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| Size/SKU | Availability | Price |
|---|---|---|
10 mg | Please contact Customer Service for Availability | $142.00 |
50 mg | Please contact Customer Service for Availability | $458.00 |
About This Item
Empirical Formula (Hill Notation):
C23H15N3O
CAS Number:
Molecular Weight:
349.38
MDL number:
UNSPSC Code:
12352200
Assay:
≥98% (HPLC)
Form:
powder
$142.00
Please contact Customer Service for Availability
Quality Segment
assay
≥98% (HPLC)
form
powder
drug control
USDEA Schedule III
color
white to beige
solubility
DMSO: 2 mg/mL, clear
storage temp.
-10 to -25°C
Biochem/physiol Actions
Perampanel is an orally active, noncompetitive AMPA receptor antagonist that inhibits 2 μM AMPA-, but not NMDA-, induced Ca2+ in cultured rat cortical neurones (IC50 = 93 nM) and display therapeutic efficacy in murine models of epilepsy in vivo (audiogenic, MES-induced, and PTZ-induced seizures in mice ED50 = 0.47, 1.6, and 0.94 mg/kg p.o., respectively) and a rat amygdala-kindling model (1-10 mg/kg p.o.).
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This Item | |
|---|---|
| description ≥98% (HPLC) | description solid |
| form powder | form solid |
| assay ≥98% (HPLC) | assay - |
| drug control USDEA Schedule III | drug control - |
| Quality Level 100 | Quality Level 200 |
| storage temp. -10 to -25°C | storage temp. - |
| solubility DMSO: 2 mg/mL, clear | solubility H2O: 1 mg/mL (warm), 0.1 M HCl: 3.5 mg/mL, 1 M HCl: 50 mg/mL, 0.1 M NaOH: 4.3 mg/mL, DMSO: 4.3 mg/mL |
Signal Word
Warning
Hazard Codes
Precautionary Statements
Hazard Classifications
Acute Tox. 4 Oral - Aquatic Chronic 4
Storage Class
11 - Combustible Solids
Flash Point (°F)
Not applicable
Flash Point (°C)
Not applicable
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