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Merck

CHRM2

cholinergic receptor, muscarinic 2

Sinônimos:
HM2
Espécies:
ID UniProtKB:
ID do gene:
  • Human(1129) Summary: The muscarinic cholinergic receptors belong to a larger family of G protein-coupled receptors. The functional diversity of these receptors is defined by the binding of acetylcholine to these receptors and includes cellular responses such as adenylate cyclase inhibition, phosphoinositide degeneration, and potassium channel mediation. Muscarinic receptors influence many effects of acetylcholine in the central and peripheral nervous system. The muscarinic cholinergic receptor 2 is involved in mediation of bradycardia and a decrease in cardiac contractility. Multiple alternatively spliced transcript variants have been described for this gene. [provided by RefSeq, Jul 2008]
  • Mouse(243764) cholinergic receptor, muscarinic 2, cardiac
  • Rat(81645) cholinergic receptor, muscarinic 2
  • Domestic Rabbit(100342878) cholinergic receptor, muscarinic 2
  • naked mole-rat(101714286) cholinergic receptor, muscarinic 2
  • chicken(418126) cholinergic receptor, muscarinic 2
  • domestic guinea pig(100715343) cholinergic receptor, muscarinic 2
  • dog(403858) cholinergic receptor, muscarinic 2
  • cow(522170) cholinergic receptor, muscarinic 2
  • domestic cat(101099790) cholinergic receptor, muscarinic 2
  • sheep(101102897) cholinergic receptor, muscarinic 2
  • sheep(100628317) cholinergic receptor, muscarinic 2

Custom & Knockdown Gene Products

Small Molecule - Agonist

Número do produto
Descrição
Espécies
Pilocarpina, ≥99% (titration), powder,
Espécies
human
Acetyl-β-methylcholine chloride, ≥98% (TLC), powder,
Espécies
human
Pilocarpine nitrate salt, ≥98% (HPLC),
Espécies
human
Oxotremorine M, solid,
Espécies
human
(±)-Muscarine chloride hydrate, ≥98% (HPLC),
Espécies
human

Small Molecule - Antagonist

Número do produto
Descrição
Espécies
Methoctramine hydrate, ≥97% (NMR), solid,
Espécies
human
Darifenacin hydrobromide, ≥98% (HPLC),
Espécies
human
Oxybutynin hydrochloride, British Pharmacopoeia (BP) Reference Standard,
Espécies
human
Atropine Sulfate, Pharmaceutical Secondary Standard; Certified Reference Material,
Espécies
human
Propantheline Bromide, Pharmaceutical Secondary Standard; Certified Reference Material,
Espécies
human

Antibodies

Número do produto
Descrição
Reatividade de espécies
Aplicação
Anti-Muscarinic Acetylcholine Receptor m2 Antibody, clone M2-2-B3, clone M2-2-B3, Chemicon®, from rat,
Reatividade de espécies
human, mammals, monkey, rat
Aplicação
immunocytochemistry
immunohistochemistry

immunoprecipitation (IP)
Anti-Muscarinic Acetylcholine Receptor M2 Antibody, Chemicon®, from rabbit,
Reatividade de espécies
human
Aplicação
immunohistochemistry
Monoclonal Anti-CHRM2 antibody produced in mouse, clone 4B5, purified immunoglobulin, buffered aqueous solution,
Reatividade de espécies
human
Aplicação
ELISA
western blot
Anti-Muscarinic AChR M2 (ACM2) Antibody, clone 3T5W8, Rabbit Monoclonal, ,
Reatividade de espécies
human, rat
Aplicação
immunohistochemistry
western blot

Small Molecule - Inhibitor

Número do produto
Descrição
Espécies
Harmaline, ≥95%,
Espécies
human, rat

Small Molecule - Ligand

Número do produto
Descrição
Espécies
Aminobenztropine, solid,
Espécies
human

Proteins

Número do produto
Descrição
Espécies
ChemiSCREEN Membrane Preparation Recombinant Human M2 Muscarinic Acetylcholine Receptor, Human M2 GPCR membrane prepation for Radioligand binding Assays.,
Espécies
human

esiRNA

Número do produto
Descrição
Espécies
MISSION® esiRNA, targeting human CHRM2,
Espécies
human