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FRET Studies of Quinolone-Based Bitopic Ligands and Their Structural Analogues at the Muscarinic M

ACS chemical biology (2017-01-25)
Regina Messerer, Michael Kauk, Daniela Volpato, Maria Consuelo Alonso Canizal, Jessika Klöckner, Ulrike Zabel, Susanne Nuber, Carsten Hoffmann, Ulrike Holzgrabe
RESUMEN

Aiming to design partial agonists as well as allosteric modulators for the M

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Sigma-Aldrich
Acetylcholine bromide, ≥99%
Sigma-Aldrich
BQCA, ≥98% (HPLC)