SML0168

Fluorescent Histamine H3/H4 receptor Antagonist (H3-633-AN) synthetic

• Fórmula empírica (notación de Hill): C₄₄H₄₈BF₂N₈O₃S₂
• Peso molecular: 849.84
• NACRES: NA.77
• UNSPSC Code: 12352200

Propiedades

• storage temp.: −20°C
• Quality Level: 200

Descripción

Biochem/physiol Actions

The SML0168 ligand was shown to antagonize the activity of the histamine agonist, histamine, in two separate recombinant CHO cell lines expressing either the human H2 or H3-receptor and a cyclic-AMP responsive secreted placental alkaline phosphatase (SPAP) reporter gene.

Features and Benefits

This compound is featured on the Histamine Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Preparation Note

Dissolve 0.2 mg in 23.5 ul of DMSO to give a 10mM stock solution. Once reconstituted into DMSO the product, must be stored, preferably in smaller aliquots, at -20°C.

Información de seguridad

• Clase de almacenamiento: 11 - Combustible Solids
• wgk: WGK 3
• flash_point_f: Not applicable
• flash_point_c: Not applicable