Heteroaryl Boronic Acids

Select, Compare, and Buy Heteroaryl Boronic Acids for Suzuki Coupling

Heteroaryl boronic acids are one type of synthetic intermediate commonly used in the Suzuki-Miyaura palladium catalyzed cross-coupling reaction, among others. These building blocks are heterocyclic and aromatic. They are also used in Chan-Lam coupling, homologations, conjugate additions, electrophilic allyl shifts, Lieberskind-Strogl coupling, Sonogashira coupling, and Stille coupling.

See other types of boronic acids. Our boronic acids and derivatives page has additional information on MIDA boronates and links to related technical spotlights and relevant articles from the Aldrichimica Acta and ChemFiles.

Use the table below to browse heteroaryl boronic acids by name, structure, product number, molecular formula, and price. Many of our heteroaryl boronic acids are also available (as indicated) through the AldrichCPR platform in custom amounts from 1 mg to several grams.

Product detail pages also include the empirical formula, synonyms, molecular weight, MDL number, and PubChem substance ID.

Request a bulk order for heteroaryl boronic acids or other discovery chemistry reagents from any product page. Our team will review your request for bulk materials along with any unique or large package size requirements to ensure you a smooth single order or a customized regular supply to suit your needs.

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CDS007044 isoxazole-4-boronic acid AldrichCPR C3H4BNO3
720429 1H-Pyrazol-3-ylboronic acid hydrate C3H5BN2O2 · xH2O
706256 1H-Pyrazole-4-boronic acid ≥95.0% C3H5BN2O2
CDS014043 1H-Pyrazole-5-boronic acid AldrichCPR C3H5BN2O2
CDS015511 Imidazole-2-boronic acid AldrichCPR C3H5BN2O2
557684 5-Bromo-2-thienylboronic acid ≥95% C4H4BBrO2S
CDS004266 3-chlorothiophene-2-boronic acid AldrichCPR C4H4BClO2S
499935 5-Chloro-2-thienylboronic acid C4H4BClO2S
CDS013999 pyrimidine-5-boronic acid AldrichCPR C4H5BN2O2
CDS001345 Uracil-5-boronic acid AldrichCPR C4H5BN2O4
436836 2-Thienylboronic acid ≥95.0% C4H5BO2S
436844 3-Thienylboronic acid ≥95.0% C4H5BO2S
464910 2-Furanylboronic acid ≥95.0% C4H5BO3
512168 3-Furanylboronic acid ≥95.0% C4H5BO3
706221 2-Aminopyrimidine-5-boronic acid ≥95.0% C4H6BN3O2
470317 2,5-Thiophenediylbisboronic acid ≥95.0% C4H6B2O4S
CDS006785 2,3-dichloropyridine-4-boronic acid AldrichCPR C5H4BCl2NO2
CDS007852 2,6-dichloropyridine-3-boronic acid AldrichCPR C5H4BCl2NO2
CDS010298 2,6-difluoropyridine-4-boronic acid AldrichCPR C5H4BF2NO2
686816 5-Bromopyridine-3-boronic acid ≥95% C5H5BBrNO2
666556 6-Bromo-3-pyridinylboronic acid ≥95% C5H5BBrNO2
666513 2-Chloro-4-pyridinylboronic acid ≥95.0% C5H5BClNO2
697095 2-Chloropyridine-3-boronic acid C5H5BClNO2
721034 5-Chloro-3-pyridineboronic acid ≥95% C5H5BClNO2
CDS002921 5-Chloropyridine-2-boronic acid AldrichCPR C5H5BClNO2
637386 6-Chloro-3-pyridinylboronic acid ≥95.0% C5H5BClNO2
