C102

8-Cyclopentyl-1,3-dimethylxanthine

Name: 8-Cyclopentyl-1,3-dimethylxanthine
Brand: SIGMA
Price: 263 CHF

≥98% (HPLC), powder

Synonym(e):

8-Cyclopentyltheophylline, CPT

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100 MG

CHF 263.00

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Über diesen Artikel

Empirische Formel (Hill-System):

C₁₂H₁₆N₄O₂

CAS-Nummer:

35873-49-5

Molekulargewicht:

248.28

NACRES:

NA.77

PubChem Substance ID:

24277730

UNSPSC Code:

12352200

MDL number:

MFCD00055116

Assay:

≥98% (HPLC)

Form:

powder

Quality level:

100

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InChI

1S/C12H16N4O2/c1-15-10-8(11(17)16(2)12(15)18)13-9(14-10)7-5-3-4-6-7/h7H,3-6H2,1-2H3,(H,13,14)

SMILES string

CN1C(=O)N(C)c2nc([nH]c2C1=O)C3CCCC3

InChI key

SCVHFRLUNIOSGI-UHFFFAOYSA-N

assay

≥98% (HPLC)

form

powder

color

white to off-white

solubility

H₂O: slightly soluble <0.28 mg/mL, 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 0.77 mg/mL, DMSO: ~16 mg/mL at 60 °C, 0.1 M NaOH: soluble

Quality Level

100

Gene Information

human ... ADORA1(134)

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Dieser Artikel	H127	A9657	H1512
Sigma-Aldrich C102 8-Cyclopentyl-1,3-dimethylxanthine	Sigma-Aldrich H127 p-Fluorohexahydro-sila-difenidol hydrochloride	Sigma-Aldrich A9657 DL-Aminoglutethimide	Sigma-Aldrich H1512 Haloperidol
form powder	form powder	form powder or crystals	form powder
assay ≥98% (HPLC)	assay ≥98% (HPLC)	assay ≥98% (TLC)	assay -
Quality Level 100	Quality Level 100	Quality Level 200	Quality Level 200
solubility H₂O: slightly soluble <0.28 mg/mL, DMSO: ~16 mg/mL at 60 °C, 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 0.77 mg/mL, 0.1 M NaOH: soluble	solubility H₂O: slightly soluble 1.5 mg/mL, 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: >14 mg/mL, ethanol: soluble	solubility H₂O: slightly soluble 0.2 mg/mL, 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 1.2 mg/mL, 0.1 M HCl: soluble, acetonitrile: soluble, methanol: soluble	solubility 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 0.39 mg/mL, 0.1 M HCl: 3 mg/mL, DMSO: soluble, H₂O: insoluble, ethanol: soluble
color white to off-white	color white to beige	color white	color white
Gene Information human ... ADORA1(134)	Gene Information human ... CHRM3(1131)	Gene Information human ... CYP11A1(1583), CYP17A1(1586), CYP19A1(1588) rat ... Cyp19a1(25147)	Gene Information human ... ABCB1(5243), ADRA1A(148), ADRA2A(150), ADRA2C(152), CHRM1(1128), DRD2(1813), DRD3(1814), DRD4(1815), EBP(10682), HRH1(3269), HTR2A(3356), HTR2C(3358), HTR7(3363), KCNH1(3756), KCNH2(3757), PRNP(5621) rat ... Adra1a(29412), Adra2a(25083), Chrm1(25229), Chrm2(81645), Drd1a(24316), Drd2(24318), Drd3(29238), Drd4(25432), Hrh1(24448), Htr1a(24473), Htr1b(25075), Htr2a(29595), Htr2c(25187), Oprs1(29336), Slc6a3(24898), Slc6a4(25553)

Biochem/physiol Actions

Selective A₁ adenosine receptor antagonist.

Features and Benefits

This compound is featured on the Adenosine Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Lagerklasse

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

ppe

Eyeshields, Gloves, type N95 (US)

Hier finden Sie alle aktuellen Versionen:

Analysenzertifikate (COA)

Lot/Batch Number

0000526424

0000474799

0000469282

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8-Cyclopentyl-1,3-dimethylxanthine