The storage temperature and solution stability after reconstitution in DMSO have not been tested. It is recommended to make the solution fresh upon usage.
P1793
匹莫齐特
≥98% (TLC), powder, D₂ dopamine receptor antagonist
同義詞:
1-[1-[4,4-双（4-氟苯基）丁基]-4-哌啶基]-1,3-二氢-2H-苯并咪唑-2-酮
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選擇尺寸
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經驗公式（希爾表示法）:
C28H29F2N3O
CAS 編號:
分子量：:
461.55
EC號碼:
MDL號碼:
分類程式碼代碼:
12352200
PubChem物質ID:
NACRES:
NA.77
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產品名稱
匹莫齐特,
形狀
powder
品質等級
溶解度
DMSO: 18 mg/mL(lit.)
chloroform: 5 mg/mL
H2O: insoluble(lit.)
起源
Teva
儲存溫度
2-8°C
SMILES 字串
Fc1ccc(cc1)C(CCCN2CCC(CC2)N3C(=O)Nc4ccccc34)c5ccc(F)cc5
InChI
1S/C28H29F2N3O/c29-22-11-7-20(8-12-22)25(21-9-13-23(30)14-10-21)4-3-17-32-18-15-24(16-19-32)33-27-6-2-1-5-26(27)31-28(33)34/h1-2,5-14,24-25H,3-4,15-19H2,(H,31,34)
InChI 密鑰
YVUQSNJEYSNKRX-UHFFFAOYSA-N
基因資訊
human ... ABCB1(5243), CACNA1G(8913), CYP3A4(1576), DRD1(1812), DRD2(1813), DRD3(1814), DRD4(1815), DRD5(1816), HTR2A(3356), HTR7(3363), KCNH1(3756), KCNH2(3757), OPRD1(4985)
mouse ... Abcb1a(18671), Abcb1b(18669)
rat ... Scnn1g(24768)
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相關類別
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本產品 | P1750000 | BP682 | P-168 |
|---|---|---|---|
| form powder | form - | form solid | form - |
| Quality Level 200 | Quality Level - | Quality Level - | Quality Level 300 |
| storage temp. 2-8°C | storage temp. 2-8°C | storage temp. 2-8°C | storage temp. -10 to -25°C |
| solubility DMSO: 18 mg/mL(lit.), H2O: insoluble(lit.), chloroform: 5 mg/mL | solubility - | solubility - | solubility - |
| originator Teva | originator - | originator - | originator - |
| Gene Information human ... ABCB1(5243), CACNA1G(8913), CYP3A4(1576), DRD1(1812), DRD2(1813), DRD3(1814), DRD4(1815), DRD5(1816), HTR2A(3356), HTR7(3363), KCNH1(3756), KCNH2(3757), OPRD1(4985) | Gene Information human ... DRD1(1812), DRD2(1813), DRD3(1814), DRD4(1815), DRD5(1816), HTR2A(3356) | Gene Information human ... DRD1(1812), DRD2(1813), DRD3(1814), DRD4(1815), DRD5(1816), HTR2A(3356) | Gene Information - |
生化／生理作用
D 2 多巴胺受体拮抗剂；与克隆的 5-HT 7 受体高亲和力结合；Ca 2 + 通道拮抗剂；抗精神病药
特點和優勢
该化合物在受体分类和信号转导手册的环核苷酸门控（CNG）和超极化激活的环核苷酸门控（HCN）通道页面上有详细描述。想要浏览手册的其他页面， 请单击此处。
该化合物是环核苷酸研究的特色产品。 点击此处 ，发现更多特色环核苷酸产品。。在 sigma.com/discover-bsm了解更多关于其他研究领域的生物活性小分子。
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文章
Cyclic nucleotides like cAMP modulate cell function via PKA activation and ion channels.
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When dissolved in DMSO, at what temperature should I store the solution?
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