696579 2-Fluoro-3-pyridineboronic acid ≥95% C5H5BFNO2
CDS003936 2-fluoropyridine-4-boronic acid AldrichCPR C5H5BFNO2
CDS007991 3-fluoropyridine-4-boronic acid AldrichCPR C5H5BFNO2
639184 6-Fluoro-3-pyridinylboronic acid C5H5BFNO2
499900 2-Formyl-3-thiopheneboronic acid ≥95% C5H5BO3S
499919 3-Formyl-2-thienylboronic acid ≥95% C5H5BO3S
514055 5-Formyl-2-thienylboronic acid ≥95.0% C5H5BO3S
CDS004568 5-formylthiophene-3-boronic acid AldrichCPR C5H5BO3S
512346 5-Formyl-2-furanylboronic acid ≥95% C5H5BO4
CDS005028 3-borono-2-thiophenecarboxylic acid AldrichCPR C5H5BO4S
CDS004504 5-(Dihydroxyboryl)-2-thiophenecarboxylic acid AldrichCPR C5H5BO4S
CDS020044 2,6-Difluoropyridine-3-boronic acid hydrate AldrichCPR C5H6BF2NO3
731730 1-Methyl-3-trifluoromethyl-1H-pyrazole-5-boronic acid ≥95% C5H6BF3N2O2
CDS009263 2-Pyridineboronic acid AldrichCPR C5H6BNO2
512125 3-Pyridinylboronic acid ≥95.0% C5H6BNO2
634492 4-Pyridinylboronic acid 90% C5H6BNO2
CDS006321 pyridine-4-boronic acid hydrochloride AldrichCPR C5H7BClNO2
CDS003645 4-methylthiophene-2-boronic acid AldrichCPR C5H7BO2S
CDS019945 5-Methyl-2-furanboronic acid AldrichCPR C5H7BO3
720410 3,5-Dimethylisoxazol-4-yl-4-boronic acid ≥95% C5H8BNO3
CDS007058 1,3-dimethylpyrazole-5-boronic acid AldrichCPR C5H9BN2O2
CDS007030 1-ethylpyrazole-4-boronic acid AldrichCPR C5H9BN2O2
CDS010102 2-(trifluoromethyl)pyridine-4-boronic acid AldrichCPR C6H5BF3NO2
CDS009086 5-cyano-3-pyridinyl boronic acid AldrichCPR C6H5BN2O2
CDS009971 3-chloro-2-methoxypyridine-4-boronic acid AldrichCPR C6H7BClNO3
CDS015768 4-(trifluoromethyl)pyridine-3-boronic acid hydrate AldrichCPR C6H7BF3NO3
701939 2-Acetyl-3-thiopheneboronic acid C6H7BO3S
499927 5-Acetyl-2-thienylboronic acid C6H7BO3S
CDS019614 2-Methylpyridine-3-boronic acid AldrichCPR C6H8BNO2
CDS003860 4-methylpyridine-3-boronic acid AldrichCPR C6H8BNO2
CDS020146 5-Methylpyridine-3-boronic acid AldrichCPR C6H8BNO2
CDS020001 6-Methylpyridine-3-boronic acid AldrichCPR C6H8BNO2
SYX00028 2-Methylthiopyridine-5-boronic acid AldrichCPR C6H8BNO2S
684589 2-Methoxy-3-pyridinylboronic acid ≥95.0% C6H8BNO3
CDS007799 2-methoxypyridine-4-boronic acid AldrichCPR C6H8BNO3
CDS004292 5-methoxypyridine-3-boronic acid AldrichCPR C6H8BNO3
CDS010165 6-(hydroxymethyl)pyridine-3-boronic acid AldrichCPR C6H8BNO3
637610 6-Methoxy-3-pyridinylboronic acid ≥95.0% C6H8BNO3
CDS005381 2-ethoxypyrimidine-5-boronic acid AldrichCPR C6H9BN2O3
666491 2,4-Dimethoxy-5-pyrimidinylboronic acid 90% C6H9BN2O4
CDS005265 2-dimethylaminopyrimidinyl-5-boronic acid AldrichCPR C6H10BN3O2
CDS008131 1,3,5-Trimethyl-1H-pyrazol-4-ylboronic acid AldrichCPR C6H11BN2O2
CDS019261 1,3-Benzothiazol-6-ylboronic acid AldrichCPR C7H6BNO2S
724017 1H-Indazole-5-boronic acid ≥95% C7H7BN2O2
CDS009958 Imidazo[1,2-a]pyridine-6-boronic acid AldrichCPR C7H7BN2O2
720828 Indazole-6-boronic acid C7H7BN2O2
715409 1H-Indazole-5-boronic acid hydrochloride C7H8BClN2O2
