P0547
Pentamidine isethionate salt
NMDA glutamate receptor antagonist, powder
Synonym(s):
1,5-Bis(p-amidinophenoxy)pentane bis(2-hydroxyethanesulfonate salt), 4,4′-(Pentamethylenedioxy)dibenzamidine bis(2-hydroxyethanesulfonate)
Select a Size
| Size/SKU | Availability | Price |
|---|---|---|
100 mg | Check Cart for Availability | $52.30 |
25 mg | Check Cart for Availability | $50.60 |
250 mg | Check Cart for Availability | $94.80 |
1 g | Check Cart for Availability | $185.00 |
About This Item
Product Name
Pentamidine isethionate salt, powder
form
powder
Quality Segment
mp
188-194 °C (lit.)
antibiotic activity spectrum
fungi
mode of action
enzyme | inhibits
originator
Celgene
storage temp.
−20°C
SMILES string
OCCS(O)(=O)=O.OCCS(O)(=O)=O.NC(=N)c1ccc(OCCCCCOc2ccc(cc2)C(N)=N)cc1
InChI
1S/C19H24N4O2.2C2H6O4S/c20-18(21)14-4-8-16(9-5-14)24-12-2-1-3-13-25-17-10-6-15(7-11-17)19(22)23;2*3-1-2-7(4,5)6/h4-11H,1-3,12-13H2,(H3,20,21)(H3,22,23);2*3H,1-2H2,(H,4,5,6)
InChI key
YBVNFKZSMZGRAD-UHFFFAOYSA-N
Gene Information
Application
- as a positive control for anti-leishmanial, anti-plasmodial and cytotoxic assays
- as a prototypical compound to analyse the inhibitor effect on human ether-a-go-go-related gene (HERG) K+ channel trafficking
- as an anti-leishmanial agent in promastigotes
Biochem/physiol Actions
Features and Benefits
1 of 1
This Item | |||
|---|---|---|---|
| description powder | description United States Pharmacopeia (USP) Reference Standard | description European Pharmacopoeia (EP) Reference Standard | description ≥98% (HPLC) |
| form powder | form - | form - | form powder |
| Quality Level 100 | Quality Level - | Quality Level - | Quality Level 100 |
| storage temp. −20°C | storage temp. - | storage temp. 2-8°C | storage temp. room temp |
| originator Celgene | originator - | originator - | originator - |
| mp 188-194 °C (lit.) | mp 188-194 °C (lit.) | mp 188-194 °C (lit.) | mp - |
| Gene Information human ... GRIN1(2902), GRIN2A(2903), GRIN2B(2904), GRIN2C(2905), GRIN2D(2906), GRINA(2907), NOS1(4842), NOS2(4843), NOS2B(201288), NOS2C(645740), NOS3(4846) | Gene Information - | Gene Information - | Gene Information - |
Signal Word
Warning
Hazard Codes
Precautionary Statements
Hazard Classifications
Eye Irrit. 2 - Skin Irrit. 2 - Skin Sens. 1 - STOT SE 3
Target Organs
Respiratory system
Storage Class
11 - Combustible Solids
WGK
WGK 3
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