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A0487   Argatroban monohydrate ≥98% (HPLC) Argatroban has a high affinity and binds to arginine in thrombin active site resulting in steric hindrance for substrate binding. Argatroban is effective in preventing thrombus formation and favors thrombolysis than unfractionated heparin. It is recommended for acute ischemic stroke treatment.
Argatroban is a potent, seletive, univalent direct inhibitor of thrombin. It directly inhibits thrombin by binding only to its active site (thus univalent) as compared to Bivalent DTIs (hirudin and analogs) which bind both to the active site and exosite 1.
E8031 Esmolol hydrochloride ≥98% (HPLC), solid Esmolol hydrochloride is a ultrashort-acting β1 adrenoceptor antagonist (β1 receptor occupancy = 84.7%).
human ... ADRB1(153), ADRB2(154)
L1764 (±)-Lorazepam Anxiolytic; ligand for the GABAA receptor benzodiazepine modulatory site.
human ... GABRA1(2554), GABRA2(2555), GABRA3(2556), GABRA4(2557), GABRA5(2558), GABRA6(2559), GABRB1(2560), GABRB2(2561), GABRB3(2562), GABRD(2563), GABRE(2564), GABRG1(2565), GABRG2(2566), GABRG3(2567), GABRP(2568), GABRQ(55879)
M0763 Metoclopramide hydrochloride solid D2 antagonist; 5-HT3 antagonist; antipsychotic; anti-emetic.
human ... DRD2(1813), HTR3A(3359), HTR3B(9177), HTR3C(170572), HTR3D(200909), HTR3E(285242), HTR4(3360)
M8777 Morphine sulfate salt pentahydrate Narcotic analgesic; prototypic μ opioid receptor agonist; also agonist at κ opioid receptors.
human ... OPRM1(4988)
P6656 Promazine hydrochloride D2 dopamine receptor antagonist; phenothiazine antipsychotic.
human ... DRD2(1813), DRD3(1814), DRD4(1815), HTR2A(3356)