709379 Indazole-4-boronic acid hydrochloride C7H8BClN2O2
CDS005468 2-(methylcarboxy)pyridine-5-boronic acid AldrichCPR C7H8BNO4
CDS006725 5-bromo-2-ethoxy-4-pyridineboronic acid AldrichCPR C7H9BBrNO3
CDS020467 5-Chloro-6-ethoxypyridine-3-boronic acid AldrichCPR C7H9BClNO3
CDS010143 2,5-dimethylpyridine-3-boronic acid AldrichCPR C7H10BNO2
718815 6-Ethoxy-3-pyridinylboronic acid C7H10BNO3
CDS019714 6-Methoxy-5-methylpyridine-3-boronic acid AldrichCPR C7H10BNO3
706086 2,6-Dimethoxy-3-pyridineboronic acid ≥95% C7H10BNO4
CDS006698 5-bromobenzo[b]thiophene-2-boronic acid AldrichCPR C8H6BBrO2S
499978 Benzo[b]thien-2-ylboronic acid ≥95% C8H7BO2S
512117 Benzo[b]thien-3-ylboronic acid ≥95.0% C8H7BO2S
499943 2-Benzofuranylboronic acid ≥95% C8H7BO3
CDS013896 Benzopyrazine-6-boronic acid hydrochloride AldrichCPR C8H8BClN2O2
666467 5-Indolylboronic acid ≥95% C8H8BNO2
666459 6-Indolylboronic acid ≥95% C8H8BNO2
CDS013942 indole-4-boronic acid AldrichCPR C8H8BNO2
CDS020541 2-Methylbenzothiazole-5-boronic acid AldrichCPR C8H8BNO2S
CDS019574 (1-Methyl-1H-benzimidazol-5-yl)boronic acid AldrichCPR C8H9BN2O2
CDS010063 1-Methyl-1H-benzoimidazole-6-boronic acid AldrichCPR C8H9BN2O2
720798 1-Methyl-1H-indazole-6-boronic acid ≥95% C8H9BN2O2
720836 2-Methyl-2H-indazole-6-boronic acid C8H9BN2O2
635995 1,4-Benzodioxane-6-boronic acid ≥95% C8H9BO4
723606 1-Methyl-1H-indazole-4-boronic acid hydrochloride C8H10BClN2O2
CDS020489 5-Chloro-6-isopropoxypyridine-3-boronic acid AldrichCPR C8H11BClNO3
CDS005072 2-isoproxypyridine-5-boronic acid AldrichCPR C8H12BNO3
CDS020475 2-Morpholinopyrimidin-5-ylboronic acid AldrichCPR C8H12BN3O3
CDS010360 1-(Tetrahydro-2H-pyran-2-yl)-1H-pyrazol-5-ylboronic acid AldrichCPR C8H13BN2O3
CDS009357 1-(3-Methylbutyl)-1H-pyrazole-4-boronic acid AldrichCPR C8H15BN2O2
696684 2-Chloro-3-quinolineboronic acid ≥95% C9H7BClNO2
709522 3-Quinolineboronic acid C9H8BNO2
691909 3-Quinolineboronic acid technical grade C9H8BNO2
686867 5-Isoquinolineboronic acid ≥95.0% C9H8BNO2
542865 8-Quinolinylboronic acid technical grade C9H8BNO2
CDS010117 isoquinoline-6-boronic acid AldrichCPR C9H8BNO2
CDS009275 isoquinoline-7-boronic acid AldrichCPR C9H8BNO2
CDS007971 3-pyrazol-1-yl-phenylboronic acid AldrichCPR C9H9BN2O2
CDS009959 4-pyrazol-1-yl-phenylboronic acid AldrichCPR C9H9BN2O2
716480 1H-Inden-3-ylboronic acid 95% C9H9BO2
CDS005944 N-Methylindole-5-boronic acid AldrichCPR C9H10BNO2
CDS018401 4-(5-oxopyrazolidin-3-yl)phenylboronic acid AldrichCPR C9H11BN2O3
704768 2-(Pyrrolidin-1-yl)pyridine-3-boronic acid C9H13BN2O2
CDS020160 6-(Pyrrolidin-1-yl)pyridine-3-boronic acid AldrichCPR C9H13BN2O2
705039 2-Morpholinopyridine-3-boronic acid C9H13BN2O3
15047 N-Boc-2-pyrroleboronic acid ≥98.0% (T) C9H14BNO4
CDS020479 (2-Piperidin-1-ylpyrimidin-5-yl)boronic acid AldrichCPR C9H14BN3O2
CDS020497 2-(4-Methylpiperazin-1-yl)pyrimidin-5-ylboronic acid AldrichCPR C9H15BN4O2
797049 (6-Methyl-5-quinolinyl)boronic acid 95% C10H10BNO2
