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E5156

Epinastine hydrochloride

≥98% (HPLC), H1 histamine receptor antagonist, solid

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Synonym(s):

9,13b-Dihydro-1H-dibenz[cf]imidazo[1,5-a]azepine hydrochloride, WAL-801Cl

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10 mg

Available to ship TODAYfromMILWAUKEE

$185.00
50 mg

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$709.00

About This Item

Empirical Formula (Hill Notation):
C16H15N3 · HCl
CAS Number:
108929-04-0
Molecular Weight:
285.77
UNSPSC Code:
12352200
PubChem Substance ID:
24894608
NACRES:
NA.77
MDL number:
MFCD00933434
Assay:
≥98% (HPLC)
Form:
solid
Storage condition:
desiccated

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Product Name

Epinastine hydrochloride, ≥98% (HPLC), solid

Quality Segment

assay

≥98% (HPLC)

form

solid

storage condition

desiccated

color

white

solubility

H2O: 38 mg/mL

originator

Boehringer Ingelheim

storage temp.

2-8°C

SMILES string

Cl[H].NC1=NCC2N1c3ccccc3Cc4ccccc24

InChI

1S/C16H15N3.ClH/c17-16-18-10-15-13-7-3-1-5-11(13)9-12-6-2-4-8-14(12)19(15)16;/h1-8,15H,9-10H2,(H2,17,18);1H

InChI key

VKXSGUIOOQPGAF-UHFFFAOYSA-N

Gene Information

human ... HRH1(3269)

General description

Epinastine has antihistamine functions. In mast cells, it may modulate cytokine and chemokine production. In dendritic cells, it controls T helper cell mediated immune response. Epinastine hydrochloride does not traverse the brain barrier. Oral dosage of epinastine hydrochloride is prescribed for children with sleep-disordered breathing (SDB) and nasal inflammation. Ophthalmic solution of epinastine is effective for allergic conjunctivitis.

Biochem/physiol Actions

Epinastine hydrochloride is a non-sedating H1 histamine receptor antagonist.

Features and Benefits

This compound is featured on the Histamine Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
This compound was developed by Boehringer Ingelheim. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

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This Item
1236889Y0001139Y0002208
Epinastine hydrochloride ≥98% (HPLC), solid

Sigma-Aldrich

E5156

Epinastine hydrochloride

Epinastine hydrochloride United States Pharmacopeia (USP) Reference Standard

USP

1236889

Epinastine hydrochloride

Epinastine hydrochloride European Pharmacopoeia (EP) Reference Standard

Y0001139

Epinastine hydrochloride

Epinastine for system suitability A European Pharmacopoeia (EP) Reference Standard

Y0002208

Epinastine for system suitability A

description

≥98% (HPLC), solid

description

United States Pharmacopeia (USP) Reference Standard

description

European Pharmacopoeia (EP) Reference Standard

description

European Pharmacopoeia (EP) Reference Standard

assay

≥98% (HPLC)

assay

-

assay

-

assay

-

form

solid

form

-

form

-

form

-

Quality Level

100

Quality Level

-

Quality Level

-

Quality Level

-

storage temp.

2-8°C

storage temp.

-

storage temp.

2-8°C

storage temp.

2-8°C

storage condition

desiccated

storage condition

-

storage condition

-

storage condition

-

solubility

H2O: 38 mg/mL

solubility

-

solubility

-

solubility

-

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Pictograms

Skull and crossbones
GHS06

Signal Word

Danger

Hazard Codes

H301

Hazard Classifications

Acute Tox. 3 Oral

Storage Class

6.1C - Combustible acute toxic Cat.3 / toxic compounds or compounds which causing chronic effects

WGK

WGK 3

Flash Point (°F)

Not applicable

Flash Point (°C)

Not applicable

PPE (personal protective equipment)

Eyeshields, Faceshields, Gloves, type P2 (EN 143) respirator cartridges

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Certificates of Analysis (COA)

Lot/Batch Number
0000377982
0000015706
0000015707
0000149323
0000050089

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