G5668
GW1929 hydrate
>98% (HPLC), solid
Synonym(s):
N-(2-Benzoylphenyl)-O-[2-(methyl-2-pyridinylamino)ethyl]-L-tyrosine hydrate
Select a Size
| Size/SKU | Availability | Price |
|---|---|---|
5 mg | Check Cart for Availability | $252.00 $214.20 |
About This Item
$214.20
List Price$252.00Save 15%Quality Segment
assay
>98% (HPLC)
form
solid
solubility
DMSO: 20 mg/mL
originator
GlaxoSmithKline
SMILES string
[H]O[H].CN(CCOc1ccc(C[C@H](Nc2ccccc2C(=O)c3ccccc3)C(O)=O)cc1)c4ccccn4
InChI
1S/C30H29N3O4.H2O/c1-33(28-13-7-8-18-31-28)19-20-37-24-16-14-22(15-17-24)21-27(30(35)36)32-26-12-6-5-11-25(26)29(34)23-9-3-2-4-10-23;/h2-18,27,32H,19-21H2,1H3,(H,35,36);1H2/t27-;/m0./s1
InChI key
XSITZVFUXCLFMK-YCBFMBTMSA-N
Gene Information
human ... PPARG(5468)
Application
- to study its effects on plant homeodomain finger protein 16 (Phf16) and patatin-like phospholipase domain containing 3 (Pnpla3) expression involved in adipogenesis
- to study its effects on complement component 3 (C3) gene expression in human hepatoma cells
- to activate PPARγ in human breast cancer cells
Biochem/physiol Actions
Features and Benefits
Legal Information
1 of 1
This Item | |
|---|---|
| description >98% (HPLC), solid | description A potent, tyrosine-based peroxisome proliferator-activated receptor γ (PPARγ) agonist (EC50 = 13 nM for murine receptor and 6.2 nM for human receptor in cell-based transactivation assays). |
| form solid | form crystalline solid |
| assay >98% (HPLC) | assay - |
| Quality Level 100 | Quality Level 100 |
| solubility DMSO: 20 mg/mL | solubility DMSO: 100 mg/mL |
| originator GlaxoSmithKline | originator - |
| Gene Information human ... PPARG(5468) | Gene Information - |
Storage Class
11 - Combustible Solids
WGK
WGK 3
Flash Point (°F)
Not applicable
Flash Point (°C)
Not applicable
PPE (personal protective equipment)
Eyeshields, Gloves, type N95 (US)
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