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Merck

ESR1

estrogen receptor 1

Sinónimos:
ER, ESR, ESRA, ESTRR, Era, NR3A1
Especie:
ID UniProtKB:
ID del gen:
  • Human(2099) Summary: This gene encodes an estrogen receptor, a ligand-activated transcription factor composed of several domains important for hormone binding, DNA binding, and activation of transcription. The protein localizes to the nucleus where it may form a homodimer or a heterodimer with estrogen receptor 2. Estrogen and its receptors are essential for sexual development and reproductive function, but also play a role in other tissues such as bone. Estrogen receptors are also involved in pathological processes including breast cancer, endometrial cancer, and osteoporosis. Alternative splicing results in several transcript variants, which differ in their 5' UTRs and use different promoters. [provided by RefSeq, Jul 2008]
  • Mouse(13982) estrogen receptor 1 (alpha)
  • Rat(24890) estrogen receptor 1
  • domestic cat(552888) estrogen receptor 1
  • dog(403640) estrogen receptor 1
  • chicken(396099) estrogen receptor 1
  • Thale Cress(837856) ethylene-responsive transcription factor ESR1
  • Horse(791249) estrogen receptor 1
  • Zebrafish(259252) estrogen receptor 1
  • cow(407238) estrogen receptor 1
  • Goat(100860768) estrogen receptor 1
  • sheep(443228) estrogen receptor 1
  • domestic guinea pig(100713276) estrogen receptor 1

Custom & Knockdown Gene Products

Small Molecule - Activator

Número de producto
Descripción
Especie
4-Phenylazophenol, 98%,
Especie
human
βDinucleótido de β-nicotinamida y adenina sodium salt, ,
Especie
human
βDinucleótido de β-nicotinamida y adenina hydrate, ≥96.5% (HPLC), ≥96.5% (spectrophotometric assay), from yeast,
Especie
human
trans-Stilbene, 96%,
Especie
human, rat
βDinucleótido de β-nicotinamida y adenina hydrate, ≥95% (HPLC),
Especie
human

Small Molecule - Agonist

Número de producto
Descripción
Especie
17α-etinilestradiol, Pharmaceutical Secondary Standard; Certified Reference Material,
Especie
human
Estrone, Pharmaceutical Secondary Standard; Certified Reference Material,
Especie
human
β-Estradiol, Pharmaceutical Secondary Standard; Certified Reference Material,
Especie
human
β-Estradiol, United States Pharmacopeia (USP) Reference Standard,
Especie
human
Etinil estradiol, United States Pharmacopeia (USP) Reference Standard,
Especie
human

Small Molecule - Allosteric Modulator

Número de producto
Descripción
Especie
Toremifene citrate salt, ≥98% (HPLC),
Especie
human

Small Molecule - Antagonist

Número de producto
Descripción
Especie
Dibutyl phthalate, 99%,
Especie
mouse
Benzyl butyl phthalate, 98%,
Especie
mouse
Zearalenone, fungal mycotoxin,
Especie
mouse
4-tert-Octylphenol, 97%,
Especie
mouse
2-tert-Butylphenol, 99%,
Especie
mouse

Antibodies

Número de producto
Descripción
Reactividad de especies
Aplicación
Anti-ESR1 antibody produced in rabbit, Prestige Antibodies® Powered by Atlas Antibodies, affinity isolated antibody, buffered aqueous glycerol solution,
Reactividad de especies
human
Aplicación
immunofluorescence
immunohistochemistry

western blot
Anti-Estrogen Receptor-α antibody produced in rabbit, affinity isolated antibody,
Reactividad de especies
human
Aplicación
ELISA
immunohistochemistry

western blot
Anti-ESR1 antibody produced in rabbit, Ab2, Prestige Antibodies® Powered by Atlas Antibodies, affinity isolated antibody, buffered aqueous glycerol solution,
Reactividad de especies
human
Aplicación
ChIP
immunohistochemistry

western blot
Monoclonal Anti-ESR1 antibody produced in mouse, Prestige Antibodies® Powered by Atlas Antibodies, clone CL1196, purified immunoglobulin, buffered aqueous glycerol solution,
Reactividad de especies
human
Aplicación
immunofluorescence
immunohistochemistry

western blot
Anti-Estrogen Receptor-α antibody produced in rabbit, affinity isolated antibody,
Reactividad de especies
human, mouse, rat
Aplicación
ELISA
immunohistochemistry

western blot

Small Molecule - Ligand

Número de producto
Descripción
Especie
Progesterone, VETRANAL®, analytical standard,
Especie
human
Diethylstilbestrol, mixture of cis and trans, 97%,
Especie
human, mouse, rat
Progesterone, powder, BioReagent, suitable for cell culture,
Especie
mouse, human, rat
Progesterone, ≥99%,
Especie
mouse, human, rat
Progesterone, meets USP testing specifications,
Especie
mouse, human, rat

Small Molecule - Mixed Agonist/Antagonist

Número de producto
Descripción
Especie
α-Estradiol, powder, ≥98% (TLC),
Especie
human, rat
Diethylstilbestrol, mixture of cis and trans, 97%,
Especie
human, mouse, rat
Medroxyprogesterone 17-acetate, ≥97% (HPLC),
Especie
human, rat
β-Estradiol, meets USP testing specifications,
Especie
human, mouse, rat
β-Estradiol, BioReagent, powder, suitable for cell culture,
Especie
human, mouse, rat

Proteins

Número de producto
Descripción
Especie
Estrogen Receptor-α human, ≥80% (SDS-PAGE), recombinant, expressed in baculovirus infected insect cells, buffered aqueous glycerol solution,
Especie
human

esiRNA

Número de producto
Descripción
Especie
MISSION® esiRNA, targeting human ESR1,
Especie
human