SML0979
Bantag-1 trifluoroacetate salt
≥95% (HPLC)
Synonym(s):
Boc-Phe-His-4-amino-5-cyclohexyl-2,4,5-trideoxypentonyl-Leu-(3-dimethylamino) benzylamide N-methylammonium trifluoroacetate salt
Sign In to View Organizational & Contract Pricing.
Select a Size
Change View
| Pack Size | SKU | Availability | Price |
|---|---|---|---|
| 1 mg | Available to ship TODAYfromMILWAUKEE | $385.00 |
About This Item
Empirical Formula (Hill Notation):
C48H73N8O7 · xC2HF3O2
Molecular Weight:
874.14 (free base basis)
NACRES:
NA.77
UNSPSC Code:
12352200
$385.00
Available to ship TODAYDetails
General description
Bantag-1 is a peptide-antagonist. It is soluble in aqueous solutions.[1]
Biochem/physiol Actions
Bantag-1 is a very specific, high affinity antagonist of the orphan GPCR Bombesin receptor subtype-3 (BRS-3).
Bantag-1 is a very specific, high affinity antagonist of the orphan GPCR Bombesin receptor subtype-3 (BRS-3). The binding affinity of Bantag-1 in BRS-3 expressing cells is 1.3 nM.
1 of 1
This Item | |||
|---|---|---|---|
| form powder | form powder | form powder | form lyophilized powder |
| assay ≥95% (HPLC) | assay ≥95% (HPLC) | assay ≥95% (HPLC) | assay >98% (HPLC) |
| Quality Level 100 | Quality Level 100 | Quality Level 100 | Quality Level 100 |
| storage temp. −20°C | storage temp. −20°C | storage temp. −20°C | storage temp. −20°C |
| color white to off-white | color white to off-white | color colorless to pale yellow | color white to tan |
Storage Class
11 - Combustible Solids
wgk
WGK 3
flash_point_f
Not applicable
flash_point_c
Not applicable
Choose from one of the most recent versions:
Already Own This Product?
Find documentation for the products that you have recently purchased in the Document Library.
Molecular basis for high affinity and selectivity of peptide antagonist, Bantag-1, for the orphan BB3 receptor.
Nakamura T, et al.
Biochemical Pharmacology, 115, 64-76 (2016)
Xiao-Ming Guan et al.
Cell metabolism, 11(2), 101-112 (2010-01-26)
Bombesin receptor subtype 3 (BRS-3) is a G protein coupled receptor whose natural ligand is unknown. We developed potent, selective agonist (Bag-1, Bag-2) and antagonist (Bantag-1) ligands to explore BRS-3 function. BRS-3-binding sites were identified in the hypothalamus, caudal brainstem
Global Trade Item Number
| SKU | GTIN |
|---|---|
| SML0979-1MG | 04061826745816 |