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| Size/SKU | Availability | Price |
|---|---|---|
5 mg | Check Cart for Availability | $70.60 |
25 mg | Check Cart for Availability | $288.00 |
About This Item
Empirical Formula (Hill Notation):
C72H95ClN14O14 · xC2H4O2
CAS Number:
Molecular Weight:
1416.06 (free base basis)
NACRES:
NA.77
UNSPSC Code:
12352200
Assay:
≥97% (HPLC)
Form:
film or powder
Biochem/physiol Actions
Abarelix (PPI-149) is a gonadotropin releasing hormone (GnRH)/luteinizing hormone releasing hormone (LHRH) receptor (GnRHR, LHRHR) antagonist with low histamine release induction propensity (EC50 = 100 μg/mL; rat mast cells). Abarelix exhibits good in vivo efficacy via iv. or sc. in suppressing LH levels in castrated male rats (plasma LH = 12/1.2/0.9/1.2 ng/mL 6 hrs post 0/12.5/50/200 μg/kg in 5% mannitol sc.) and in lowering testosterone among intact male rats (plasma testosterone = 1.64/0.29 ng/mL 6 hrs post 0/3 μg/kg sc.).
Gonadotropin releasing hormone (GnRH)/ luteinizing hormone releasing hormone (LHRH) receptor (GnRHR, LHRHR) antagonist.
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This Item | |||
|---|---|---|---|
| description - | description ≥98% (HPLC) | description ≥95% (HPLC) | description ≥98% (HPLC) |
| assay ≥97% (HPLC) | assay ≥98% (HPLC) | assay ≥95% (HPLC) | assay ≥98% (HPLC) |
| form film or powder | form powder | form lyophilized powder | form powder |
| Quality Level 100 | Quality Level 100 | Quality Level 100 | Quality Level 100 |
| storage temp. −20°C | storage temp. −20°C | storage temp. −20°C | storage temp. −20°C |
| color white to beige | color white to beige | color white | color white to off-white |
signalword
Warning
hcodes
Hazard Classifications
Repr. 2
Storage Class
11 - Combustible Solids
wgk
WGK 3
flash_point_f
Not applicable
flash_point_c
Not applicable
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