SML1587

Perlapine

≥98% (HPLC)

• Synonym(e): 6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepine, 6-(4-Methyl-1-piperazinyl)morphanthridine, CID 16106
• Empirische Formel (Hill-System): C₁₉H₂₁N₃
• CAS-Nummer: 1977-11-3
• Molekulargewicht: 291.39
• UNSPSC Code: 12352200
• PubChem Substance ID: 329825973
• NACRES: NA.77
• Assay: ≥98% (HPLC)
• Form: powder

Eigenschaften

• assay: ≥98% (HPLC)
• form: powder
• color: white to beige
• solubility: DMSO: 10 mg/mL, clear
• storage temp.: room temp
• SMILES string: CC(C)(C1=CC=C(CN2CCN(C(C3=CC=C(Cl)C=C3)C4=CC=CC=C4)CC2)C=C1)C.[H]Cl.[H]Cl
• InChI: 1S/C28H33ClN2.2ClH/c1-28(2,3)25-13-9-22(10-14-25)21-30-17-19-31(20-18-30)27(23-7-5-4-6-8-23)24-11-15-26(29)16-12-24;;/h4-16,27H,17-21H2,1-3H3;2*1H
• InChI key: SDBHDSZKNVDKNU-UHFFFAOYSA-N
• Gene Information: human ... HRH1(3269)

Beschreibung

Biochem/physiol Actions

Perlapine is a potent and selective agonist of hM3Dq DREADD (Designer Receptors Exclusively Activated by Designer Drugs), which does not activate the native human M3 receptor. Perlapine is a neuroleptic agent that exhibits sedative and sleep-promoting properties.

Potent and selective agonist of hM3Dq DREADD

Sicherheitshinweise

• Piktogramme: GHS07
• Signalwort: Warning
• Gefahrencodes: H302,H315,H319,H413
• Sicherheitshinweise: P264 - P270 - P273 - P301 + P312 - P302 + P352 - P305 + P351 + P338
• Hazard Classifications: Acute Tox. 4 Oral - Aquatic Chronic 4 - Eye Irrit. 2 - Skin Irrit. 2
• Lagerklasse: 11 - Combustible Solids
• WGK: WGK 3
• Flammpunkt (°F): Not applicable
• Flammpunkt (°C): Not applicable