SML0165

Fluorescent GABA-B receptor Antagonist (GB-633-AN) synthetic

• Empirische Formel (Hill-System): C₄₅H₅₃N₅O₆PCl₂F₂BS
• Molekulargewicht: 942.68
• NACRES: NA.77
• UNSPSC Code: 12352200
• Assay: ≥97% (HPLC)

Eigenschaften

• assay: ≥97% (HPLC)
• storage temp.: −20°C

Beschreibung

Biochem/physiol Actions

The SML0165 ligand was shown to antagonize the activity of the GABA-B agonist, GABA, in a recombinant CHO cell line expressing the human GABA-B1 and GABA-B2 receptors and a serum-responsive secreted placental alkaline phosphatase (SPAP) reporter gene.

Features and Benefits

This compound is featured on the GABAB Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Preparation Note

Dissolve 0.2 mg in 21.2 ul of DMSO to give a 10mM stock solution. Once reconstituted into DMSO the product, must be stored, preferably in smaller aliquots, at -20°C.

Sicherheitshinweise

• Lagerklasse: 13 - Non Combustible Solids
• Was ist los?: WGK 3
• Flammpunkt (°F): Not applicable
• Flammpunkt (°C): Not applicable