SML3090

EN4-2

≥98% (HPLC)

• Synonym(e): (E)-4-(but-2-enamidomethyl)-N-(2-(4-ethoxyphenoxy)phenyl)benzamide
• Empirische Formel (Hill-System): C₂₆H₂₆N₂O₄
• Molekulargewicht: 430.50
• NACRES: NA.77
• UNSPSC Code: 12352200
• Assay: ≥98% (HPLC)
• Form: powder

Eigenschaften

• Quality Segment: 100
• assay: ≥98% (HPLC)
• form: powder
• color: white to beige
• solubility: DMSO: 2 mg/mL, clear
• storage temp.: 2-8°C

Beschreibung

Biochem/physiol Actions

EN4-2 is a cell penetrant, potent and selective covalent c-MYC inhibitor that targets cysteine 171 located within a predicted intrinsically disordered region of MYC. EN4-2 inhibits MYC transcriptional activity, downregulates multiple MYC transcriptional targets, reduces MYC and MAX thermal stability, and impairs tumorigenesis.

cell penetrant, potent and selective covalent c-MYC inhibitor that targets cysteine 171

Sicherheitshinweise

• Lagerklasse: 11 - Combustible Solids
• Was ist los?: WGK 3
• Flammpunkt (°F): Not applicable
• Flammpunkt (°C): Not applicable