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SML1504

Tegaserod maleate

≥98% (HPLC)

Synonym(s):

2-[(5-Methoxy-1H-indol-3-yl)methylene]-N-pentyl-hydrazinecarboximidamide maleate

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Size/SKUAvailabilityPrice
10 mg
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$157.00
50 mg
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$639.00

About This Item

Empirical Formula (Hill Notation):
C16H23N5O · C4H4O4
CAS Number:
Molecular Weight:
417.46
NACRES:
NA.77
PubChem Substance ID:
UNSPSC Code:
12352200
MDL number:
Assay:
≥98% (HPLC)
Form:
powder

$157.00

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Quality Segment

assay

≥98% (HPLC)

form

powder

color

white to beige

solubility

DMSO: 20 mg/mL, clear

storage temp.

2-8°C

SMILES string

N=C(NCCCCC)N/N=C/C1=CNC2=C1C=C(OC)C=C2.OC(/C=C\C(O)=O)=O

InChI

1S/C16H23N5O.C4H4O4/c1-3-4-5-8-18-16(17)21-20-11-12-10-19-15-7-6-13(22-2)9-14(12)15;5-3(6)1-2-4(7)8/h6-7,9-11,19H,3-5,8H2,1-2H3,(H3,17,18,21);1-2H,(H,5,6)(H,7,8)/b20-11+;2-1-

InChI key

CPDDZSSEAVLMRY-FEQFWAPWSA-N

Gene Information

human ... HTR4(3360)

Application

Tegaserod maleate has been used to study its cytotoxic effects on human astrocytes and to study its effects as an anti-glioblastoma agent.

Biochem/physiol Actions

Tegaserod is a potent full agonist at serotonin 5-HT4 receptors with an EC50 of 7 nM.
Tegaserod is a serotonin 5-HT4 agonist.
It stimulates neurotransmitter release from enteric nerves and regularizes gastrointestinal function. Tegaserod has been used to treat irritable bowel syndrome associated with constipation and chronic constipation.

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This Item
SML0204SML1887SML1679
form

powder

form

powder

form

powder

form

powder

assay

≥98% (HPLC)

assay

≥98% (HPLC)

assay

≥98% (HPLC)

assay

≥98% (HPLC)

Quality Level

100

Quality Level

100

Quality Level

100

Quality Level

100

storage temp.

2-8°C

storage temp.

2-8°C

storage temp.

2-8°C

storage temp.

−20°C

solubility

DMSO: 20 mg/mL, clear

solubility

DMSO: ≥10 mg/mL at 60 °C

solubility

DMSO: 10 mg/mL, clear

solubility

DMSO: 10 mg/mL, clear

color

white to beige

color

white to tan

color

white to beige

color

white to beige


Storage Class

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable



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