductase enzymes type I (2 nM) and type 2 (3 nM).

Safety & Documentation

Safety Information

RIDADR 
NONH for all modes of transport
WGK Germany 
3

Documents

Certificate of Analysis


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Protocols & Articles

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