720445 1-Benzyl-1H-pyrazole-4-boronic acid ≥95% C10H11BN2O2
715441 3-(Trifluoromethyl)-1H-pyrazole-4-boronic acid pinacol ester 97% C10H14BF3N2O2
CDS018247 2-(morpholino)phenylboronic acid AldrichCPR C10H14BNO3
CDS005076 4-morpholinophenylboronic acid AldrichCPR C10H14BNO3
CDS005103 3-(pyrrolidin-1-ylsulfonyl)phenylboronic acid AldrichCPR C10H14BNO4S
CDS007679 4-(4-morpholinylsulfonyl)phenylboronic acid AldrichCPR C10H14BNO5S
CDS020471 6-(Piperidin-1-yl)pyridin-3-ylboronic acid AldrichCPR C10H15BN2O2
CBR01468 {6-[(2,2-Dimethylpropanoyl)amino]-3-pyridinyl}boronic acid AldrichCPR C10H15BN2O3
CDS007390 4-(2-(1H-Pyrazol-1-yl)ethoxy)phenylboronic acid AldrichCPR C11H13BN2O3
CDS004397 3-(pyrrolidine-1-carbonyl)phenylboronic acid AldrichCPR C11H14BNO3
CDS003611 4-(pyrrolidine-1-carbonyl)phenylboronic acid AldrichCPR C11H14BNO3
CDS005937 4-(morpholine-4-carbonyl)phenylboronic acid AldrichCPR C11H14BNO4
CDS011838 3-(1-pyrrolidinylmethyl)phenylboronic acid AldrichCPR C11H16BNO2
CDS014065 2-(4-morpholinylmethyl)phenylboronic acid AldrichCPR C11H16BNO3
CDS012386 [4-(morpholinomethyl)phenyl]boronic acid AldrichCPR C11H16BNO3
CDS010139 3-(piperidin-1-ylsulfonyl)phenylboronic acid AldrichCPR C11H16BNO4S
CBR00606 (8-Methoxy-2-methylquinolin-5-yl)boronic acid trihydrate AldrichCPR C11H18BNO6
499986 4-Dibenzothienylboronic acid ≥95.0% C12H9BO2S
CBR01389 Dibenzo[b,d]thien-2-ylboronic acid AldrichCPR C12H9BO2S
512214 1-Thianthrenylboronic acid ≥95% C12H9BO2S2
499951 4-(Dibenzofuranyl)boronic acid ≥95.0% C12H9BO3
ADE001429 (1-(tert-Butoxycarbonyl)-5-chloro-1H-pyrrolo[3,2-b]pyridin-3-yl)boronic acid AldrichCPR C12H14BClN2O4
CDS004586 3-(piperidine-1-carbonyl)phenylboronic acid AldrichCPR C12H16BNO3
CDS005409 4-(4-Methylpiperazine-1-carbonyl)phenylboronic acid hydrochloride AldrichCPR C12H18BClN2O3
CDS005378 3-(piperidin-1-ylmethyl)phenylboronic acid AldrichCPR C12H18BNO2
637394 (N-Boc-5-bromo-2-indolyl)boronic acid C13H15BBrNO4
741795 (N-Boc-5-chloro-2-indolyl)boronic acid 95% C13H15BClNO4
CDS005070 1-(tert-Butoxycarbonyl)-6-chloro-1H-indol-2-ylboronic acid AldrichCPR C13H15BClNO4
675911 N-Boc-indole-2-boronic acid ≥95% C13H16BNO4
CDS015480 4-(2-morpholinoethylcarbamoyl)phenylboronic acid AldrichCPR C13H19BN2O4
CDS003849 1-(triisopropylsilyl)pyrrole-3-boronic acid AldrichCPR C13H26BNO2Si
563870 1-(Phenylsulfonyl)-3-indolylboronic acid 97% C14H12BNO4S
CDS005099 1-Boc-6-methylindole-2-boronic acid AldrichCPR C14H18BNO4
680516 N-Boc-5-methoxy-2-indolylboronic acid ≥95% C14H18BNO5
CDS005504 1-(tert-Butyldimethylsilyl)-1H-indol-6-ylboronic acid AldrichCPR C14H22BNO2Si
CDS006675 1-(t-Butoxycarbonyl)-6-(methoxycarbonyl)-1H-indol-2-ylboronic acid AldrichCPR C15H18BNO6
CDS005906 2,4-bis(benzyloxy)pyrimidine-5-boronic acid AldrichCPR C18H17BN2O4
CDS007945 4-Benzyloxy-1-tert-butoxycarbonylindole-2-boronic acid AldrichCPR C20H22BNO5
CDS005096 5-benzyloxy-1-Boc-indole-2-boronic acid AldrichCPR C20H22BNO5