R1908

Remifentanil hydrochloride

≥97% (HPLC), Mu opioid receptor agonist, powder

• Synonym(s): 3-[methoxycarbonyl-4-[(1-oxopropyl)phenylamino]1-piperidine]propanoic acid methyl ester hydrochloride, GI-87084B, Remifentanyl, Ultiva
• Empirical Formula (Hill Notation): C₂₀H₂₈N₂O₅·HCl
• CAS Number: 132539-07-2
• Molecular Weight: 412.91
• PubChem Substance ID: 329824010
• UNSPSC Code: 12352200
• MDL number: MFCD00910882
• Assay: ≥97% (HPLC)
• Form: powder
• Storage condition: desiccated

Properties

• Product Name: Remifentanil hydrochloride, ≥97% (HPLC), powder
• Quality Segment: 100
• assay: ≥97% (HPLC)
• form: powder
• drug control: USDEA Schedule II; regulated under CDSA - not available from Sigma-Aldrich Canada; estupefaciente (Spain); Decreto Lei 15/93: Tabela IA (Portugal), kontrollierte Droge in Deutschland
• storage condition: desiccated
• color: white to off-white
• solubility: H₂O: ≥20 mg/mL
• storage temp.: 2-8°C
• SMILES string: O=C(CC)N(C1(CCN(CCC(OC)=O)CC1)C(OC)=O)C2=CC=CC=C2.[H]Cl
• InChI: 1S/C20H28N2O5.ClH/c1-4-17(23)22(16-8-6-5-7-9-16)20(19(25)27-3)11-14-21(15-12-20)13-10-18(24)26-2;/h5-9H,4,10-15H2,1-3H3;1H
• InChI key: WFBMIPUMYUHANP-UHFFFAOYSA-N
• Gene Information: human ... OPRM1(4988)

Description

Biochem/physiol Actions

Remifentanil hydrochloride is a mu opioid receptor agonist, anesthetic, and analgesic compound.

Remifentanil hydrochloride is a mu opioid receptor agonist, anesthetic, and analgesic compound. Remifentanil was developed as an ultra-short-acting mu opioid receptor agonist with improved pharmacodynamic properties.

Features and Benefits

This compound is featured on the Opioid Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Legal Information

German
Dieses Produkt fällt unter das Betäubungsmittelgesetz (BtMG). Für eine Bestellung dieses Produktes ist eine Erlaubnis nach § 3 BtMG zwingend erforderlich, es sei denn, es greift eine Ausnahme von der Erlaubnispflicht nach § 4 oder § 26 BtMG.

English
This product is subject to the German Narcotics Act. A permit under Section 3 of the German Narcotics Act is mandatory for ordering this product unless an exemption from the permit requirement under Section 4 or Section 26 of the German Narcotics Act applies.

Safety Information

• Pictograms: GHS08
• Signal Word: Warning
• Hazard Codes: H371
• Precautionary Statements: P260 - P264 - P270 - P308 + P311 - P405 - P501
• Hazard Classifications: STOT SE 2
• Target Organs: Respiratory system
• Storage Class: 11 - Combustible Solids
• WGK: WGK 1
• Flash Point (°F): Not applicable
• Flash Point (°C): Not applicable