S106

SR-95531

≥98% (HPLC), powder

• Synonym(s): 2-(3-Carboxypropyl)-3-amino-6-(4 methoxyphenyl)pyridazinium bromide, Gabazine
• Empirical Formula (Hill Notation): C₁₅H₁₈BrN₃O₃
• CAS Number: 104104-50-9
• Molecular Weight: 368.23
• MDL number: MFCD00055135
• UNSPSC Code: 12352200
• PubChem Substance ID: 24278819
• NACRES: NA.77

Properties

• Quality Level: 100
• assay: ≥98% (HPLC)
• form: powder
• color: white
• solubility: H₂O: >10 mg/mL
• SMILES string: [Br-].COc1ccc(cc1)-c2ccc(N)[n+](CCCC(O)=O)n2
• InChI: 1S/C15H17N3O3.BrH/c1-21-12-6-4-11(5-7-12)13-8-9-14(16)18(17-13)10-2-3-15(19)20;/h4-9,16H,2-3,10H2,1H3,(H,19,20);1H
• InChI key: GFZHNFOGCMEYTA-UHFFFAOYSA-N
• Gene Information: human ... GABRA1(2554), GABRA2(2555), GABRA3(2556), GABRA4(2557), GABRA5(2558), GABRA6(2559), GABRB1(2560), GABRB2(2561), GABRB3(2562) ; rat ... Gabra2(29706)

Description

Biochem/physiol Actions

SR-95531 is a specific GABA_A receptor antagonist that does not affect GABA-transaminase or glutamate-decarboxylase activities.

Features and Benefits

This compound is a featured product for Neuroscience research. Click here to discover more featured Neuroscience products. Learn more about bioactive small molecules for other areas of research at sigma.com/discover-bsm.

This compound is featured on the GABAA Receptors and GABAC Receptors pages of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Safety Information

• Storage Class: 11 - Combustible Solids
• wgk_germany: WGK 3
• flash_point_f: Not applicable
• flash_point_c: Not applicable
• ppe: Eyeshields, Gloves, type N95 (US)